JP2008508188A5 - - Google Patents

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Publication number
JP2008508188A5
JP2008508188A5 JP2007504792A JP2007504792A JP2008508188A5 JP 2008508188 A5 JP2008508188 A5 JP 2008508188A5 JP 2007504792 A JP2007504792 A JP 2007504792A JP 2007504792 A JP2007504792 A JP 2007504792A JP 2008508188 A5 JP2008508188 A5 JP 2008508188A5
Authority
JP
Japan
Prior art keywords
thiazol
ethyl
phenyl
amino
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2007504792A
Other languages
English (en)
Japanese (ja)
Other versions
JP4978464B2 (ja
JP2008508188A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/JP2005/014136 external-priority patent/WO2006011631A2/en
Publication of JP2008508188A publication Critical patent/JP2008508188A/ja
Publication of JP2008508188A5 publication Critical patent/JP2008508188A5/ja
Application granted granted Critical
Publication of JP4978464B2 publication Critical patent/JP4978464B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2007504792A 2004-07-27 2005-07-27 Ｖａｐ−１阻害剤活性を有するチアゾール誘導体 Expired - Fee Related JP4978464B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AU2004904196A AU2004904196A0 (en) 2004-07-27 Thiazole Derivatives Having VAP-1 Inhibitory Activity
AU2004904196 2004-07-27
PCT/JP2005/014136 WO2006011631A2 (en) 2004-07-27 2005-07-27 Thiazole derivatives having vap-1 inhibitory activity

Publications (3)

Publication Number Publication Date
JP2008508188A JP2008508188A (ja) 2008-03-21
JP2008508188A5 true JP2008508188A5 (cg-RX-API-DMAC7.html) 2008-08-14
JP4978464B2 JP4978464B2 (ja) 2012-07-18

Family

ID=35734947

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007504792A Expired - Fee Related JP4978464B2 (ja) 2004-07-27 2005-07-27 Ｖａｐ−１阻害剤活性を有するチアゾール誘導体

Country Status (10)

Country Link
US (1) US20070254931A1 (cg-RX-API-DMAC7.html)
EP (1) EP1786792B1 (cg-RX-API-DMAC7.html)
JP (1) JP4978464B2 (cg-RX-API-DMAC7.html)
KR (1) KR20070050932A (cg-RX-API-DMAC7.html)
CN (1) CN101031555A (cg-RX-API-DMAC7.html)
AT (1) ATE427941T1 (cg-RX-API-DMAC7.html)
CA (1) CA2575411A1 (cg-RX-API-DMAC7.html)
DE (1) DE602005013793D1 (cg-RX-API-DMAC7.html)
ES (1) ES2324922T3 (cg-RX-API-DMAC7.html)
WO (1) WO2006011631A2 (cg-RX-API-DMAC7.html)

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JP5369257B2 (ja) 2006-02-15 2013-12-18 アッヴィ・インコーポレイテッド 新規なアセチル−ＣｏＡカルボキシラーゼ（ＡＣＣ）阻害薬およびそれらの糖尿病、肥満および代謝症候群での使用
CA2641766A1 (en) * 2006-02-15 2007-08-23 Abbott Laboratories Novel acetyl-coa carboxylase (acc) inhibitors and their use in diabetes, obesity and metabolic syndrome
TW200913999A (en) 2007-06-25 2009-04-01 R Tech Ueno Ltd Composition for eye diseases acompany hypoxia or ischemia
CN103120690A (zh) * 2007-10-19 2013-05-29 株式会社·R-技术上野 用于治疗白内障的药物组合物
WO2009061830A1 (en) * 2007-11-06 2009-05-14 Massachusetts Eye & Ear Infirmary Methods and compositions for treating conditions associated with angiogenesis using a vascular adhesion protein-1 (vap-1) inhibitor
EP2240468B1 (en) * 2008-01-18 2013-10-16 Allergan, Inc. Selective subtype alpha 2 adrenergic agents and methods for use thereof
TWI437986B (zh) 2008-01-31 2014-05-21 R Tech Ueno Ltd 噻唑衍生物及使用該衍生物作為ｖａｐ－１抑制劑之用途
TWI490214B (zh) * 2008-05-30 2015-07-01 艾德克 上野股份有限公司 苯或噻吩衍生物及該等作為ｖａｐ－１抑制劑之用途
NZ592603A (en) * 2008-10-21 2013-02-22 Metabolex Inc Aryl gpr120 receptor agonists and uses thereof
UA112154C2 (uk) 2009-09-08 2016-08-10 Біоті Терапіс Корп. Застосування повністю людського анти-vap-1-антитіла для лікування фіброзних станів
FI20115234A0 (fi) 2011-03-08 2011-03-08 Biotie Therapies Corp Uusia pyridatsinoni- ja pyridoniyhdisteitä
UA110515C2 (ru) 2011-03-15 2016-01-12 Astellas Pharma Inc Гуанідинова сполука
WO2013057944A1 (ja) 2011-10-19 2013-04-25 興和株式会社 新規なスピロインドリン化合物、及びそれを含有する医薬
CA2915163A1 (en) 2013-06-12 2014-12-18 Proximagen Limited New therapeutic uses of enzyme inhibitors
HUE042625T2 (hu) 2014-04-15 2019-07-29 Pecsi Tudomanyegyetem Szemikarbazid-szenzitiv amin-oxidáz gátlók fájdalomcsillapítóként való alkalmazásra traumás neuropátiában és neurogén gyulladásban
WO2015189534A1 (en) 2014-06-12 2015-12-17 Proximagen Limited Vap-1 inhibitors for treating muscular dystrophy
CN104478828B (zh) * 2014-12-10 2016-07-06 漳州片仔癀药业股份有限公司 2-氨基-7-取代苯并噻唑类化合物及其制备方法与用途
JOP20200093A1 (ar) 2015-01-09 2017-06-16 Kyowa Kirin Co Ltd طريقة لإنتاج مشتق ثيازول
JP2018076236A (ja) 2015-06-05 2018-05-17 株式会社アールテック・ウエノ がんを処置するための医薬組成物
EP3333163A4 (en) 2015-08-06 2019-01-09 UBE Industries, Ltd. SUBSTITUTED GUANIDINE DERIVATIVE
AU2016366635A1 (en) 2015-12-07 2018-06-21 Benevolentai Cambridge Limited VAP-1 inhibitors for treating pain
KR20190003995A (ko) * 2016-05-12 2019-01-10 베링거 인겔하임 인터내셔날 게엠베하 피리디닐 유도체, 약제학적 조성물 및 이의 aoc3 저해제로서의 용도
KR102607007B1 (ko) * 2016-12-28 2023-11-29 유비이 가부시키가이샤 치환 구아니딘 화합물
US10213306B2 (en) 2017-03-31 2019-02-26 Neochord, Inc. Minimally invasive heart valve repair in a beating heart

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US4699928A (en) * 1984-07-13 1987-10-13 Merrell Dow Pharmaceuticals Inc. Fluoroallylamine derivatives
IT1181871B (it) * 1985-04-01 1987-09-30 Consiglio Nazionale Ricerche Inibitori selettivi delle benzilamminossidasi rispetto ad altre amminossidasi
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US4650907A (en) * 1985-12-05 1987-03-17 Merrell Dow Pharmaceuticals Inc. Nonaromatic fluoroallylamine MAO inhibitors
US5021456A (en) * 1988-02-25 1991-06-04 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
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US4943593A (en) * 1988-02-25 1990-07-24 Merrell Dow Pharmaceuticals Inc. Inhibitors of lysyl oxidase
US5059814A (en) * 1988-11-30 1991-10-22 The California Institute Of Technology Winner-take-all circuits for neural computing systems
JPH0848664A (ja) * 1994-08-05 1996-02-20 Hisamitsu Pharmaceut Co Inc 新規なグアニジノ安息香酸エステル誘導体
GB9506188D0 (en) * 1995-03-27 1995-05-17 Fujisawa Pharmaceutical Co Amidine derivatives
JP2004502682A (ja) * 2000-07-05 2004-01-29 バイオティ　セラピーズ　コーポレイション 銅含有アミン・オキシダーゼの阻害剤
WO2002038153A1 (en) * 2000-11-09 2002-05-16 Biovitrum Ab New use of 4, 5, 6, 7-tetrahydroimidazo-[4,5-c]pyridine derivatives
US7125901B2 (en) * 2003-01-27 2006-10-24 Astellas Pharma Inc. Thiazole derivatives
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US20070208068A1 (en) * 2004-03-18 2007-09-06 R-Tech Ueno, Ltd. & Astellas Pharma Inc. Aqueous Composition Comprising Thiazole Derivative

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