JP2009534458A5 - - Google Patents

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Publication number
JP2009534458A5
JP2009534458A5 JP2009507166A JP2009507166A JP2009534458A5 JP 2009534458 A5 JP2009534458 A5 JP 2009534458A5 JP 2009507166 A JP2009507166 A JP 2009507166A JP 2009507166 A JP2009507166 A JP 2009507166A JP 2009534458 A5 JP2009534458 A5 JP 2009534458A5
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JP
Japan
Prior art keywords
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Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2009507166A
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English (en)
Japanese (ja)
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JP2009534458A (ja
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Publication date
Priority claimed from GB0608269A external-priority patent/GB0608269D0/en
Application filed filed Critical
Priority claimed from PCT/GB2007/001537 external-priority patent/WO2007125331A2/en
Publication of JP2009534458A publication Critical patent/JP2009534458A/ja
Publication of JP2009534458A5 publication Critical patent/JP2009534458A5/ja
Withdrawn legal-status Critical Current

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JP2009507166A 2006-04-26 2007-04-26 アミノ−エチル−アミノ−アリール(aeaa)化合物およびそれらの使用 Withdrawn JP2009534458A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74563006P 2006-04-26 2006-04-26
GB0608269A GB0608269D0 (en) 2006-04-26 2006-04-26 Therapeutic compounds
PCT/GB2007/001537 WO2007125331A2 (en) 2006-04-26 2007-04-26 Amino-ethyl-amino-aryl (aeaa) compounds and their use

Publications (2)

Publication Number Publication Date
JP2009534458A JP2009534458A (ja) 2009-09-24
JP2009534458A5 true JP2009534458A5 (https=) 2010-06-17

Family

ID=38581449

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009507166A Withdrawn JP2009534458A (ja) 2006-04-26 2007-04-26 アミノ−エチル−アミノ−アリール(aeaa)化合物およびそれらの使用

Country Status (8)

Country Link
US (1) US20090247519A1 (https=)
EP (1) EP2024333A2 (https=)
JP (1) JP2009534458A (https=)
AU (1) AU2007245496A1 (https=)
CA (1) CA2649995A1 (https=)
IL (1) IL194899A0 (https=)
MX (1) MX2008013718A (https=)
WO (1) WO2007125331A2 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008069976A2 (en) * 2006-12-01 2008-06-12 President And Fellows Of Harvard College Compounds and methods for enzyme-mediated tumor imaging and therapy
MX2009010127A (es) * 2007-03-22 2009-11-05 Vertex Pharma Compuestos utiles como inhibidores de janus cinasas.
CA2727196A1 (en) 2008-06-10 2009-12-17 Novartis Ag Organic compounds
JP2011522865A (ja) * 2008-06-13 2011-08-04 ノバルティス アーゲー Ia心不全および癌の治療に有用なプロテインキナーゼd阻害剤としての2,4’−ビピリジニル化合物
CA2778931A1 (en) 2009-06-12 2010-12-16 Marianne Allard Guanine riboswitch binding compounds and their use as antibiotics
WO2011036074A1 (en) * 2009-09-24 2011-03-31 Basf Se Aminoquinazoline compounds for combating invertebrate pests
EP2528606B1 (en) * 2010-01-28 2014-09-24 Alexander Levitzki Quinazoline-based t cell proliferation inhibitors
JP2013529181A (ja) * 2010-03-25 2013-07-18 ザ ジェイ. デヴィッド グラッドストーン インスティテューツ 神経障害を治療するための組成物および方法
WO2018172250A1 (en) 2017-03-21 2018-09-27 Bayer Pharma Aktiengesellschaft 2-methyl-quinazolines
US20220274979A1 (en) 2018-04-18 2022-09-01 Bayer Pharma Aktiengesellschaft 2-methyl-aza-quinazolines
US12522587B2 (en) 2018-05-04 2026-01-13 Remedy Plan, Inc. Cancer treatments targeting cancer stem cells
US20220388962A1 (en) * 2019-08-22 2022-12-08 Biohaven Therapeutics Ltd. Molecules that bind to tdp-43 for the treatment of amyotrophic lateral sclerosis and related disorders
EP4055008A1 (en) 2019-11-06 2022-09-14 Remedy Plan, Inc. Cancer treatments targeting cancer stem cells
CA3188260A1 (en) 2020-08-07 2022-02-10 Dimitrios Iliopoulos Small molecules for the treatment of autoimmune diseases and cancer
EP4052700A1 (en) * 2021-03-03 2022-09-07 Instytut Biologii doswiadczalnej imienia Marcelego Nenckiego Polskiej Akademii Nauk Inhibitor of protein kinase d (pkd) for use in prevention or treatment of obesity and a pharmaceutical composition for such use
JP2024511298A (ja) 2021-03-03 2024-03-13 インスティチュート バイオロジー ドスウィアドチュルネジ アイエム. マルセレゴ ネンキエゴ ポルスカ アカデミア ノーク 高脂血症の予防または治療に使用するためのタンパク質キナーゼdの阻害剤

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1377554A1 (en) * 1999-06-16 2004-01-07 University Of Iowa Research Foundation Antagonism of immunostimulatory cpg-oligonucleotides by 4-aminoquinolines and other weak bases
JP4272338B2 (ja) * 2000-09-22 2009-06-03 バイエル アクチェンゲゼルシャフト ピリジン誘導体
ATE466581T1 (de) * 2001-12-07 2010-05-15 Vertex Pharma Verbindungen auf pyrimidin-basis als gsk-3-hemmer
WO2004030672A1 (en) * 2002-10-02 2004-04-15 Merck Patent Gmbh Use of 4 amino-quinazolines as anti cancer agents
CL2004000409A1 (es) * 2003-03-03 2005-01-07 Vertex Pharma Compuestos derivados de 2-(cilo sustituido)-1-(amino u oxi sustituido)-quinazolina, inhibidores de canales ionicos de sodio y calcio dependientes de voltaje; composicion farmaceutica; y uso del compuesto en el tratamiento de dolor agudo, cronico, neu
TW200519094A (en) * 2003-07-02 2005-06-16 Vertex Pharma Pyrimidines useful as modulators of voltage-gated ion channels
CR9465A (es) * 2005-03-25 2008-06-19 Surface Logix Inc Compuestos mejorados farmacocineticamente

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