JP2009524675A5 - - Google Patents

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Publication number
JP2009524675A5
JP2009524675A5 JP2008552415A JP2008552415A JP2009524675A5 JP 2009524675 A5 JP2009524675 A5 JP 2009524675A5 JP 2008552415 A JP2008552415 A JP 2008552415A JP 2008552415 A JP2008552415 A JP 2008552415A JP 2009524675 A5 JP2009524675 A5 JP 2009524675A5
Authority
JP
Japan
Prior art keywords
bioavailability
tetracycline compound
hydrogen
use according
enhancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008552415A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009524675A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/002081 external-priority patent/WO2007087416A2/en
Publication of JP2009524675A publication Critical patent/JP2009524675A/ja
Publication of JP2009524675A5 publication Critical patent/JP2009524675A5/ja
Pending legal-status Critical Current

Links

JP2008552415A 2006-01-24 2007-01-24 テトラサイクリンの経口バイオアベイラビリティーを増加する方法 Pending JP2009524675A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76181906P 2006-01-24 2006-01-24
PCT/US2007/002081 WO2007087416A2 (en) 2006-01-24 2007-01-24 Methods of increasing oral bioavailability of tetracyclines

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010013625A Division JP2010106043A (ja) 2006-01-24 2010-01-25 テトラサイクリンの経口バイオアベイラビリティーを増加する方法

Publications (2)

Publication Number Publication Date
JP2009524675A JP2009524675A (ja) 2009-07-02
JP2009524675A5 true JP2009524675A5 (https=) 2010-03-18

Family

ID=38181071

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2008552415A Pending JP2009524675A (ja) 2006-01-24 2007-01-24 テトラサイクリンの経口バイオアベイラビリティーを増加する方法
JP2010013625A Pending JP2010106043A (ja) 2006-01-24 2010-01-25 テトラサイクリンの経口バイオアベイラビリティーを増加する方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010013625A Pending JP2010106043A (ja) 2006-01-24 2010-01-25 テトラサイクリンの経口バイオアベイラビリティーを増加する方法

Country Status (6)

Country Link
US (2) US9078811B2 (https=)
EP (2) EP2298324A1 (https=)
JP (2) JP2009524675A (https=)
AU (2) AU2007208214B2 (https=)
CA (1) CA2639406A1 (https=)
WO (1) WO2007087416A2 (https=)

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CA2531728A1 (en) 2003-07-09 2005-02-03 Paratek Pharmaceuticals, Inc. Substituted tetracycline compounds
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AU2006206359B2 (en) * 2005-01-21 2011-03-31 Allergan Pharmaceuticals International Limited A tetracycline metal complex in a solid dosage form
WO2006084265A1 (en) 2005-02-04 2006-08-10 Paratek Pharmaceuticals, Inc. 11a, 12-DERIVATIVES OF TETRACYCLINE COMPOUNDS
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PT2120963T (pt) 2006-12-21 2018-12-17 Paratek Pharm Innc Compostos tetraciclina substituídos para tratamento de distúrbios inflamatórios da pele
PL2109602T3 (pl) * 2006-12-21 2014-09-30 Paratek Pharm Innc Pochodne tetracyliny do leczenia zakażeń bakteryjnych, wirusowych i pasożytniczych
JP2010523684A (ja) 2007-04-12 2010-07-15 パラテック ファーマシューティカルズ インコーポレイテッド テトラサイクリン化合物を用いる、脊髄筋委縮症を治療するための方法
CA2717703A1 (en) 2008-03-05 2009-09-11 Paratek Pharmaceuticals, Inc. Minocycline compounds and methods of use thereof
PT2271348T (pt) * 2008-03-28 2018-04-16 Paratek Pharm Innc Formulação de comprimido oral de composto de tetraciclina
JP2011517697A (ja) * 2008-04-14 2011-06-16 パラテック ファーマシューティカルズ インコーポレイテッド 置換テトラサイクリン化合物
TW202216656A (zh) * 2008-05-19 2022-05-01 美商Ｐｒｔｋ Ｓｐｖ２公司 四環素化合物之甲苯磺酸鹽及同素異形體
PT2323972E (pt) 2008-08-08 2013-10-09 Tetraphase Pharmaceuticals Inc Compostos de tetraciclina substituídos com c7-flúor
EP2341771A4 (en) * 2008-09-19 2012-08-15 Paratek Pharm Innc TETRACYCLINE COMPOUNDS FOR THE TREATMENT OF RHEUMATOID ARTHRITIS AND RELATED THERAPEUTIC METHODS
EP2427425B1 (en) 2009-05-08 2017-03-08 Tetraphase Pharmaceuticals, Inc. Tetracycline compounds
IN2012DN02502A (https=) 2009-08-28 2015-08-28 Tetraphase Pharmaceuticals Inc
US9119793B1 (en) 2011-06-28 2015-09-01 Medicis Pharmaceutical Corporation Gastroretentive dosage forms for doxycycline
JP5952912B2 (ja) 2011-12-15 2016-07-13 アルカーメス ファーマ アイルランド リミテッド 二級アミン化合物のプロドラッグ
BR112015004523B1 (pt) 2012-08-31 2020-08-04 Tetraphase Pharmaceuticals, Inc Compostos de tetraciclina, composições farmacêuticas e seus usos
US10842802B2 (en) 2013-03-15 2020-11-24 Medicis Pharmaceutical Corporation Controlled release pharmaceutical dosage forms
WO2017165729A1 (en) * 2016-03-24 2017-09-28 Paratek Pharmaceuticals, Inc. Methods for treating and preventing c. difficile infection
CN110582486B (zh) 2016-10-19 2024-01-12 四相制药公司 艾若威四环素的结晶形式
BR112019008897A2 (pt) 2016-11-01 2019-08-13 Paratek Pharm Innc método para tratar pneumonia bacteriana adquirida na comunidade.
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas
WO2023238143A1 (en) * 2022-06-11 2023-12-14 Gufic Biosciences Limited A freeze dried parenteral composition of omadacycline tosylate with improved stability

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