JP2008519056A - 特定の［１，４］ジアゼピノ［６，７，１−ｉｊ］キノリン誘導体の代謝物ならびにそれらの調製および使用方法 - Google Patents
特定の［１，４］ジアゼピノ［６，７，１−ｉｊ］キノリン誘導体の代謝物ならびにそれらの調製および使用方法 Download PDFInfo
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| US62533504P | 2004-11-05 | 2004-11-05 | |
| PCT/US2005/040289 WO2006052886A1 (en) | 2004-11-05 | 2005-11-04 | Metabolites of certain [1,4]diazepino[6,7,1-ij]quinoline derivatives and methods of preparation and use thereof |
Publications (2)
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| JP2008519056A true JP2008519056A (ja) | 2008-06-05 |
| JP2008519056A5 JP2008519056A5 (https=) | 2008-10-09 |
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| JP (1) | JP2008519056A (https=) |
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| BR (1) | BRPI0517100A (https=) |
| CA (1) | CA2586122A1 (https=) |
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| RU (1) | RU2007116264A (https=) |
| TW (1) | TW200635926A (https=) |
| WO (1) | WO2006052886A1 (https=) |
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| GT200500317A (es) * | 2004-11-05 | 2006-10-27 | Proceso para preparar compuestos de quinolina y productos obtenidos de los mismos | |
| AR054849A1 (es) * | 2005-07-26 | 2007-07-18 | Wyeth Corp | Diazepinoquinolinas, sintesis de las mismas, e intermediarios para obtenerlas |
| TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
| AU2007230997A1 (en) * | 2006-03-24 | 2007-10-04 | Wyeth | Treatment of pain |
| EP1998773A2 (en) * | 2006-03-24 | 2008-12-10 | Wyeth a Corporation of the State of Delaware | New therapeutic combinations for the treatment of depression |
| US20070225278A1 (en) * | 2006-03-24 | 2007-09-27 | Wyeth | Methods for treating cognitive and other disorders |
| CL2008002777A1 (es) * | 2007-09-21 | 2010-01-22 | Wyeth Corp | Metodo de preparacion de compuestos diazepinoquinolinicos quirales por recristalizacion en un sistema de solvente ternario. |
| WO2015066344A1 (en) | 2013-11-01 | 2015-05-07 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists and compositions and methods of use |
| CN111303218B (zh) * | 2020-03-17 | 2021-03-30 | 连江仁泽生物科技有限公司 | 一种马鞭草苷的合成方法及应用 |
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| US3714149A (en) * | 1969-11-03 | 1973-01-30 | Upjohn Co | Pyridobenzodiazepinones |
| WO1990015058A1 (en) * | 1989-06-09 | 1990-12-13 | The Upjohn Company | Heterocyclic amines having central nervous system activity |
| WO2003091251A1 (en) * | 2002-04-25 | 2003-11-06 | Wyeth | 1,2,3,4,7,8-hexahydro-6h-[1,4]diazepino[6,7,1-1j]quinoline derivatives as antipsychotic and antiobesity agents |
| WO2003091250A1 (en) * | 2002-04-25 | 2003-11-06 | Wyeth | [1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents |
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| US3158619A (en) * | 1962-06-14 | 1964-11-24 | Searle & Co | Certain sulfur-containing ortho-fused polycyclic pyrazole derivatives |
| US3235564A (en) * | 1964-03-27 | 1966-02-15 | Searle & Co | Intermediates to certain sulfur-containing ortho-fused polycyclic pyrazole derivatives |
| US3296252A (en) * | 1964-04-02 | 1967-01-03 | Sandoz Ag | Tetracyclic diazepinone compounds |
| US3335134A (en) * | 1964-04-02 | 1967-08-08 | Sandoz Ag | Certain 3, 4-dihydrofluoreno[1, 9a, 9-e, f]1, 4-diazepin-3(2h)-ones |
| GB1120463A (en) * | 1964-07-06 | 1968-07-17 | Manuf Prod Pharma | Derivatives of 1,3-diazafluoranthene-1-oxide |
| US3329676A (en) * | 1964-11-09 | 1967-07-04 | American Home Prod | Fused 1, 4-diazepine ring systems |
| US3417101A (en) * | 1964-11-09 | 1968-12-17 | American Home Prod | Fused ring compounds |
| US3914250A (en) * | 1974-08-01 | 1975-10-21 | American Home Prod | 1,4-Diazepino{8 6,5,4-jk{9 carbazoles |
| US4880814A (en) * | 1987-11-13 | 1989-11-14 | Abbott Laboratories | 7-cycloalkyl naphthyridines |
| GB8812636D0 (en) * | 1988-05-27 | 1988-06-29 | Glaxo Group Ltd | Chemical compounds |
| JPH02180885A (ja) * | 1988-09-01 | 1990-07-13 | Glaxo Group Ltd | ラクタム誘導体 |
| NZ314105A (en) * | 1996-02-02 | 1997-12-19 | Sumitomo Pharma | Guanidine derivative substituted with a substituted indole which is peri condensed with a heterocyclic ring |
| US6380166B1 (en) * | 1999-09-13 | 2002-04-30 | American Home Products Corporation | Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols |
| US6761904B2 (en) * | 2000-03-31 | 2004-07-13 | Nycomed Austria Gmbh | Pharmaceutical kit comprising midodrine as active drug substance |
| US6414144B1 (en) * | 2000-11-03 | 2002-07-02 | Wyeth | Process for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi] indole derivatives |
| US6916922B2 (en) * | 2000-11-03 | 2005-07-12 | Wyeth | Process for the preparation of 1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta [B] [1,4] diazepino- [6,7,1-hi] indole derivatives |
| AR031202A1 (es) * | 2000-11-03 | 2003-09-10 | Wyeth Corp | Ciclopenta(b) (1,4)diazepino(6,7,1-hi) indoles y derivados |
| US6759405B2 (en) * | 2000-11-03 | 2004-07-06 | Wyeth | Cycloocta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| AR031199A1 (es) * | 2000-11-03 | 2003-09-10 | Wyeth Corp | Ciclohepta/b//1,4/diacepino/6,7,1-hi/indoles y derivados |
| AR031197A1 (es) * | 2000-11-03 | 2003-09-10 | Wyeth Corp | Procedimiento para la preparacion de derivados de 1,2,3,4,8,9,10,10a-octahidro-7bh-ciclopenta(b) diazepino(6,7,1-hi)indol |
| US6784172B2 (en) * | 2000-11-03 | 2004-08-31 | Wyeth | Processes for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
| US6503900B2 (en) * | 2000-11-03 | 2003-01-07 | Wyeth | [1,4]diazepino [6,7,1-jk ]carbazoles and derivatives |
| SK7042003A3 (en) * | 2000-12-20 | 2004-07-07 | Bristol Myers Squibb Co | Substituted pyridoindoles as serotonin agonists and antagonists |
| MXPA04001202A (es) * | 2001-08-06 | 2005-02-17 | Pharmacia & Upjhon Company | Ligandos tetraciclicos terapeuticamente utiles. |
| TW200307540A (en) * | 2002-04-25 | 2003-12-16 | Wyeth Corp | [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents |
| WO2004056324A2 (en) * | 2002-12-19 | 2004-07-08 | Bristol-Myers Squibb Company | Substituted tricyclic gamma-carbolines as serotonin receptor agonists and antagonists |
| TW200734334A (en) * | 2006-01-13 | 2007-09-16 | Wyeth Corp | Treatment of substance abuse |
| US20070225278A1 (en) * | 2006-03-24 | 2007-09-27 | Wyeth | Methods for treating cognitive and other disorders |
-
2005
- 2005-11-03 TW TW094138587A patent/TW200635926A/zh unknown
- 2005-11-03 AR ARP050104611A patent/AR052227A1/es unknown
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- 2007-05-02 CR CR9092A patent/CR9092A/es not_active Application Discontinuation
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3714149A (en) * | 1969-11-03 | 1973-01-30 | Upjohn Co | Pyridobenzodiazepinones |
| WO1990015058A1 (en) * | 1989-06-09 | 1990-12-13 | The Upjohn Company | Heterocyclic amines having central nervous system activity |
| WO2003091251A1 (en) * | 2002-04-25 | 2003-11-06 | Wyeth | 1,2,3,4,7,8-hexahydro-6h-[1,4]diazepino[6,7,1-1j]quinoline derivatives as antipsychotic and antiobesity agents |
| WO2003091250A1 (en) * | 2002-04-25 | 2003-11-06 | Wyeth | [1,4]diazepino[6,7,1-ij]quinoline derivatives as anti psychotic and antiobesity agents |
| US20040009970A1 (en) * | 2002-04-25 | 2004-01-15 | Wyeth | [1,4]Diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1812436A1 (en) | 2007-08-01 |
| CN101124225A (zh) | 2008-02-13 |
| CR9092A (es) | 2007-10-23 |
| AR052227A1 (es) | 2007-03-07 |
| WO2006052886A1 (en) | 2006-05-18 |
| IL182755A0 (en) | 2007-07-24 |
| NO20072165L (no) | 2007-07-25 |
| WO2006052886A8 (en) | 2007-06-14 |
| AU2005304757A1 (en) | 2006-05-18 |
| BRPI0517100A (pt) | 2008-09-30 |
| GT200500319A (es) | 2006-06-02 |
| PE20060939A1 (es) | 2006-11-10 |
| CA2586122A1 (en) | 2006-05-18 |
| US20060111305A1 (en) | 2006-05-25 |
| RU2007116264A (ru) | 2008-12-10 |
| TW200635926A (en) | 2006-10-16 |
| KR20070084009A (ko) | 2007-08-24 |
| MX2007005475A (es) | 2007-05-24 |
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