JP2009533338A5 - - Google Patents
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- Publication number
- JP2009533338A5 JP2009533338A5 JP2009504144A JP2009504144A JP2009533338A5 JP 2009533338 A5 JP2009533338 A5 JP 2009533338A5 JP 2009504144 A JP2009504144 A JP 2009504144A JP 2009504144 A JP2009504144 A JP 2009504144A JP 2009533338 A5 JP2009533338 A5 JP 2009533338A5
- Authority
- JP
- Japan
- Prior art keywords
- styrylquinazoline
- patent document
- compounds
- rastinejad
- mutant
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- AIVRDUVZOFTAGC-UHFFFAOYSA-N 2-(2-phenylethenyl)quinazoline Chemical compound N=1C=C2C=CC=CC2=NC=1C=CC1=CC=CC=C1 AIVRDUVZOFTAGC-UHFFFAOYSA-N 0.000 description 3
- 150000001875 compounds Chemical class 0.000 description 2
- 230000002209 hydrophobic effect Effects 0.000 description 1
- 238000005556 structure-activity relationship Methods 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NZ546477A NZ546477A (en) | 2006-04-07 | 2006-04-07 | 4-Alkylamino-2-(heterocyclic)quinazolines and their use in cancer therapy |
| PCT/NZ2007/000077 WO2007117161A1 (en) | 2006-04-07 | 2007-04-04 | Substituted ring fused azines and their use in cancer therapy |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009533338A JP2009533338A (ja) | 2009-09-17 |
| JP2009533338A5 true JP2009533338A5 (https=) | 2010-05-06 |
Family
ID=38581368
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009504144A Pending JP2009533338A (ja) | 2006-04-07 | 2007-04-04 | 置換環縮合アジンおよび癌治療におけるそれらの使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20090318479A1 (https=) |
| EP (1) | EP2004637A4 (https=) |
| JP (1) | JP2009533338A (https=) |
| CN (1) | CN101460490A (https=) |
| AU (1) | AU2007235751A1 (https=) |
| CA (1) | CA2648323A1 (https=) |
| NZ (1) | NZ546477A (https=) |
| WO (1) | WO2007117161A1 (https=) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012046207A1 (en) * | 2010-10-08 | 2012-04-12 | Paraco Technology Limited | Anti-parasitic substituted ring fused azine compounds |
| US8710064B2 (en) * | 2011-10-20 | 2014-04-29 | China Medical University | 2-aryl-4-quinazolinones and their pharmaceutical compositions |
| CN104540830A (zh) | 2012-06-07 | 2015-04-22 | 霍夫曼-拉罗奇有限公司 | 端锚聚合酶的吡唑并嘧啶酮和吡唑并吡啶酮抑制剂 |
| WO2013182580A1 (en) | 2012-06-07 | 2013-12-12 | F. Hoffmann-La Roche Ag | Pyrrolopyrimidone and pyrrolopyridone inhibitors of tankyrase |
| EP2970199A1 (en) | 2013-03-11 | 2016-01-20 | Bristol-Myers Squibb Company | Isoquinolines as potassium ion channel inhibitors |
| JP6527513B2 (ja) | 2013-11-20 | 2019-06-05 | シグナルケム・ライフサイエンシーズ・コーポレイションＳｉｇｎａｌｃｈｅｍ Ｌｉｆｅｓｃｉｅｎｃｅｓ Ｃｏｒｐｏｒａｔｉｏｎ | Ｔａｍファミリーキナーゼ阻害剤としてのキナゾリン誘導体 |
| NZ730475A (en) * | 2014-10-29 | 2018-09-28 | Dong A St Co Ltd | Novel pyridopyrimidinone compounds for modulating the catalytic activity of histone lysine demethylases (kdms) |
| US20170057955A1 (en) * | 2015-08-26 | 2017-03-02 | Dong-A Socio Holdings Co., Ltd. | Pyridopyrimidinone Compounds for Modulating the Catalytic Activity of Histone Lysine Demethylases (KDMs) |
| CN107721982B (zh) * | 2017-10-16 | 2019-12-03 | 中山大学 | 一种抗肥胖症化合物及其制备方法和应用 |
| CN110483394A (zh) * | 2019-09-02 | 2019-11-22 | 广东工业大学 | 一种化合物的应用 |
| CN113072543B (zh) * | 2020-01-03 | 2022-07-22 | 南方医科大学 | 一种2-芳杂环基喹唑啉酮类化合物及其制备方法和用途 |
| US20230339866A1 (en) * | 2020-02-04 | 2023-10-26 | TroBio Therapeutics Pty Ltd | Quinazoline compounds and the use thereof in the treatment of cancer |
| MX2023003273A (es) | 2020-09-21 | 2023-04-26 | Landos Biopharma Inc | Ligandos de nlrx1. |
| CN114044769B (zh) * | 2021-11-25 | 2023-12-12 | 中山大学 | 一种β-吲哚喹唑啉酮衍生物及其制备方法和应用 |
| CN117247374B (zh) * | 2022-06-10 | 2026-03-17 | 四川科伦博泰生物医药股份有限公司 | 一种bcl-xl抑制剂及其制药用途 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3897432A (en) * | 1971-04-21 | 1975-07-29 | Merck & Co Inc | Substituted benzimidazole derivatives |
| AU1290700A (en) * | 1998-12-02 | 2000-06-19 | Pfizer Products Inc. | Methods and compositions for restoring conformational stability of a protein of the p53 family |
| DK1088818T3 (da) * | 1999-10-01 | 2005-03-14 | Hoffmann La Roche | Quinolin-4-yl-derivater |
| CN1186324C (zh) * | 2000-04-27 | 2005-01-26 | 山之内制药株式会社 | 稠合杂芳基衍生物 |
| WO2002062767A1 (en) * | 2001-02-07 | 2002-08-15 | Sumitomo Pharmaceuticals Company, Limited | Novel quinazoline derivatives |
-
2006
- 2006-04-07 NZ NZ546477A patent/NZ546477A/en not_active IP Right Cessation
-
2007
- 2007-04-04 CN CNA2007800204647A patent/CN101460490A/zh active Pending
- 2007-04-04 JP JP2009504144A patent/JP2009533338A/ja active Pending
- 2007-04-04 US US12/296,377 patent/US20090318479A1/en not_active Abandoned
- 2007-04-04 CA CA002648323A patent/CA2648323A1/en not_active Abandoned
- 2007-04-04 WO PCT/NZ2007/000077 patent/WO2007117161A1/en not_active Ceased
- 2007-04-04 AU AU2007235751A patent/AU2007235751A1/en not_active Abandoned
- 2007-04-04 EP EP07747705A patent/EP2004637A4/en not_active Withdrawn
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