JP2007532649A5 - - Google Patents

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Publication number
JP2007532649A5
JP2007532649A5 JP2007508407A JP2007508407A JP2007532649A5 JP 2007532649 A5 JP2007532649 A5 JP 2007532649A5 JP 2007508407 A JP2007508407 A JP 2007508407A JP 2007508407 A JP2007508407 A JP 2007508407A JP 2007532649 A5 JP2007532649 A5 JP 2007532649A5
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JP
Japan
Prior art keywords
group
alkyl group
compound
medicament
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007508407A
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English (en)
Japanese (ja)
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JP2007532649A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/012028 external-priority patent/WO2005108378A2/en
Publication of JP2007532649A publication Critical patent/JP2007532649A/ja
Publication of JP2007532649A5 publication Critical patent/JP2007532649A5/ja
Pending legal-status Critical Current

Links

JP2007508407A 2004-04-15 2005-04-12 (4−アルキルピペラジニル)(フェニル)メタノン Pending JP2007532649A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56264304P 2004-04-15 2004-04-15
PCT/US2005/012028 WO2005108378A2 (en) 2004-04-15 2005-04-12 Use of (4-alkylpiperazinyl) (phenyl) methanones in the treatment of alzheimer’s disease

Publications (2)

Publication Number Publication Date
JP2007532649A JP2007532649A (ja) 2007-11-15
JP2007532649A5 true JP2007532649A5 (https=) 2008-05-29

Family

ID=35058789

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007508407A Pending JP2007532649A (ja) 2004-04-15 2005-04-12 (4−アルキルピペラジニル)(フェニル)メタノン

Country Status (7)

Country Link
US (1) US20090197891A1 (https=)
EP (1) EP1755605A2 (https=)
JP (1) JP2007532649A (https=)
CN (1) CN101022806A (https=)
AU (1) AU2005240991A1 (https=)
CA (1) CA2564068A1 (https=)
WO (1) WO2005108378A2 (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10303974A1 (de) 2003-01-31 2004-08-05 Abbott Gmbh & Co. Kg Amyloid-β(1-42)-Oligomere, Verfahren zu deren Herstellung und deren Verwendung
HRP20140240T4 (hr) 2005-11-30 2017-02-24 Abbvie Inc. Monoklonalna antitijela protiv amiloidnih beta proteina i njihova upotreba
US8691224B2 (en) 2005-11-30 2014-04-08 Abbvie Inc. Anti-Aβ globulomer 5F7 antibodies
US8455626B2 (en) 2006-11-30 2013-06-04 Abbott Laboratories Aβ conformer selective anti-aβ globulomer monoclonal antibodies
US8895004B2 (en) 2007-02-27 2014-11-25 AbbVie Deutschland GmbH & Co. KG Method for the treatment of amyloidoses
US8987419B2 (en) 2010-04-15 2015-03-24 AbbVie Deutschland GmbH & Co. KG Amyloid-beta binding proteins
EP3533803B1 (en) 2010-08-14 2021-10-27 AbbVie Inc. Anti-amyloid-beta antibodies
IL283725B2 (en) 2017-06-20 2024-04-01 Imbria Pharmaceuticals Inc Compositions and methods for increasing efficiency of cardiac metabolism
CN108329282B (zh) * 2018-01-16 2022-01-07 新乡医学院 一种苯基哌嗪类衍生物及其制备方法和应用
EP3866794B1 (en) 2018-10-17 2024-12-04 Imbria Pharmaceuticals, Inc. Methods of treating rheumatic diseases using trimetazidine-based compounds
EP3976101A4 (en) 2019-05-31 2023-06-21 Imbria Pharmaceuticals, Inc. FIBROSIS TREATMENT METHODS USING COMPOUNDS THAT PROMOTE GLUCOSE OXIDATION
US11530184B2 (en) 2020-06-30 2022-12-20 Imbria Pharmaceuticals, Inc. Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11780811B2 (en) 2020-06-30 2023-10-10 Imbria Pharmaceuticals, Inc. Methods of synthesizing 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate
US11883396B2 (en) 2021-05-03 2024-01-30 Imbria Pharmaceuticals, Inc. Methods of treating kidney conditions using modified forms of trimetazidine
WO2022246115A1 (en) * 2021-05-19 2022-11-24 Cornell University Apt1 and apt2 inhibitors and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2304155A1 (de) * 1973-01-29 1974-08-01 Ichthyol Ges Cordes Hermanni & N-acylierte substituierte piperazinbzw. homopiperazinderivate, sowie verfahren zu ihrer herstellung
US5693804A (en) * 1994-11-17 1997-12-02 Molecular Geriatrics Corporation Substituted 1-aryl-3-piperazin-1'-yl propanones
DE19934433A1 (de) * 1999-07-22 2001-01-25 Merck Patent Gmbh N-(Indolcarbonyl-)piperazinderivate
US20040034019A1 (en) * 2002-08-08 2004-02-19 Ronald Tomlinson Piperazine and piperidine derivatives
GB0224084D0 (en) * 2002-10-16 2002-11-27 Glaxo Group Ltd Novel compounds
AU2004245484A1 (en) * 2003-06-02 2004-12-16 Georgetown University Neuroprotective benzoate and benzamide compounds

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