JP2008540573A - 4−ビアリーリル−1−フェニラゼチジン−2−オン類 - Google Patents

4−ビアリーリル−1−フェニラゼチジン−2−オン類 Download PDF

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JP2008540573A
JP2008540573A JP2008511448A JP2008511448A JP2008540573A JP 2008540573 A JP2008540573 A JP 2008540573A JP 2008511448 A JP2008511448 A JP 2008511448A JP 2008511448 A JP2008511448 A JP 2008511448A JP 2008540573 A JP2008540573 A JP 2008540573A
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group
lower alkyl
fluorophenyl
hydroxypropyl
phenyl
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Inventor
ステファン アントネッリ
ティモシー シー. バーデン
ブライアン カリ
マーク ジー. カリー
レジーナ ランドリガン−サウシー
ジンジン ヤン
ピーター エス. ヨーギー
ダニエル ピー. ジマー
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Microbia Inc
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Microbia Inc
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JP2008511448A 2005-05-13 2006-05-15 4−ビアリーリル−1−フェニラゼチジン−2−オン類 Pending JP2008540573A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US68123205P 2005-05-13 2005-05-13
US69598805P 2005-07-01 2005-07-01
PCT/US2006/018616 WO2006124713A2 (en) 2005-05-13 2006-05-15 4-biarylyl-1-phenylazetidin-2-ones

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JP2008540573A true JP2008540573A (ja) 2008-11-20

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EP (1) EP1885694A2 (de)
JP (1) JP2008540573A (de)
TW (1) TW200740752A (de)
WO (1) WO2006124713A2 (de)

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US10983108B2 (en) 2017-03-31 2021-04-20 Quest Diagnostics Investments Llc Methods for quantitation of insulin and C-peptide
US11486874B2 (en) 2015-03-03 2022-11-01 Quest Diagnostics Investments Llc Methods for quantitation of insulin levels by mass spectrometry

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US20060287254A1 (en) * 2001-01-26 2006-12-21 Schering Corporation Use of substituted azetidinone compounds for the treatment of sitosterolemia
US7871998B2 (en) 2003-12-23 2011-01-18 Astrazeneca Ab Diphenylazetidinone derivatives possessing cholesterol absorption inhibitory activity
UY29607A1 (es) 2005-06-20 2007-01-31 Astrazeneca Ab Compuestos quimicos
AR057072A1 (es) 2005-06-22 2007-11-14 Astrazeneca Ab Compuestos quimicos derivados de 2-azetidinona, formulacion farmaceutica y un proceso de preparacion del compuesto
SA06270191B1 (ar) 2005-06-22 2010-03-29 استرازينيكا ايه بي مشتقات من 2- أزيتيدينون جديدة باعتبارها مثبطات لامتصاص الكوليسترول لعلاج حالات فرط نسبة الدهون في الدم
AR060623A1 (es) 2006-04-27 2008-07-02 Astrazeneca Ab Compuestos derivados de 2-azetidinona y un metodo de preparacion
JO3598B1 (ar) 2006-10-10 2020-07-05 Infinity Discovery Inc الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني
WO2008061238A2 (en) * 2006-11-16 2008-05-22 Ironwood Pharmaceuticals, Inc. Processes for production of 4-biphenylyazetidin-2-ones
JPWO2008108486A1 (ja) 2007-03-06 2010-06-17 帝人ファーマ株式会社 1−ビアリールアゼチジノン誘導体
AR065850A1 (es) * 2007-03-28 2009-07-08 Takeda Pharmaceutical Composicion farmaceutica solida que comprende un derivado de benzimidazol-7-carboxilato y un agente de control de ph
TW201000107A (en) 2008-04-09 2010-01-01 Infinity Pharmaceuticals Inc Inhibitors of fatty acid amide hydrolase
CA2732018C (en) 2008-07-31 2017-07-04 Takeda Pharmaceutical Company Limited Solid pharmaceutical composition
WO2010118159A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
WO2010118155A1 (en) 2009-04-07 2010-10-14 Infinity Pharmaceuticals, Inc. Inhibitors of fatty acid amide hydrolase
CN102834401B (zh) 2010-02-03 2016-08-24 无限药品股份有限公司 脂肪酸酰胺水解酶抑制剂
EP2575821B1 (de) 2010-05-26 2015-08-12 Satiogen Pharmaceuticals, Inc. Gallensäurerückflusshemmer und satiogene zur behandlung von diabetes, adipositas und entzündlichen magen-darm-erkrankungen
CN102370648B (zh) * 2010-08-10 2013-05-29 山东新时代药业有限公司 一种药物组合物及其用途
EA029581B1 (ru) 2011-10-28 2018-04-30 ЛУМЕНА ФАРМАСЬЮТИКАЛС ЭлЭлСи Применение ингибиторов рециркуляции желчных кислот для лечения холестатического заболевания печени или прурита
CN107375932B (zh) 2011-10-28 2021-12-21 夏尔人类遗传性治疗公司 用于治疗小儿胆汁淤积性肝病的胆汁酸再循环抑制剂
CA2907230A1 (en) 2013-03-15 2014-09-18 Lumena Pharmaceuticals, Inc. Bile acid recycling inhibitors for treatment of primary sclerosing cholangitis and inflammatory bowel disease
EP2968262A1 (de) 2013-03-15 2016-01-20 Lumena Pharmaceuticals, Inc. Gallensäurerückflusshemmer zur behandlung von barrett-ösophagus und gastroösophagealem reflux
MX2021009622A (es) 2019-02-12 2021-11-04 Mirum Pharmaceuticals Inc Metodos para tratar la colestasis.
CN116023273A (zh) * 2023-03-29 2023-04-28 思合基因(北京)生物科技有限公司 一种新型碳糖苷及其制备方法

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