JP2008543780A - グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 - Google Patents

グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 Download PDF

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JP2008543780A
JP2008543780A JP2008515997A JP2008515997A JP2008543780A JP 2008543780 A JP2008543780 A JP 2008543780A JP 2008515997 A JP2008515997 A JP 2008515997A JP 2008515997 A JP2008515997 A JP 2008515997A JP 2008543780 A JP2008543780 A JP 2008543780A
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indazol
trifluoro
fluorophenyl
propan
phenyl
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JP2008543780A5 (https=
Inventor
インゴ アンドレアス ムゲ
マイケル ジェイソン バーク
マーク スティーブン ラルフ
ディヴィッド エス トムソン
アブデルハキム ハムマック
ジェニファー エイ コワルスキー
ヨルグ マルティン ベンツィエン
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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  • Chemical & Material Sciences (AREA)
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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Otolaryngology (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
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JP2008515997A 2005-06-10 2006-06-08 グルココルチコイド模倣薬、それらの製造方法、医薬組成物及びそれらの使用 Pending JP2008543780A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68941205P 2005-06-10 2005-06-10
PCT/US2006/022651 WO2006135826A1 (en) 2005-06-10 2006-06-08 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

Publications (2)

Publication Number Publication Date
JP2008543780A true JP2008543780A (ja) 2008-12-04
JP2008543780A5 JP2008543780A5 (https=) 2009-08-13

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US (1) US7622594B2 (https=)
EP (1) EP1893588A1 (https=)
JP (1) JP2008543780A (https=)
KR (1) KR20080027828A (https=)
CN (1) CN101193869B (https=)
AR (1) AR058006A1 (https=)
AU (1) AU2006257861A1 (https=)
BR (1) BRPI0611620A2 (https=)
CA (1) CA2610588A1 (https=)
IL (1) IL187976A0 (https=)
MX (1) MX2007014811A (https=)
NZ (1) NZ564696A (https=)
PE (1) PE20070112A1 (https=)
RU (1) RU2007148225A (https=)
TW (1) TW200716573A (https=)
WO (1) WO2006135826A1 (https=)
ZA (1) ZA200709430B (https=)

Cited By (1)

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Publication number Priority date Publication date Assignee Title
JP2023535279A (ja) * 2020-06-22 2023-08-17 コーセプト セラピューティクス， インコーポレイテッド ４級インダゾールグルココルチコイド受容体アンタゴニスト

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WO2004019935A1 (en) * 2002-08-29 2004-03-11 Boehringer Ingelheim Pharmaceuticals, Inc. -3 (sulfonamidoethyl) -indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
UY28526A1 (es) * 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos
US7795272B2 (en) 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
CA2592514A1 (en) * 2004-12-27 2006-07-06 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
EP2061767B1 (de) 2006-08-08 2014-12-17 Sanofi Arylaminoaryl-alkyl-substituierte Imidazolidin-2,4-dione, Verfahren zu ihrer Herstellung, diese Verbindungen enthaltende Arzneimittel und ihre Verwendung
WO2008057857A1 (en) * 2006-11-01 2008-05-15 Bristol-Myers Squibb Company MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-ϰB ACTIVITY AND USE THEREOF
TW200829578A (en) 2006-11-23 2008-07-16 Astrazeneca Ab Chemical compounds 537
AU2007329548A1 (en) * 2006-12-06 2008-06-12 Boehringer Ingelheim International Gmbh Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
JO2754B1 (en) * 2006-12-21 2014-03-15 استرازينكا ايه بي Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders
WO2008079073A1 (en) * 2006-12-22 2008-07-03 Astrazeneca Ab Indazolyl sulphonamide derivatives for the treatment of glucocorticoid receptor mediated disorders
MX2009008439A (es) * 2007-02-12 2009-08-13 Intermune Inc Nuevos inhibidores de la replicacion del virus de hepatitis c.
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