JP2008507539A - 置換アリール−アミン誘導体および使用方法 - Google Patents

置換アリール−アミン誘導体および使用方法 Download PDF

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JP2008507539A
JP2008507539A JP2007522715A JP2007522715A JP2008507539A JP 2008507539 A JP2008507539 A JP 2008507539A JP 2007522715 A JP2007522715 A JP 2007522715A JP 2007522715 A JP2007522715 A JP 2007522715A JP 2008507539 A JP2008507539 A JP 2008507539A
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Prior art keywords
pyridinecarboxamide
phenyl
methyl
isoquinolinylamino
dihydro
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JP2008507539A5 (enExample
Inventor
ユアン，チエスター・チエンクワン
ヤン，ケビン
フアンデルプラス，シモン
リアヒ，ババツク
ポタシユマン，ミシエル
パテル，ビノツド・エフ
ノマツク，ラナ
リ，アイウエン
ホワン，チー
アルマンジユ，ジヤン−クリストフ
アスキユー，ベニー・シー，ジユニア
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アムジエン・インコーポレーテツド
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Publication of JP2008507539A publication Critical patent/JP2008507539A/ja
Publication of JP2008507539A5 publication Critical patent/JP2008507539A5/ja
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
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  • Diabetes (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
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  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
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  • Biotechnology (AREA)
JP2007522715A 2004-07-22 2005-07-20 置換アリール−アミン誘導体および使用方法 Withdrawn JP2008507539A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US59054404P 2004-07-22 2004-07-22
US11/185,556 US7507748B2 (en) 2004-07-22 2005-07-19 Substituted aryl-amine derivatives and methods of use
PCT/US2005/025800 WO2006012374A1 (en) 2004-07-22 2005-07-20 Substituted aryl-amine derivatives and methods of use

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Publication Number Publication Date
JP2008507539A true JP2008507539A (ja) 2008-03-13
JP2008507539A5 JP2008507539A5 (enExample) 2008-06-26

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US (2) US7507748B2 (enExample)
EP (1) EP1773817B1 (enExample)
JP (1) JP2008507539A (enExample)
AT (1) ATE440834T1 (enExample)
AU (1) AU2005267161B2 (enExample)
CA (1) CA2571627C (enExample)
DE (1) DE602005016261D1 (enExample)
ES (1) ES2331318T3 (enExample)
MX (1) MX2007000672A (enExample)
WO (1) WO2006012374A1 (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2016516812A (ja) * 2013-04-19 2016-06-09 リサーチ コーポレーション ファウンデーション オブ ヨンナム ユニバーシティ アミドピリジンオール誘導体またはその薬剤学的に許容可能な塩、及びそれを有効成分として含有する薬学組成物
JP2022508277A (ja) * 2018-11-28 2022-01-19 バイエル、アクチエンゲゼルシャフト 殺真菌性化合物としてのピリダジン（チオ）アミド
JP2022104792A (ja) * 2020-12-29 2022-07-11 ヒュサイオン カンパニー リミテッド ピペルロングミン系化合物及びこれを含む免疫調節剤

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7507748B2 (en) * 2004-07-22 2009-03-24 Amgen Inc. Substituted aryl-amine derivatives and methods of use
EP1781284B1 (en) * 2004-08-25 2010-10-13 The University of Chicago Use of the combination comprising temozolomide and tnf-alpha for treating glioblastoma
EP2202223B1 (en) 2007-10-18 2017-01-25 Takeda Pharmaceutical Company Limited Heterocyclic compound as blood rbp4 lowering agent
WO2011161217A2 (en) 2010-06-23 2011-12-29 Palacký University in Olomouc Targeting of vegfr2
EP2630122B1 (en) * 2010-10-18 2016-11-30 RaQualia Pharma Inc Arylamide derivatives as ttx-s blockers
US9029553B2 (en) * 2011-02-14 2015-05-12 Council Of Scientific & Industrial Research 2-anilino nicotinyl linked 2-amino benzothiazole conjugates and process for the preparation thereof
CN103717757A (zh) * 2011-05-24 2014-04-09 威斯特研究所 用于调节爱泼斯坦-巴尔核抗原1的活性的组合物和方法
KR101412794B1 (ko) 2011-07-27 2014-07-01 보령제약 주식회사 혈관생성억제 작용을 갖는 신규한 화합물, 이의 제조방법 및 이를 포함하는 약학적 조성물
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