JP2008531715A - 統合失調症及び関連疾患の治療用及び/又は予防用の医薬組成物 - Google Patents

統合失調症及び関連疾患の治療用及び/又は予防用の医薬組成物 Download PDF

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JP2008531715A
JP2008531715A JP2007558203A JP2007558203A JP2008531715A JP 2008531715 A JP2008531715 A JP 2008531715A JP 2007558203 A JP2007558203 A JP 2007558203A JP 2007558203 A JP2007558203 A JP 2007558203A JP 2008531715 A JP2008531715 A JP 2008531715A
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antagonist
pharmaceutical composition
acid addition
schizophrenia
pharmaceutically acceptable
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JP2008531715A5 (enExample
Inventor
ロバート パイク
アンジェロ チェチ
Original Assignee
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/405Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
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    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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  • Animal Behavior & Ethology (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2007558203A 2005-03-04 2006-02-28 統合失調症及び関連疾患の治療用及び/又は予防用の医薬組成物 Pending JP2008531715A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65856605P 2005-03-04 2005-03-04
PCT/US2006/007379 WO2006096439A2 (en) 2005-03-04 2006-02-27 Pharmaceutical compositions for the treatment and/or prevention of schizophrenia and related diseases

Publications (2)

Publication Number Publication Date
JP2008531715A true JP2008531715A (ja) 2008-08-14
JP2008531715A5 JP2008531715A5 (enExample) 2009-04-16

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JP2007558203A Pending JP2008531715A (ja) 2005-03-04 2006-02-28 統合失調症及び関連疾患の治療用及び/又は予防用の医薬組成物

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US (1) US20060204486A1 (enExample)
EP (1) EP1858517A2 (enExample)
JP (1) JP2008531715A (enExample)
CA (1) CA2599699A1 (enExample)
WO (1) WO2006096439A2 (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
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JP2013533306A (ja) * 2010-08-10 2013-08-22 ルピン・リミテッド ブロナンセリン経口放出制御型医薬組成物

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