JP2008540626A5 - - Google Patents
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- Publication number
- JP2008540626A5 JP2008540626A5 JP2008511793A JP2008511793A JP2008540626A5 JP 2008540626 A5 JP2008540626 A5 JP 2008540626A5 JP 2008511793 A JP2008511793 A JP 2008511793A JP 2008511793 A JP2008511793 A JP 2008511793A JP 2008540626 A5 JP2008540626 A5 JP 2008540626A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- compound
- amino
- substituted
- carbocyclic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68268705P | 2005-05-19 | 2005-05-19 | |
| GB0510252A GB0510252D0 (en) | 2005-05-19 | 2005-05-19 | Pharmaceutical compounds |
| PCT/GB2006/001851 WO2006123165A2 (en) | 2005-05-19 | 2006-05-19 | Pyrimidine derivatives as hsp90 inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008540626A JP2008540626A (ja) | 2008-11-20 |
| JP2008540626A5 true JP2008540626A5 (https=) | 2009-07-09 |
Family
ID=37431622
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008511793A Pending JP2008540626A (ja) | 2005-05-19 | 2006-05-19 | 医薬化合物 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20090215777A1 (https=) |
| EP (1) | EP2049497A2 (https=) |
| JP (1) | JP2008540626A (https=) |
| WO (1) | WO2006123165A2 (https=) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102006008880A1 (de) * | 2006-02-27 | 2007-09-06 | Merck Patent Gmbh | Aminopyrimidinderivate |
| AR061185A1 (es) | 2006-05-26 | 2008-08-13 | Chugai Pharmaceutical Co Ltd | Compuestos heterociclicos como inhibidores de hsp90. composiciones farmaceuticas. |
| CL2008000467A1 (es) | 2007-02-14 | 2008-08-22 | Janssen Pharmaceutica Nv | Compuestos derivados de 2-aminopirimidina, moduladores del receptor histamina h4; su procedimiento de preparacion; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar un trastorno inflamatorio seleccionado de alegia, asma |
| MX2009008756A (es) | 2007-03-01 | 2009-08-27 | Chugai Pharmaceutical Co Ltd | Compuesto macrociclico. |
| EP2155694B1 (en) * | 2007-03-27 | 2012-01-04 | Synta Pharmaceuticals Corp. | Triazinone and diazinone derivatives useful as hsp90 inhibitors |
| KR100965726B1 (ko) | 2007-11-23 | 2010-06-24 | 재단법인서울대학교산학협력재단 | 피리미딘-2,4,6-트라이온 유도체를 함유하는 Hsp90억제제 및 이를 이용한 항암제 |
| WO2009086277A1 (en) | 2007-12-20 | 2009-07-09 | Envivo Pharmaceuticals, Inc. | Tetrasubstituted benzenes |
| MX353308B (es) | 2008-05-21 | 2018-01-08 | Ariad Pharma Inc | Derivados fosforosos como inhibidores de cinasa. |
| US9273077B2 (en) | 2008-05-21 | 2016-03-01 | Ariad Pharmaceuticals, Inc. | Phosphorus derivatives as kinase inhibitors |
| UY32582A (es) | 2009-04-28 | 2010-11-30 | Amgen Inc | Inhibidores de fosfoinositida 3 cinasa y/u objetivo mamífero |
| EP2704572B1 (en) | 2011-05-04 | 2015-12-30 | Ariad Pharmaceuticals, Inc. | Compounds for inhibiting cell proliferation in egfr-driven cancers |
| WO2013169401A1 (en) | 2012-05-05 | 2013-11-14 | Ariad Pharmaceuticals, Inc. | Compounds for inhibiting cell proliferation in egfr-driven cancers |
| EP2972394A4 (en) | 2013-03-15 | 2016-11-02 | Sloan Kettering Inst Cancer | HSP90-DESIGNING AND THERAPY |
| US9611283B1 (en) | 2013-04-10 | 2017-04-04 | Ariad Pharmaceuticals, Inc. | Methods for inhibiting cell proliferation in ALK-driven cancers |
| JP6779867B2 (ja) * | 2014-06-13 | 2020-11-04 | ユマ セラピューティクス,インコーポレーテッド | ピリミジン化合物およびその使用方法 |
| MX387627B (es) | 2014-09-17 | 2025-03-18 | Memorial Sloan Kettering Cancer Center | Formación de imágenes de inflamación e infección dirigida a hsp90 y terapia |
| PL3303330T3 (pl) * | 2015-06-03 | 2019-10-31 | Bristol Myers Squibb Co | Agoniści 4 - hydroksy - 3 - ( heteroarylo ) pirydyno - 2 - onowi receptora apj do stosowania w leczeniu zaburzeń sercowo-naczyniowych |
| CN115845818B (zh) * | 2022-12-13 | 2024-02-23 | 南京工业大学 | 一种木质素接枝n-[(二甲氨基)亚甲基]硫脲型重金属吸附剂及其制备方法与应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7439359B2 (en) * | 2000-11-02 | 2008-10-21 | Sloan-Kettering Institute For Cancer Research | Small molecule compositions for binding to hsp90 |
| WO2003075828A2 (en) * | 2002-03-11 | 2003-09-18 | Zetiq Technologies Ltd. | Compounds useful in the treatment of cancer |
| ES2273047T3 (es) * | 2002-10-28 | 2007-05-01 | Bayer Healthcare Ag | Fenilaminopirimidinas sustituidas con heteroariloxi como inhibidores de rho-cinasa. |
-
2006
- 2006-05-19 EP EP06727141A patent/EP2049497A2/en not_active Withdrawn
- 2006-05-19 WO PCT/GB2006/001851 patent/WO2006123165A2/en not_active Ceased
- 2006-05-19 JP JP2008511793A patent/JP2008540626A/ja active Pending
- 2006-05-19 US US11/914,728 patent/US20090215777A1/en not_active Abandoned
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