JP2010090130A5 - - Google Patents

Download PDF

Info

Publication number
JP2010090130A5
JP2010090130A5 JP2009263603A JP2009263603A JP2010090130A5 JP 2010090130 A5 JP2010090130 A5 JP 2010090130A5 JP 2009263603 A JP2009263603 A JP 2009263603A JP 2009263603 A JP2009263603 A JP 2009263603A JP 2010090130 A5 JP2010090130 A5 JP 2010090130A5
Authority
JP
Japan
Prior art keywords
cys
arg
phe
seq
trp
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009263603A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010090130A (ja
JP5889513B2 (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2010090130A publication Critical patent/JP2010090130A/ja
Publication of JP2010090130A5 publication Critical patent/JP2010090130A5/ja
Application granted granted Critical
Publication of JP5889513B2 publication Critical patent/JP5889513B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009263603A 2005-07-08 2009-11-19 メラノコルチン受容体リガンド Active JP5889513B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US69777905P 2005-07-08 2005-07-08
US60/697,779 2005-07-08
US74885005P 2005-12-09 2005-12-09
US60/748,850 2005-12-09

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2008520417A Division JP4734411B2 (ja) 2005-07-08 2006-07-10 メラノコルチン受容体リガンド

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2013165312A Division JP2013253090A (ja) 2005-07-08 2013-08-08 メラノコルチン受容体リガンド
JP2015140154A Division JP5965520B2 (ja) 2005-07-08 2015-07-14 メラノコルチン受容体リガンド

Publications (3)

Publication Number Publication Date
JP2010090130A JP2010090130A (ja) 2010-04-22
JP2010090130A5 true JP2010090130A5 (OSRAM) 2011-06-23
JP5889513B2 JP5889513B2 (ja) 2016-03-22

Family

ID=37637790

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2008520417A Active JP4734411B2 (ja) 2005-07-08 2006-07-10 メラノコルチン受容体リガンド
JP2009263603A Active JP5889513B2 (ja) 2005-07-08 2009-11-19 メラノコルチン受容体リガンド
JP2013165312A Pending JP2013253090A (ja) 2005-07-08 2013-08-08 メラノコルチン受容体リガンド
JP2015140154A Active JP5965520B2 (ja) 2005-07-08 2015-07-14 メラノコルチン受容体リガンド

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2008520417A Active JP4734411B2 (ja) 2005-07-08 2006-07-10 メラノコルチン受容体リガンド

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2013165312A Pending JP2013253090A (ja) 2005-07-08 2013-08-08 メラノコルチン受容体リガンド
JP2015140154A Active JP5965520B2 (ja) 2005-07-08 2015-07-14 メラノコルチン受容体リガンド

Country Status (20)

Country Link
US (8) US8039435B2 (OSRAM)
EP (6) EP3354273B1 (OSRAM)
JP (4) JP4734411B2 (OSRAM)
KR (2) KR101232201B1 (OSRAM)
CN (5) CN119119190A (OSRAM)
AU (2) AU2006269261B2 (OSRAM)
CA (4) CA2793119C (OSRAM)
DK (4) DK3354273T3 (OSRAM)
ES (4) ES2663916T3 (OSRAM)
FR (1) FR21C1060I2 (OSRAM)
HU (4) HUE031731T2 (OSRAM)
IL (3) IL188545A (OSRAM)
NL (1) NL301150I2 (OSRAM)
NZ (2) NZ565217A (OSRAM)
PL (4) PL2286825T3 (OSRAM)
PT (4) PT3354273T (OSRAM)
RU (2) RU2439079C2 (OSRAM)
SG (1) SG163585A1 (OSRAM)
SI (1) SI3354273T1 (OSRAM)
WO (1) WO2007008704A2 (OSRAM)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4734411B2 (ja) * 2005-07-08 2011-07-27 イプセン ファルマ ソシエテ パール アクシオン サンプリフィエ メラノコルチン受容体リガンド
DE102007020152A1 (de) * 2007-04-26 2008-10-30 Charité - Universitätsmedizin Berlin Mittel zur antiinfektiven Behandlung eines Patienten
US8563000B2 (en) 2007-05-25 2013-10-22 Ipsen Pharma S.A.S. Melanocortin receptor ligands modified with hydantoin
TW200848424A (en) * 2007-06-15 2008-12-16 Sod Conseils Rech Applic Cyclic peptide melanocortin receptor ligands
CN101980717A (zh) * 2007-11-05 2011-02-23 益普生制药股份有限公司 黑皮质素治疗胰岛素敏感的应用
EP2816055B1 (en) 2008-05-27 2018-12-19 Genzyme Corporation Peptide analogs of alpha-melanocyte stimulating hormons
CA2727317C (en) 2008-06-09 2015-02-17 Palatin Technologies, Inc. Melanocortin receptor-specific peptides for treatment of sexual dysfunction
UY32690A (es) 2009-06-08 2011-01-31 Astrazeneca Ab Péptidos específicos para receptores de melanocortina
WO2010144341A2 (en) 2009-06-08 2010-12-16 Palatin Technologies, Inc. Lactam-bridged melanocortin receptor-specific peptides
CA2761607C (en) 2009-06-08 2018-09-04 Yi-Qun Shi Melanocortin receptor-specific peptides
IN2012DN01493A (OSRAM) * 2009-08-05 2015-06-05 Ipsen Pharma Sas
HUE031856T2 (en) * 2009-08-31 2017-08-28 Tensive Controls Inc Stabilized melanocortin ligands
CN102686601A (zh) * 2009-11-16 2012-09-19 益普生制药股份有限公司 合成Ac-Arg-环(Cys-D-Ala-His-D-Phe-Arg-Trp-Cys)-NH2的方法
EP2501225B1 (en) 2009-11-16 2017-11-01 Ipsen Pharma S.A.S. Pharmaceutical compositions of melanocortin receptor ligands
CA2781402C (en) 2009-11-23 2017-03-21 Palatin Technologies, Inc. Melanocortin-1 receptor-specific cyclic peptides
EA201290295A1 (ru) 2009-11-23 2013-01-30 Палатин Текнолоджиз, Инк. Специфичные к рецептору меланокортина-1 линейные пептиды
JP6072020B2 (ja) * 2011-06-14 2017-02-01 イプセン ファルマ ソシエテ パール アクシオン サンプリフィエIpsen Pharma S.A.S. メラノコルチンリセプターリガンドを有効成分として含有する持続放出性組成物
LT3539551T (lt) 2011-12-29 2022-01-10 Rhythm Pharmaceuticals, Inc. Su melanokortino-4 receptoriumi susijusių sutrikimų gydymo būdas heterozigotiniuose nešiotojuose
EP2705835A1 (en) 2012-06-08 2014-03-12 Ipsen Pharma S.A.S. Aqueous gelling compositions of soluble active pharmaceutical peptides providing modified release
EP2722340B1 (en) 2012-10-19 2015-03-04 TXP Pharma GmbH Alpha- and gamma-MSH analogues
EP2968475A2 (en) 2013-03-14 2016-01-20 Questcor Pharmaceuticals, Inc. Acth for treatment of acute respiratory distress syndrome
EP2970389B1 (en) * 2013-03-15 2020-08-19 Rhythm Pharmaceuticals, Inc. Pharmaceutical compositions
US10196425B2 (en) 2013-03-15 2019-02-05 Rhythm Pharmaceuticals, Inc. Peptide compositions
BR112016024494B1 (pt) 2014-04-22 2024-02-06 Txp Pharma Gmbh Análogo de peptídeo e seu uso
PT3356386T (pt) * 2015-09-30 2024-05-17 Rhythm Pharmaceuticals Inc Método de tratamento de distúrbios associados à via do receptor da melanocortina-4
US11542302B2 (en) 2015-10-15 2023-01-03 Arizona Board Of Regents On Behalf Of The University Of Arizona Modulators of melanocortin receptors for the treatment of depression and anxiety
US10653743B2 (en) * 2015-10-15 2020-05-19 Arizona Board Of Regents On Behalf Of The University Of Arizona Methods for the treatment of depression and anxiety by a melanocortin 5 receptor antagonist, PG-20N
US20190255142A1 (en) * 2016-10-17 2019-08-22 Arizona Board Of Regents On Behalf Of The University Of Arizona Novel modulators of melanocortin receptors for the treatment of depression and anxiety
MA49883A (fr) * 2017-03-15 2021-04-21 Novo Nordisk As Composés bicycliques aptes à se lier au récepteur de mélanocortine 4
EP3773897A1 (en) 2018-04-06 2021-02-17 Rhythm Pharmaceuticals, Inc. Compositions for treating kidney disease
US20210221867A1 (en) * 2018-05-15 2021-07-22 Novo Nordisk A/S Compounds Capable of Binding to Melanocortin 4 Receptor
CA3100868A1 (en) * 2018-05-23 2019-11-28 Provincial Health Services Authority Radiolabeled melanocortin 1 receptor-specific alpha-melanocyte-stimulating hormone analogues for imaging or therapy
US11396535B2 (en) 2019-03-01 2022-07-26 Provincial Health Services Authority Cyclic peptide analogs of melanocortin and amanitin and methods of making such
AR123603A1 (es) * 2020-09-24 2022-12-21 Rhythm Pharmaceuticals Inc Métodos de tratamiento de los trastornos asociados a la vía del receptor de melanocortina
WO2022251650A1 (en) * 2021-05-27 2022-12-01 The Regents Of The University Of Michigan Mc3r agonist peptides
WO2024083843A1 (en) 2022-10-18 2024-04-25 Confo Therapeutics N.V. Amino acid sequences directed against the melanocortin 4 receptor and polypeptides comprising the same for the treatment of mc4r-related diseases and disorders
WO2025123059A1 (en) * 2023-12-07 2025-06-12 Endevica Bio, Inc. Non-naturally occurring melanocortin analogs and uses thereof for treating substance use disorders

Family Cites Families (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US613874A (en) 1898-11-08 George e
US1613874A (en) 1922-03-29 1927-01-11 Miner Inc W H Friction draft gear
US5652214A (en) 1989-06-05 1997-07-29 Cephalon, Inc. Treating disorders by application of insulin-like growth factors and analogs
US5672659A (en) 1993-01-06 1997-09-30 Kinerton Limited Ionic molecular conjugates of biodegradable polyesters and bioactive polypeptides
US5595760A (en) 1994-09-02 1997-01-21 Delab Sustained release of peptides from pharmaceutical compositions
US5665702A (en) 1995-06-06 1997-09-09 Biomeasure Incorporated Ionic molecular conjugates of N-acylated derivatives of poly(2-amino-2-deoxy-D-glucose) and polypeptides
US5916883A (en) 1996-11-01 1999-06-29 Poly-Med, Inc. Acylated cyclodextrin derivatives
SE9700620D0 (sv) 1997-02-21 1997-02-21 Wapharm Ab Cykliska peptider med selektivitet för MSH-receptor subtyper
US6350430B1 (en) 1997-10-27 2002-02-26 Lion Bioscience Science Ag Melanocortin receptor ligands and methods of using same
US6127381A (en) * 1998-04-28 2000-10-03 Basu; Amaresh Isoquinoline compound melanocortin receptor ligands and methods of using same
EP1100970A2 (en) * 1998-07-27 2001-05-23 Iowa State University Research Foundation, Inc. Melanocortin-4 receptor gene and use as a genetic marker for fat content, weight gain, and/or feed consumption of animals
AU775289B2 (en) 1998-08-21 2004-07-29 Children's Medical Center Corporation Use of melanin for inhibition of angiogenesis and macular degeneration
US6603058B1 (en) 1998-12-09 2003-08-05 Oklahoma Medical Research Foundation Non-human animal model for obesity and uses thereof
US6716810B1 (en) 1998-12-09 2004-04-06 Eleanor Roosevelt Institute Composition and method for regulation of body weight and associated conditions
KR100519201B1 (ko) * 1999-03-29 2005-10-06 더 프록터 앤드 갬블 캄파니 멜라노코르틴 수용체 리간드
WO2003006620A2 (en) * 2001-07-11 2003-01-23 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptides
US6579968B1 (en) * 1999-06-29 2003-06-17 Palatin Technologies, Inc. Compositions and methods for treatment of sexual dysfunction
US7176279B2 (en) 2000-06-28 2007-02-13 Palatin Technologies, Inc. Cyclic peptide compositions and methods for treatment of sexual dysfunction
AU1758401A (en) 1999-11-12 2001-06-06 Merck & Co., Inc. Melanocortin-3 receptor deficient cells, non-human transgenic animals and methods of selecting compounds which regulate body weight
US6600015B2 (en) 2000-04-04 2003-07-29 Hoffmann-La Roche Inc. Selective linear peptides with melanocortin-4 receptor (MC4-R) agonist activity
AP2001002196A0 (en) * 2000-06-28 2002-12-21 Pfizer Prod Inc Melanocortin receptor ligands.
US6720324B2 (en) 2000-07-05 2004-04-13 Synaptic Pharmaceutical Corporation Selective melanin concentrating hormone-1 (MCH1) receptor antagonists and uses thereof
JP2004510960A (ja) 2000-09-13 2004-04-08 エレノア ルーズベルト インスティテュート 肥満および糖尿病におけるインスリン抵抗性を治療する方法
US20030113263A1 (en) 2001-02-13 2003-06-19 Oregon Health And Sciences University, A Non-Profit Organization Methods and reagents for using mammalian melanocortin receptor antagonists to treat cachexia
HUP0401544A2 (hu) 2001-03-02 2004-12-28 Bristol-Myers Squibb Company Melanokortin receptor modulátoraiként hasznos vegyületek és a vegyületeket tartalmazó gyógyszerkészítmények
US6770645B2 (en) * 2001-03-16 2004-08-03 Pfizer Inc. Pharmaceutically active compounds
US7034004B2 (en) 2002-05-07 2006-04-25 University Of Florida Peptides and methods for the control of obesity
US20040128136A1 (en) * 2002-09-20 2004-07-01 Irani Pourang Polad Internet voice browser
AU2004251616A1 (en) * 2003-06-19 2005-01-06 Eli Lilly And Company Melanocortin receptor 4(MC4) agonists and their uses
WO2005000338A1 (en) 2003-06-19 2005-01-06 Eli Lilly And Company Uses of melanocortin-3 receptor (mc3r) agonist peptides
US7084111B2 (en) 2003-06-23 2006-08-01 University Of Florida Research Foundation, Inc. Melanocortin receptor templates, peptides, and use thereof
US20070293423A1 (en) 2003-08-20 2007-12-20 Eli Lilly And Company Compounds, Methods and Formulations for the Oral Delivery of a Glucagon-Like Peptide (Glp)-1 Compound or a Melanocortin-4 Receptor (Mc4) Agonist Peptide
EP1658273B1 (en) 2003-08-20 2007-01-03 Eli Lilly And Company Compounds, methods and formulations for the oral delivery of a glucagon like peptide (glp)-1 compound or an melanocortin 4 receptor (mc4) agonist peptide
WO2005040109A1 (en) * 2003-10-22 2005-05-06 Neurocrine Biosciences, Inc. Ligands of melanocortin receptors and compositions and methods related thereto
DE10355559A1 (de) 2003-11-21 2005-06-23 Orthogen Ag Transskin
US20070155660A1 (en) 2003-12-10 2007-07-05 Marsh Donald J Inhibition of voluntary ethanol consumption with selective melanocortin 4-receptor agonists
CA2557739A1 (en) * 2004-03-29 2005-11-03 Eli Lilly And Company Uses of melanocortin-4 receptor (mc4r) agonist peptides administered by continuous infusion
US8569234B2 (en) 2004-10-08 2013-10-29 Clinuvel Pharmaceuticals Limited Compositions and methods for including melanogenesis in a subject
WO2006073772A1 (en) 2005-01-05 2006-07-13 Eli Lilly And Company Polyethylene glycol linked mc4r or mc3r agonist peptides
WO2006073771A2 (en) 2005-01-05 2006-07-13 Eli Lilly And Company Polyethylene glycol linked mc4r or mc3r agonist peptides
JP4734411B2 (ja) * 2005-07-08 2011-07-27 イプセン ファルマ ソシエテ パール アクシオン サンプリフィエ メラノコルチン受容体リガンド
US8466104B2 (en) 2005-08-26 2013-06-18 Abbvie Inc. Therapeutically active alpha MSH analogues

Similar Documents

Publication Publication Date Title
JP2010090130A5 (OSRAM)
RU2401841C2 (ru) Лиганды рецепторов меланокортинов
RU2009131092A (ru) Лиганды рецепторов меланокортинов
JP2009500427A5 (OSRAM)
CA2689016A1 (en) Melanocortin receptor ligands modified with hydantoin
KR101226165B1 (ko) 피부 외용제 조성물
US6262021B1 (en) Use of substances having oxytocin activity for preparation of medicaments for wound healing
TWI619505B (zh) 脫毛症治療劑
TWI374030B (en) Use of melanocortins to treat insulin sensitivity
Blank et al. Actions of CRF and its analogs
JP2021102650A5 (OSRAM)
TW201601743A (zh) 外周kappa鴉片受體促進劑用於製備預防、抑制或治療噁心及嘔吐之藥物的用途
RU2012136530A (ru) Новые соединения, влияющие на пищевое поведение
CN108135965B (zh) 用于伤口愈合的含p物质的药物组合物
Lippert et al. Effects of oxytocin outside pregnancy
Stern Nursing posture is elicited rapidly in maternally naive, haloperidol-treated female and male rats in response to ventral trunk stimulation from active pups
RU2012106302A (ru) Аналоги инсулиноподобного фактора роста-1 (igf-1), содержащие аминокислотную замену в положении 59
JP6800372B2 (ja) 持続型パルミチン酸結合GnRH誘導体及びこれを含む薬剤学的組成物
CN110935007B (zh) 利那洛肽复方组合物、制剂及其用途和制备方法
AU2016302644A1 (en) CNP cyclic peptide, and medicine, external preparation and cosmetic each containing said cyclic peptide
CN102631663B (zh) 一种治疗男性不育、阳痿早泄的制剂及其应用
Kawakami Electro-myographic study of the human abdominal muscles affected by sexual hormones
WO2017088177A1 (zh) 贻贝粘蛋白产品及其预防和抑制神经炎症的应用
TW202116347A (zh) 肽及其作為製備治療發炎性疾病及疼痛的藥物的用途
Laurent et al. TGF-beta antibodies: a novel treatment for pulmonary fibrosis?