JP2009517417A - Crth2レセプター活性を有するオキサジアゾール誘導体類 - Google Patents
Crth2レセプター活性を有するオキサジアゾール誘導体類 Download PDFInfo
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- JP2009517417A JP2009517417A JP2008542640A JP2008542640A JP2009517417A JP 2009517417 A JP2009517417 A JP 2009517417A JP 2008542640 A JP2008542640 A JP 2008542640A JP 2008542640 A JP2008542640 A JP 2008542640A JP 2009517417 A JP2009517417 A JP 2009517417A
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Classifications
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Landscapes
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| GBGB0524428.0A GB0524428D0 (en) | 2005-11-30 | 2005-11-30 | Medicinal use of receptor ligands |
| PCT/EP2006/011216 WO2007062773A1 (en) | 2005-11-30 | 2006-11-22 | Oxadiazole derivatives with crth2 receptor activity |
Publications (2)
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| JP2009517417A true JP2009517417A (ja) | 2009-04-30 |
| JP2009517417A5 JP2009517417A5 (enExample) | 2010-01-14 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP2008542640A Withdrawn JP2009517417A (ja) | 2005-11-30 | 2006-11-22 | Crth2レセプター活性を有するオキサジアゾール誘導体類 |
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| EP (1) | EP1960376A1 (enExample) |
| JP (1) | JP2009517417A (enExample) |
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| CA (1) | CA2631652A1 (enExample) |
| CR (1) | CR10034A (enExample) |
| EA (1) | EA200801494A1 (enExample) |
| EC (1) | ECSP088479A (enExample) |
| GB (1) | GB0524428D0 (enExample) |
| HN (1) | HN2008000817A (enExample) |
| NO (1) | NO20082917L (enExample) |
| SV (1) | SV2009002925A (enExample) |
| WO (1) | WO2007062773A1 (enExample) |
| ZA (1) | ZA200804687B (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5069804B2 (ja) * | 2010-03-01 | 2012-11-07 | 隆雄 篠澤 | 筋萎縮性側索硬化症(als)の患者の進行度を判定し進行のモニターを行う方法 |
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|---|---|---|---|---|
| EP2327693B9 (en) | 2007-12-14 | 2012-10-24 | Pulmagen Therapeutics (Asthma) Limited | Indoles and their therapeutic use |
| AU2010212970A1 (en) | 2009-02-12 | 2011-08-18 | Merck Serono S.A. | Phenoxy acetic acid derivatives |
| EP2590944B1 (en) | 2010-07-05 | 2015-09-30 | Actelion Pharmaceuticals Ltd. | 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin d2 receptor modulators |
| EP2457900A1 (en) | 2010-11-25 | 2012-05-30 | Almirall, S.A. | New pyrazole derivatives having CRTh2 antagonistic behaviour |
| WO2013088109A1 (en) | 2011-12-16 | 2013-06-20 | Oxagen Limited | Combination of crth2 antagonist and a proton pump inhibitor for the treatment of eosinophilic esophagitis |
| ES2624379T3 (es) | 2011-12-21 | 2017-07-14 | Idorsia Pharmaceuticals Ltd | Derivados de heterociclilo y su uso como moduladores del receptor de prostaglandina D2 |
| US9169270B2 (en) | 2012-07-05 | 2015-10-27 | Actelion Pharmaceuticals Ltd. | 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin D2 receptor modulators |
| CN104744429B (zh) * | 2013-12-27 | 2016-09-28 | 启东韶远化学科技有限公司 | 一种环并[b]噻吩-3(2H)-酮-1,1-二氧化物的简单合成方法 |
| WO2016202341A1 (en) * | 2015-06-15 | 2016-12-22 | Nmd Pharma Aps | Compounds for use in treating neuromuscular disorders |
| EP3595777A4 (en) * | 2017-03-14 | 2021-01-20 | Dana-Farber Cancer Institute, Inc. | LOW MOLECULAR SENSITIVITY OF BAX ACTIVATION FOR INDUCING CELL DEATH |
| US11591284B2 (en) | 2017-12-14 | 2023-02-28 | Nmd Pharma A/S | Compounds for the treatment of neuromuscular disorders |
| US11147788B2 (en) | 2017-12-14 | 2021-10-19 | Nmd Pharma A/S | Compounds for the treatment of neuromuscular disorders |
| US12440477B2 (en) | 2017-12-14 | 2025-10-14 | Nmd Pharma A/S | Compounds for the treatment of neuromuscular disorders |
| US11730714B2 (en) | 2017-12-14 | 2023-08-22 | Nmd Pharma A/S | Compounds for the treatment of neuromuscular disorders |
| US10385028B2 (en) | 2017-12-14 | 2019-08-20 | Nmd Pharma A/S | Compounds for the treatment of neuromuscular disorders |
| TWI780281B (zh) * | 2017-12-14 | 2022-10-11 | 丹麥商Nmd藥品公司 | 用於治療神經肌肉病症的化合物 |
| EP3986878B1 (en) * | 2019-06-19 | 2024-09-25 | NMD Pharma A/S | Process for the preparation of clc-1 chloride channel inhibitors |
| PH12021552771A1 (en) | 2019-06-19 | 2022-10-17 | Nmd Pharma As | Compounds for the treatment of neuromuscular disorders |
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| SE0200356D0 (sv) | 2002-02-05 | 2002-02-05 | Astrazeneca Ab | Novel use |
| US7534897B2 (en) | 2002-05-16 | 2009-05-19 | Shionogi & Co., Ltd. | Indole arylsulfonaimide compounds exhibiting PGD 2 receptor antagonism |
| JPWO2003097042A1 (ja) | 2002-05-16 | 2005-09-15 | 塩野義製薬株式会社 | Pgd2受容体拮抗剤 |
| GB2388540A (en) | 2002-05-17 | 2003-11-19 | Bayer Ag | New use of Ramatroban |
| TW200307542A (en) | 2002-05-30 | 2003-12-16 | Astrazeneca Ab | Novel compounds |
| SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
| SE0301010D0 (sv) | 2003-04-07 | 2003-04-07 | Astrazeneca Ab | Novel compounds |
| SA04250253B1 (ar) | 2003-08-21 | 2009-11-10 | استرازينيكا ايه بي | احماض فينوكسي اسيتيك مستبدلة باعتبارها مركبات صيدلانية لعلاج الامراض التنفسية مثل الربو ومرض الانسداد الرئوي المزمن |
| EP2336113A1 (en) * | 2004-05-29 | 2011-06-22 | 7TM Pharma A/S | CRTH2 Receptor Ligands for Medical Use |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5069804B2 (ja) * | 2010-03-01 | 2012-11-07 | 隆雄 篠澤 | 筋萎縮性側索硬化症(als)の患者の進行度を判定し進行のモニターを行う方法 |
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| EP1960376A1 (en) | 2008-08-27 |
| BRPI0619260A2 (pt) | 2011-09-27 |
| KR20080072688A (ko) | 2008-08-06 |
| AU2006319462A1 (en) | 2007-06-07 |
| ECSP088479A (es) | 2008-07-30 |
| HN2008000817A (es) | 2010-10-01 |
| CN101316829A (zh) | 2008-12-03 |
| WO2007062773A1 (en) | 2007-06-07 |
| CR10034A (es) | 2008-07-22 |
| CA2631652A1 (en) | 2007-06-07 |
| US20080312220A1 (en) | 2008-12-18 |
| GB0524428D0 (en) | 2006-01-11 |
| ZA200804687B (en) | 2009-10-28 |
| SV2009002925A (es) | 2009-01-05 |
| NO20082917L (no) | 2008-08-29 |
| EA200801494A1 (ru) | 2008-12-30 |
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