JP2007537244A5 - - Google Patents

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Publication number
JP2007537244A5
JP2007537244A5 JP2007512735A JP2007512735A JP2007537244A5 JP 2007537244 A5 JP2007537244 A5 JP 2007537244A5 JP 2007512735 A JP2007512735 A JP 2007512735A JP 2007512735 A JP2007512735 A JP 2007512735A JP 2007537244 A5 JP2007537244 A5 JP 2007537244A5
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JP
Japan
Prior art keywords
group
alkyl
branched
linear
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007512735A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007537244A (ja
Filing date
Publication date
Priority claimed from IT000241A external-priority patent/ITRM20040241A1/it
Application filed filed Critical
Publication of JP2007537244A publication Critical patent/JP2007537244A/ja
Publication of JP2007537244A5 publication Critical patent/JP2007537244A5/ja
Withdrawn legal-status Critical Current

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JP2007512735A 2004-05-13 2005-05-04 20位にてインテグリンアンタゴニストと接合したカンプトテシン誘導体 Withdrawn JP2007537244A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT000241A ITRM20040241A1 (it) 2004-05-13 2004-05-13 Camptotecine coniugate in posizione 20 con antagonisti delle integrine.
PCT/IT2005/000261 WO2005110487A2 (en) 2004-05-13 2005-05-04 Camptothecin derivatives conjugated in position 20 with integrin antagonists

Publications (2)

Publication Number Publication Date
JP2007537244A JP2007537244A (ja) 2007-12-20
JP2007537244A5 true JP2007537244A5 (https=) 2008-06-26

Family

ID=35124307

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007512735A Withdrawn JP2007537244A (ja) 2004-05-13 2005-05-04 20位にてインテグリンアンタゴニストと接合したカンプトテシン誘導体

Country Status (12)

Country Link
US (1) US20070232639A1 (https=)
EP (1) EP1747019A2 (https=)
JP (1) JP2007537244A (https=)
CN (1) CN101010103A (https=)
AR (1) AR049275A1 (https=)
AU (1) AU2005243834A1 (https=)
BR (1) BRPI0511037A (https=)
CA (1) CA2562572A1 (https=)
IT (1) ITRM20040241A1 (https=)
MX (1) MXPA06012886A (https=)
TW (1) TW200538125A (https=)
WO (1) WO2005110487A2 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9216228B2 (en) 2007-02-16 2015-12-22 KTB Tumorforschungsgesellschaft MBM Receptor and antigen targeted prodrug
WO2013110578A1 (en) * 2012-01-27 2013-08-01 F. Hoffmann-La Roche Ag Integrin antagonist conjugates for targeted delivery to cells expressing alpha-v-beta-3
CN105399757A (zh) * 2015-12-29 2016-03-16 遵义医学院 酸敏感型喜树碱-20位去甲斑蝥酸酯衍生物及其抗肿瘤应用
CN111068068A (zh) * 2019-12-04 2020-04-28 云南民族大学 一种rgd多肽-喜树碱多肽药物偶联物及其应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19815812A1 (de) * 1998-04-08 1999-10-14 Bayer Ag Modifizierte Cytostatika
EP1044977B1 (en) * 1999-03-09 2002-05-02 Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. Camptothecin derivatives having antitumor activity
US6207832B1 (en) * 1999-04-09 2001-03-27 University Of Pittsburgh Camptothecin analogs and methods of preparation thereof
ATE438413T1 (de) * 1999-09-08 2009-08-15 Markus Albers Integrin-vermittelte arzneimittel-zielrichtung

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