JP2008500316A - 抗菌薬の中間体としてのアリール置換されたオキサゾリジノンの製造方法 - Google Patents

抗菌薬の中間体としてのアリール置換されたオキサゾリジノンの製造方法 Download PDF

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Publication number
JP2008500316A
JP2008500316A JP2007514085A JP2007514085A JP2008500316A JP 2008500316 A JP2008500316 A JP 2008500316A JP 2007514085 A JP2007514085 A JP 2007514085A JP 2007514085 A JP2007514085 A JP 2007514085A JP 2008500316 A JP2008500316 A JP 2008500316A
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Japan
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compound
formula
solution
vii
alkyl
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JP2007514085A
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English (en)
Japanese (ja)
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JP2008500316A5 (enExample
Inventor
チェリーマン，ジャネット
キュスバート，マーレイ・ワトソン
デュビエズ，ジェローム
ホーウェルズ，ガーネット・エドワード
ムルホランド，キース・レイモンド
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AstraZeneca AB
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AstraZeneca AB
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Publication of JP2008500316A publication Critical patent/JP2008500316A/ja
Publication of JP2008500316A5 publication Critical patent/JP2008500316A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2007514085A 2004-05-25 2005-05-24 抗菌薬の中間体としてのアリール置換されたオキサゾリジノンの製造方法 Pending JP2008500316A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0411596.0A GB0411596D0 (en) 2004-05-25 2004-05-25 Chemical process
PCT/GB2005/002042 WO2005116017A1 (en) 2004-05-25 2005-05-24 Process for the preparation of aryl substituted oxazolidinones as intermediates for antibacterial agents

Publications (2)

Publication Number Publication Date
JP2008500316A true JP2008500316A (ja) 2008-01-10
JP2008500316A5 JP2008500316A5 (enExample) 2008-06-26

Family

ID=32670975

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007514085A Pending JP2008500316A (ja) 2004-05-25 2005-05-24 抗菌薬の中間体としてのアリール置換されたオキサゾリジノンの製造方法

Country Status (6)

Country Link
US (1) US20090105484A1 (enExample)
EP (1) EP1753751A1 (enExample)
JP (1) JP2008500316A (enExample)
CN (1) CN100537567C (enExample)
GB (1) GB0411596D0 (enExample)
WO (1) WO2005116017A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100854211B1 (ko) 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
US8604209B2 (en) 2008-10-10 2013-12-10 Trius Therapeutics, Inc. Methods for preparing oxazolidinones and compositions containing them
BRPI1008829A2 (pt) 2009-02-03 2016-03-15 Trius Therapeutics forma cristalina de dihidrogenofosfato de (r)-3-(4-(2-(2-metiltetrazol-5-il) piridin-5-il)-3-fluorofenil)-5-hidroximetil oxazolidin-2-ona
US8580767B2 (en) 2009-05-28 2013-11-12 Trius Therapeutics, Inc. Oxazolidinone containing dimer compounds, compositions and methods to make and use

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002057207A1 (en) * 2001-01-22 2002-07-25 Council Of Scientific And Industrial Research An eco-friendly method of preparation of high purity tetrabromobisphenol-a
WO2003022824A1 (en) * 2001-09-11 2003-03-20 Astrazeneca Ab Oxazolidinone and/or isoxazoline as antibacterial agents
WO2003035648A1 (en) * 2001-10-25 2003-05-01 Astrazeneca Ab Aryl substituted oxazolidinones with antibacterial activity
WO2003072575A1 (en) * 2002-02-28 2003-09-04 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents
JP2003335762A (ja) * 2002-05-20 2003-11-28 Meiji Seika Kaisha Ltd 新規ビフェニル誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200500360A (en) * 2003-03-01 2005-01-01 Astrazeneca Ab Hydroxymethyl compounds

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002057207A1 (en) * 2001-01-22 2002-07-25 Council Of Scientific And Industrial Research An eco-friendly method of preparation of high purity tetrabromobisphenol-a
WO2003022824A1 (en) * 2001-09-11 2003-03-20 Astrazeneca Ab Oxazolidinone and/or isoxazoline as antibacterial agents
WO2003035648A1 (en) * 2001-10-25 2003-05-01 Astrazeneca Ab Aryl substituted oxazolidinones with antibacterial activity
WO2003072575A1 (en) * 2002-02-28 2003-09-04 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents
JP2003335762A (ja) * 2002-05-20 2003-11-28 Meiji Seika Kaisha Ltd 新規ビフェニル誘導体

Also Published As

Publication number Publication date
WO2005116017A1 (en) 2005-12-08
EP1753751A1 (en) 2007-02-21
US20090105484A1 (en) 2009-04-23
GB0411596D0 (en) 2004-06-30
CN1989133A (zh) 2007-06-27
CN100537567C (zh) 2009-09-09

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