JP2007518723A5 - - Google Patents

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Publication number
JP2007518723A5
JP2007518723A5 JP2006547532A JP2006547532A JP2007518723A5 JP 2007518723 A5 JP2007518723 A5 JP 2007518723A5 JP 2006547532 A JP2006547532 A JP 2006547532A JP 2006547532 A JP2006547532 A JP 2006547532A JP 2007518723 A5 JP2007518723 A5 JP 2007518723A5
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JP
Japan
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iii
temperature
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JP2006547532A
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English (en)
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JP4927563B2 (ja
JP2007518723A (ja
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Priority claimed from PCT/US2004/043823 external-priority patent/WO2005066122A2/en
Publication of JP2007518723A publication Critical patent/JP2007518723A/ja
Publication of JP2007518723A5 publication Critical patent/JP2007518723A5/ja
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Publication of JP4927563B2 publication Critical patent/JP4927563B2/ja
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Claims (1)

  1. 段階（iii）が、約−20℃〜約80℃の温度で行われる、請求項25記載の方法。
JP2006547532A 2003-12-30 2004-12-30 アシルオキシアルキルカルバメートプロドラッグ及び中間体の合成 Active JP4927563B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53364903P 2003-12-30 2003-12-30
US60/533,649 2003-12-30
US60663704P 2004-08-13 2004-08-13
US60/606,637 2004-08-13
PCT/US2004/043823 WO2005066122A2 (en) 2003-12-30 2004-12-30 Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011175796A Division JP5670842B2 (ja) 2003-12-30 2011-08-11 アシルオキシアルキルカルバメートプロドラッグの合成

Publications (3)

Publication Number Publication Date
JP2007518723A JP2007518723A (ja) 2007-07-12
JP2007518723A5 true JP2007518723A5 (ja) 2008-02-28
JP4927563B2 JP4927563B2 (ja) 2012-05-09

Family

ID=34753006

Family Applications (2)

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JP2006547532A Active JP4927563B2 (ja) 2003-12-30 2004-12-30 アシルオキシアルキルカルバメートプロドラッグ及び中間体の合成
JP2011175796A Expired - Fee Related JP5670842B2 (ja) 2003-12-30 2011-08-11 アシルオキシアルキルカルバメートプロドラッグの合成

Family Applications After (1)

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JP2011175796A Expired - Fee Related JP5670842B2 (ja) 2003-12-30 2011-08-11 アシルオキシアルキルカルバメートプロドラッグの合成

Country Status (10)

Country Link
US (5) US7227028B2 (ja)
EP (2) EP1716115B1 (ja)
JP (2) JP4927563B2 (ja)
CN (1) CN102702065A (ja)
CA (1) CA2551859C (ja)
DK (1) DK1716115T3 (ja)
ES (1) ES2405329T3 (ja)
HK (1) HK1090924A1 (ja)
IL (2) IL176341A (ja)
WO (1) WO2005066122A2 (ja)

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