JP2009161540A5 - - Google Patents
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- Publication number
- JP2009161540A5 JP2009161540A5 JP2009021716A JP2009021716A JP2009161540A5 JP 2009161540 A5 JP2009161540 A5 JP 2009161540A5 JP 2009021716 A JP2009021716 A JP 2009021716A JP 2009021716 A JP2009021716 A JP 2009021716A JP 2009161540 A5 JP2009161540 A5 JP 2009161540A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- unsubstituted
- alkoxy
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 125000000217 alkyl group Chemical group 0.000 claims 7
- 125000003545 alkoxy group Chemical group 0.000 claims 3
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 2
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 claims 2
- 229910052736 halogen Inorganic materials 0.000 claims 2
- 150000002367 halogens Chemical class 0.000 claims 2
- 229910052760 oxygen Inorganic materials 0.000 claims 2
- 239000001301 oxygen Substances 0.000 claims 2
- ZOXJGFHDIHLPTG-UHFFFAOYSA-N Boron Chemical group [B] ZOXJGFHDIHLPTG-UHFFFAOYSA-N 0.000 claims 1
- 125000000304 alkynyl group Chemical group 0.000 claims 1
- 125000004104 aryloxy group Chemical group 0.000 claims 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 1
- 229910052796 boron Inorganic materials 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 150000002431 hydrogen Chemical class 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 claims 1
- 229920002554 vinyl polymer Polymers 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43437502P | 2002-12-18 | 2002-12-18 | |
| US43609502P | 2002-12-23 | 2002-12-23 | |
| US43784903P | 2003-01-03 | 2003-01-03 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Division JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009161540A JP2009161540A (ja) | 2009-07-23 |
| JP2009161540A5 true JP2009161540A5 (enExample) | 2011-03-17 |
Family
ID=32686073
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Withdrawn JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
| JP2009021716A Withdrawn JP2009161540A (ja) | 2002-12-18 | 2009-02-02 | ボロン酸複合体を含む抗生物質および使用法 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2005502662A Withdrawn JP2006511613A (ja) | 2002-12-18 | 2003-12-18 | ボロン酸複合体を含む抗生物質および使用法 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20040224923A1 (enExample) |
| EP (2) | EP1581500A4 (enExample) |
| JP (2) | JP2006511613A (enExample) |
| KR (1) | KR20050084378A (enExample) |
| CN (1) | CN101928295A (enExample) |
| AU (1) | AU2003299821B2 (enExample) |
| BR (1) | BR0317564A (enExample) |
| CA (1) | CA2509645A1 (enExample) |
| MX (1) | MXPA05006685A (enExample) |
| NZ (1) | NZ540870A (enExample) |
| WO (1) | WO2004056322A2 (enExample) |
Families Citing this family (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2473238A1 (en) | 2002-01-10 | 2003-07-24 | The Penn State Research Foundation | Methods for the preparation of alkyl diaryl borinates and complexed diarylboronic acids |
| US7390806B2 (en) * | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
| CA2509645A1 (en) * | 2002-12-18 | 2004-07-08 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
| AR049915A1 (es) * | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Compuestos con contenido de boro y metodos de uso de los mismos |
| AR049916A1 (es) * | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Usos anti-parasitarios de complejos de acido borinico |
| US7393856B2 (en) | 2004-06-14 | 2008-07-01 | Anacor Pharmaceuticals, Inc. | Anti-viral uses of borinic acid complexes |
| AU2006214247C1 (en) | 2005-02-16 | 2012-11-08 | Anacor Pharmaceuticals, Llc | Boron-containing small molecules |
| US20060217347A1 (en) * | 2005-03-24 | 2006-09-28 | David Perry | Topical formulations of borinic acid antibiotics and their methods of use |
| WO2007079119A2 (en) * | 2005-12-28 | 2007-07-12 | Anacor Pharmaceuticals, Inc. | Process for manufacturing picolinate borinic esters |
| BRPI0621279B1 (pt) | 2005-12-30 | 2021-07-20 | Anacor Pharmaceuticals, Inc | Moléculas pequenas contendo boro |
| CA2642583C (en) | 2006-02-16 | 2016-08-23 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-inflammatory agents |
| WO2007146965A2 (en) * | 2006-06-12 | 2007-12-21 | Anacor Pharmaceuticals, Inc. | Compounds for the treatment of periodontal disease |
| US20070286822A1 (en) * | 2006-06-12 | 2007-12-13 | Anacor Pharmaceuticals Inc. | Compounds for the Treatment of Periodontal Disease |
| WO2008064345A2 (en) * | 2006-11-22 | 2008-05-29 | Anacor Pharmaceuticals, Inc. | Microorganism killing compounds |
| CN102014927A (zh) | 2008-03-06 | 2011-04-13 | 安纳考尔医药公司 | 作为抗炎药的含硼的小分子 |
| EP2285384A4 (en) * | 2008-05-12 | 2012-04-25 | Anacor Pharmaceuticals Inc | BORN SMALL MOLECULES |
| WO2010028005A1 (en) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2010027975A1 (en) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| US9493489B2 (en) | 2008-10-15 | 2016-11-15 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agents |
| AU2009335744A1 (en) * | 2008-12-17 | 2010-07-15 | Anacor Pharmaceuticals, Inc. | Polymorphs of (S)-3-aminomethyl-7-(3-hydroxy-propoxy) -3H-benzo[c][1,2] oxaborol-1-ol |
| JP2013500974A (ja) * | 2009-07-28 | 2013-01-10 | アナコール ファーマシューティカルズ，インコーポレイテッド | 三置換ホウ素含有分子 |
| AP4039A (en) | 2009-08-14 | 2017-02-28 | Daitao Chen | Boron-containing small molecules as antiprotozoal agents |
| MX2012002031A (es) * | 2009-08-19 | 2012-07-04 | Anacor Pharmaceuticals Inc | Moleculas pequeñas que contienen boro como agentes antiprotozoarios. |
| US20110124597A1 (en) * | 2009-09-25 | 2011-05-26 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules |
| US9346834B2 (en) | 2009-10-20 | 2016-05-24 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| WO2011060199A1 (en) * | 2009-11-11 | 2011-05-19 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2011094450A1 (en) | 2010-01-27 | 2011-08-04 | Anacor Pharmaceuticals, Inc | Boron-containing small molecules |
| WO2011116348A1 (en) | 2010-03-19 | 2011-09-22 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agent |
| SMT202100643T1 (it) | 2010-09-07 | 2022-01-10 | Anacor Pharmaceuticals Inc | Derivati del benzossaborolo per il trattamento delle infezioni batteriche |
| US8669207B1 (en) | 2013-01-30 | 2014-03-11 | Dow Agrosciences, Llc. | Compounds and compositions |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| EP2950644B1 (en) | 2013-01-30 | 2017-07-19 | AgroFresh Inc. | Use of benzoxaboroles as volatile antimicrobial agents on meats, plants, or plant parts |
| US9585396B2 (en) | 2013-01-30 | 2017-03-07 | Agrofresh Inc. | Volatile applications against pathogens |
| WO2015026548A1 (en) * | 2013-08-20 | 2015-02-26 | 3M Innovative Properties Company | Boron-silane polyether complex |
| KR101756785B1 (ko) * | 2015-03-10 | 2017-07-12 | 한국화학연구원 | 4배위 유기 붕소 화합물의 제조방법 |
| EP3426029B1 (en) | 2016-03-07 | 2023-08-30 | AgroFresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| US11447506B2 (en) | 2016-05-09 | 2022-09-20 | Anacor Pharmaceuticals, Inc. | Crystal forms of crisaborole in free form and preparation method and use thereof |
| IL248149B (en) | 2016-09-29 | 2020-03-31 | Garti Nissim | Formulations of dilutable cannabinoids and processes for their preparation |
| IL248150B (en) | 2016-09-29 | 2018-05-31 | Garti Nissim | A method for selective extraction of cannabinoid from plant origin |
| KR102465919B1 (ko) | 2016-10-05 | 2022-11-10 | 더 글로벌 얼라이언스 포 티비 드러그 디벨롭먼트, 잉크. | 미코박테리아 감염의 치료를 위한 헤테로아릴트리플루오로보레이트 화합물 |
| MA52337A (fr) | 2017-03-01 | 2021-03-03 | Anacor Pharmaceuticals Inc | Nouveaux analogues d'oxaborole et utilisations de ces derniers |
| AU2018230580A1 (en) * | 2017-03-09 | 2019-09-19 | The Penn State Research Foundation | Boron-containing small molecules for inhibiting activity of a receptor-like protein tyrosine phosphatase |
| CA3110179A1 (en) * | 2018-08-20 | 2020-02-27 | Senseonics, Incorporated | Mediated drug release for reducing in vivo analyte indicator degradation |
| US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
| US12357552B2 (en) | 2021-03-09 | 2025-07-15 | Juris GERMANAS | Hydroxyquinoline compounds and methods of use as pigment modifying agents |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR950012756B1 (ko) * | 1989-10-18 | 1995-10-21 | 훽스트 아크티엔게젤샤프트 | 벼의 잡초의 방제방법 |
| US5348947A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | Diarylboron ester and thioester fungicidal agents |
| US5348948A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | 2,2-diaryl-1-(oxa and thia)-2a-azonia-2-borataacenaphthene fungicidal |
| JPH0952893A (ja) * | 1995-08-10 | 1997-02-25 | Yoshitomi Pharmaceut Ind Ltd | キノロンカルボン酸誘導体の工業的な製造法およびその合成中間体 |
| DE19829947A1 (de) * | 1998-07-04 | 2000-01-05 | Bayer Ag | Elektrolumineszierende Anordnungen mit Bor-Chelaten |
| WO2000044387A1 (fr) * | 1999-01-29 | 2000-08-03 | Nitto Kasei Co., Ltd. | Composes organobores presentant une activite de coccidiostats |
| CN1370170A (zh) * | 1999-05-25 | 2002-09-18 | 宾夕法尼亚州研究基金会 | Dna甲基转移酶抑制剂 |
| DE10110051C2 (de) * | 2001-03-02 | 2003-07-03 | Clariant Gmbh | Verfahren zur Herstellung von Boron- und Borinsäuren |
| JP2002322007A (ja) * | 2001-04-27 | 2002-11-08 | Shionogi & Co Ltd | 有機ホウ素化合物を含有する植物用殺線虫剤 |
| CA2473238A1 (en) * | 2002-01-10 | 2003-07-24 | The Penn State Research Foundation | Methods for the preparation of alkyl diaryl borinates and complexed diarylboronic acids |
| CA2509645A1 (en) * | 2002-12-18 | 2004-07-08 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
| US7390806B2 (en) * | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
-
2003
- 2003-12-18 CA CA002509645A patent/CA2509645A1/en not_active Abandoned
- 2003-12-18 NZ NZ540870A patent/NZ540870A/en not_active IP Right Cessation
- 2003-12-18 BR BR0317564-2A patent/BR0317564A/pt not_active IP Right Cessation
- 2003-12-18 KR KR1020057011194A patent/KR20050084378A/ko not_active Ceased
- 2003-12-18 EP EP03800095A patent/EP1581500A4/en not_active Withdrawn
- 2003-12-18 JP JP2005502662A patent/JP2006511613A/ja not_active Withdrawn
- 2003-12-18 MX MXPA05006685A patent/MXPA05006685A/es active IP Right Grant
- 2003-12-18 AU AU2003299821A patent/AU2003299821B2/en not_active Ceased
- 2003-12-18 EP EP08155302A patent/EP1980564A1/en not_active Withdrawn
- 2003-12-18 US US10/740,304 patent/US20040224923A1/en not_active Abandoned
- 2003-12-18 WO PCT/US2003/040982 patent/WO2004056322A2/en not_active Ceased
- 2003-12-18 CN CN2010101656749A patent/CN101928295A/zh active Pending
-
2007
- 2007-09-06 US US11/851,259 patent/US20080146803A1/en not_active Abandoned
-
2009
- 2009-02-02 JP JP2009021716A patent/JP2009161540A/ja not_active Withdrawn