JP2009161540A5 - - Google Patents
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- Publication number
- JP2009161540A5 JP2009161540A5 JP2009021716A JP2009021716A JP2009161540A5 JP 2009161540 A5 JP2009161540 A5 JP 2009161540A5 JP 2009021716 A JP2009021716 A JP 2009021716A JP 2009021716 A JP2009021716 A JP 2009021716A JP 2009161540 A5 JP2009161540 A5 JP 2009161540A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- unsubstituted
- alkoxy
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 125000000217 alkyl group Chemical group 0.000 claims 7
- 125000003545 alkoxy group Chemical group 0.000 claims 3
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 2
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 claims 2
- 229910052736 halogen Inorganic materials 0.000 claims 2
- 150000002367 halogens Chemical class 0.000 claims 2
- 229910052760 oxygen Inorganic materials 0.000 claims 2
- 239000001301 oxygen Substances 0.000 claims 2
- ZOXJGFHDIHLPTG-UHFFFAOYSA-N Boron Chemical group [B] ZOXJGFHDIHLPTG-UHFFFAOYSA-N 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- 125000004104 aryloxy group Chemical group 0.000 claims 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 1
- 229910052796 boron Inorganic materials 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 150000002431 hydrogen Chemical class 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 claims 1
- 229920002554 vinyl polymer Polymers 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43437502P | 2002-12-18 | 2002-12-18 | |
| US43609502P | 2002-12-23 | 2002-12-23 | |
| US43784903P | 2003-01-03 | 2003-01-03 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Division JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009161540A JP2009161540A (ja) | 2009-07-23 |
| JP2009161540A5 true JP2009161540A5 (enExample) | 2011-03-17 |
Family
ID=32686073
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Withdrawn JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
| JP2009021716A Withdrawn JP2009161540A (ja) | 2002-12-18 | 2009-02-02 | ボロン酸複合体を含む抗生物質および使用法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Withdrawn JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20040224923A1 (enExample) |
| EP (2) | EP1581500A4 (enExample) |
| JP (2) | JP2006511613A (enExample) |
| KR (1) | KR20050084378A (enExample) |
| CN (1) | CN101928295A (enExample) |
| AU (1) | AU2003299821B2 (enExample) |
| BR (1) | BR0317564A (enExample) |
| CA (1) | CA2509645A1 (enExample) |
| MX (1) | MXPA05006685A (enExample) |
| NZ (1) | NZ540870A (enExample) |
| WO (1) | WO2004056322A2 (enExample) |
Families Citing this family (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1325504C (zh) | 2002-01-10 | 2007-07-11 | 宾夕法尼亚州研究基金会 | 制备二芳基硼酸烷基酯和络合的二芳基硼酸的方法 |
| US7390806B2 (en) * | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
| MXPA05006685A (es) * | 2002-12-18 | 2005-12-14 | Anacor Pharmaceuticals Inc | Antibioticos que contienen complejos de acido borinico y metodos de uso. |
| AR049916A1 (es) * | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Usos anti-parasitarios de complejos de acido borinico |
| AR049915A1 (es) * | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Compuestos con contenido de boro y metodos de uso de los mismos |
| EP1765360B1 (en) | 2004-06-14 | 2009-11-11 | Anacor Pharmaceuticals, Inc. | Anti-viral uses of borinic acid complexes |
| US7767657B2 (en) | 2005-02-16 | 2010-08-03 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| ES2872962T3 (es) | 2005-02-16 | 2021-11-03 | Anacor Pharmaceuticals Inc | Boronoftalidas para uso terapéutico |
| MX2007011486A (es) * | 2005-03-24 | 2007-11-20 | Anacor Pharmaceuticals Inc | Formulaciones topicas de antibioticos de acido borinico y sus metodos de uso. |
| EP1965647A2 (en) * | 2005-12-28 | 2008-09-10 | Anacor Pharmaceuticals, Inc. | Process for manufacturing picolinate borinic esters |
| RU2642628C2 (ru) | 2006-02-16 | 2018-01-25 | Анакор Фармасьютикалз, Инк. | Бор-содержащие малые молекулы в качестве противовоспалительных средств |
| US20070286822A1 (en) * | 2006-06-12 | 2007-12-13 | Anacor Pharmaceuticals Inc. | Compounds for the Treatment of Periodontal Disease |
| BRPI0713010A2 (pt) * | 2006-06-12 | 2012-10-09 | Anacor Pharmaceuticals Inc | compostos para o tratamento de doença periodontal |
| EP2069370A4 (en) * | 2006-11-22 | 2011-05-04 | Anacor Pharmaceuticals Inc | MICRO-ORGANISMS KILLING COMPOUNDS |
| EP3246034A1 (en) | 2008-03-06 | 2017-11-22 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-inflammatory agents |
| US20100256092A1 (en) * | 2008-05-12 | 2010-10-07 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2010027975A1 (en) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| US8461336B2 (en) | 2008-09-04 | 2013-06-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| US9493489B2 (en) | 2008-10-15 | 2016-11-15 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agents |
| SG172040A1 (en) * | 2008-12-17 | 2011-07-28 | Anacor Pharmaceuticals Inc | Polymorphs of (s)-3-aminomethyl-7-(3-hydroxy-propoxy)-3h-benzo[c][1,2] oxaborol-1-ol |
| EP2458995A1 (en) | 2009-07-28 | 2012-06-06 | Anacor Pharmaceuticals, Inc. | Trisubstituted boron-containing molecules |
| AP4039A (en) | 2009-08-14 | 2017-02-28 | Daitao Chen | Boron-containing small molecules as antiprotozoal agents |
| US20110207701A1 (en) * | 2009-08-19 | 2011-08-25 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| US20110124597A1 (en) * | 2009-09-25 | 2011-05-26 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules |
| WO2011049971A1 (en) | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| US8461134B2 (en) * | 2009-11-11 | 2013-06-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| US8716478B2 (en) | 2010-01-27 | 2014-05-06 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2011116348A1 (en) | 2010-03-19 | 2011-09-22 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agent |
| DK2613788T3 (en) | 2010-09-07 | 2017-08-07 | Anacor Pharmaceuticals Inc | BENZOXABOROLD DERIVATIVES FOR TREATMENT OF BACTERIA INFECTIONS |
| US8669207B1 (en) | 2013-01-30 | 2014-03-11 | Dow Agrosciences, Llc. | Compounds and compositions |
| AR094666A1 (es) | 2013-01-30 | 2015-08-19 | Dow Agrosciences Llc | Uso de benzoxaborolas como agentes antimicrobianos volátiles en carnes, plantas o partes de plantas |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| US9585396B2 (en) | 2013-01-30 | 2017-03-07 | Agrofresh Inc. | Volatile applications against pathogens |
| BR112016003692B1 (pt) * | 2013-08-20 | 2022-02-08 | 3M Innovative Properties Company | Complexo poliéter boro-silano |
| KR101756785B1 (ko) * | 2015-03-10 | 2017-07-12 | 한국화학연구원 | 4배위 유기 붕소 화합물의 제조방법 |
| WO2017155879A1 (en) | 2016-03-07 | 2017-09-14 | Agrofresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| US11447506B2 (en) | 2016-05-09 | 2022-09-20 | Anacor Pharmaceuticals, Inc. | Crystal forms of crisaborole in free form and preparation method and use thereof |
| IL248150B (en) | 2016-09-29 | 2018-05-31 | Garti Nissim | Method for selective extraction of cannabinoids from a plant source |
| IL248149B (en) | 2016-09-29 | 2020-03-31 | Garti Nissim | Dilutable formulations of cannbinoids and processes for their preparation |
| EP3522892A4 (en) * | 2016-10-05 | 2020-05-13 | The Global Alliance for TB Drug Development, Inc. | HETEROARYL TRIFLUORBORATE COMPOUNDS FOR TREATING MYCOBACTERIAL INFECTIONS |
| US10961261B2 (en) | 2017-03-01 | 2021-03-30 | Anacor Pharmaceuticals, Inc. | Oxaborole analogs and uses thereof |
| CA3054138A1 (en) * | 2017-03-09 | 2018-09-13 | The Penn State Research Foundation | Boron-containing small molecules for inhibiting activity of a receptor-like protein tyrosine phosphatase |
| EP3840637B1 (en) * | 2018-08-20 | 2025-08-06 | Senseonics, Incorporated | Mediated drug release for reducing in vivo analyte indicator degradation |
| WO2022043936A1 (en) | 2020-08-31 | 2022-03-03 | Pfizer Inc. | Methods of protecting rna |
| US12357552B2 (en) | 2021-03-09 | 2025-07-15 | Juris GERMANAS | Hydroxyquinoline compounds and methods of use as pigment modifying agents |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0496757B1 (de) * | 1989-10-18 | 1995-07-12 | Hoechst Schering AgrEvo GmbH | Verfahren zur bekämpfung von schadpflanzen in reis |
| US5348947A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | Diarylboron ester and thioester fungicidal agents |
| US5348948A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | 2,2-diaryl-1-(oxa and thia)-2a-azonia-2-borataacenaphthene fungicidal |
| JPH0952893A (ja) * | 1995-08-10 | 1997-02-25 | Yoshitomi Pharmaceut Ind Ltd | キノロンカルボン酸誘導体の工業的な製造法およびその合成中間体 |
| DE19829947A1 (de) * | 1998-07-04 | 2000-01-05 | Bayer Ag | Elektrolumineszierende Anordnungen mit Bor-Chelaten |
| EP1155698A4 (en) * | 1999-01-29 | 2003-01-15 | Nitto Kasei Co Ltd | ORGANOBORAL COMPOUNDS HAVING COCCIDIOSTAT ACTIVITY |
| CN1370170A (zh) * | 1999-05-25 | 2002-09-18 | 宾夕法尼亚州研究基金会 | Dna甲基转移酶抑制剂 |
| DE10110051C2 (de) * | 2001-03-02 | 2003-07-03 | Clariant Gmbh | Verfahren zur Herstellung von Boron- und Borinsäuren |
| JP2002322007A (ja) * | 2001-04-27 | 2002-11-08 | Shionogi & Co Ltd | 有機ホウ素化合物を含有する植物用殺線虫剤 |
| CN1325504C (zh) * | 2002-01-10 | 2007-07-11 | 宾夕法尼亚州研究基金会 | 制备二芳基硼酸烷基酯和络合的二芳基硼酸的方法 |
| MXPA05006685A (es) * | 2002-12-18 | 2005-12-14 | Anacor Pharmaceuticals Inc | Antibioticos que contienen complejos de acido borinico y metodos de uso. |
| US7390806B2 (en) * | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
-
2003
- 2003-12-18 MX MXPA05006685A patent/MXPA05006685A/es active IP Right Grant
- 2003-12-18 CN CN2010101656749A patent/CN101928295A/zh active Pending
- 2003-12-18 AU AU2003299821A patent/AU2003299821B2/en not_active Ceased
- 2003-12-18 KR KR1020057011194A patent/KR20050084378A/ko not_active Ceased
- 2003-12-18 EP EP03800095A patent/EP1581500A4/en not_active Withdrawn
- 2003-12-18 JP JP2005502662A patent/JP2006511613A/ja not_active Withdrawn
- 2003-12-18 US US10/740,304 patent/US20040224923A1/en not_active Abandoned
- 2003-12-18 WO PCT/US2003/040982 patent/WO2004056322A2/en not_active Ceased
- 2003-12-18 NZ NZ540870A patent/NZ540870A/en not_active IP Right Cessation
- 2003-12-18 CA CA002509645A patent/CA2509645A1/en not_active Abandoned
- 2003-12-18 EP EP08155302A patent/EP1980564A1/en not_active Withdrawn
- 2003-12-18 BR BR0317564-2A patent/BR0317564A/pt not_active IP Right Cessation
-
2007
- 2007-09-06 US US11/851,259 patent/US20080146803A1/en not_active Abandoned
-
2009
- 2009-02-02 JP JP2009021716A patent/JP2009161540A/ja not_active Withdrawn