JP2007517783A5 - - Google Patents

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Publication number
JP2007517783A5
JP2007517783A5 JP2006545583A JP2006545583A JP2007517783A5 JP 2007517783 A5 JP2007517783 A5 JP 2007517783A5 JP 2006545583 A JP2006545583 A JP 2006545583A JP 2006545583 A JP2006545583 A JP 2006545583A JP 2007517783 A5 JP2007517783 A5 JP 2007517783A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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JP2006545583A
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Japanese (ja)
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JP5546717B2 (ja
JP2007517783A (ja
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Priority claimed from PCT/US2004/042976 external-priority patent/WO2005058835A2/en
Publication of JP2007517783A publication Critical patent/JP2007517783A/ja
Publication of JP2007517783A5 publication Critical patent/JP2007517783A5/ja
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Publication of JP5546717B2 publication Critical patent/JP5546717B2/ja
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JP2006545583A 2003-12-16 2004-12-16 アリピプラゾール結晶質形態を調製する方法 Expired - Lifetime JP5546717B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US53029703P 2003-12-16 2003-12-16
US60/530,297 2003-12-16
US53383103P 2003-12-30 2003-12-30
US60/533,831 2003-12-30
US61840404P 2004-10-13 2004-10-13
US60/618,404 2004-10-13
US61896004P 2004-10-14 2004-10-14
US60/618,960 2004-10-14
PCT/US2004/042976 WO2005058835A2 (en) 2003-12-16 2004-12-16 Methods of preparing aripiprazole crystalline forms

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2013147411A Division JP2013237682A (ja) 2003-12-16 2013-07-16 アリピプラゾール結晶質形態を調製する方法

Publications (3)

Publication Number Publication Date
JP2007517783A JP2007517783A (ja) 2007-07-05
JP2007517783A5 true JP2007517783A5 (https=) 2008-04-17
JP5546717B2 JP5546717B2 (ja) 2014-07-09

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Family Applications (2)

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JP2006545583A Expired - Lifetime JP5546717B2 (ja) 2003-12-16 2004-12-16 アリピプラゾール結晶質形態を調製する方法
JP2013147411A Pending JP2013237682A (ja) 2003-12-16 2013-07-16 アリピプラゾール結晶質形態を調製する方法

Family Applications After (1)

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JP2013147411A Pending JP2013237682A (ja) 2003-12-16 2013-07-16 アリピプラゾール結晶質形態を調製する方法

Country Status (11)

Country Link
US (2) US7504504B2 (https=)
EP (1) EP1613598B1 (https=)
JP (2) JP5546717B2 (https=)
AT (1) ATE529409T1 (https=)
CA (1) CA2550726A1 (https=)
ES (1) ES2374922T3 (https=)
IL (1) IL175512A (https=)
PL (1) PL1613598T3 (https=)
PT (1) PT1613598E (https=)
TW (1) TW200529850A (https=)
WO (1) WO2005058835A2 (https=)

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TWI394753B (zh) 2006-03-17 2013-05-01 Otsuka Pharma Co Ltd 新穎替妥牟拉（ｔｅｔｏｍｉｌａｓｔ）晶體
US7799790B2 (en) 2006-07-20 2010-09-21 Helm Ag Amorphous aripiprazole and process for the preparation thereof
EP1880714A1 (en) 2006-07-20 2008-01-23 Helm AG Amorphous Aripiprazole and Process for the Preparation thereof
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WO2008051541A2 (en) * 2006-10-24 2008-05-02 Cambrex Charles City, Inc. Process for preparing anhydrous aripirazole type i
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EP2238976B1 (en) 2009-04-03 2012-06-27 Hexal AG Oral films comprising 7-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]-3,4-dihydro- 1H-quinolin-2-one base or salts or hydrates thereof
CN101948426A (zh) * 2010-09-13 2011-01-19 浙江华海药业股份有限公司 一种制备阿立哌唑晶型b的新方法
US9757374B2 (en) 2010-10-28 2017-09-12 Aequus Pharmaceuticals Inc. Aripiprazole compositions and methods for its transdermal delivery
BR112013010190B1 (pt) 2010-10-28 2019-12-31 Aequus Pharmaceuticals Inc composição farmacêutica
WO2012077134A1 (en) * 2010-12-07 2012-06-14 Ind-Swift Laboratories Limted Process for preparing aripiprazole polymorphs
KR101340214B1 (ko) * 2011-03-31 2013-12-10 주식회사 대웅제약 무수 아리피프라졸 ⅱ형 결정의 제조방법
CN102850268B (zh) * 2011-06-27 2015-07-15 上海中西制药有限公司 阿立哌唑ⅰ型微晶、阿立哌唑固体制剂及制备方法
KR101372840B1 (ko) * 2012-08-02 2014-03-12 주식회사 에스텍파마 무수 아리피프라졸 결정의 제조방법
EP3065700A1 (en) 2013-11-07 2016-09-14 Synthon B.V. Orodispersible pharmaceutical compositions comprising aripiprazole
AR099354A1 (es) 2013-11-15 2016-07-20 Akebia Therapeutics Inc Formas sólidas de ácido {[5-(3-clorofenil)-3-hidroxipiridin-2-carbonil]amino}acético, composiciones, y sus usos
CN106474058B (zh) 2015-08-31 2020-01-07 南京诺瑞特医药科技有限公司 具有延长的保质期的阿立哌唑可注射悬浮液制剂
TWI665194B (zh) * 2016-02-19 2019-07-11 諾瑞特國際藥業股份有限公司 阿立哌唑的新晶型

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WO2006053780A1 (en) * 2004-11-18 2006-05-26 Synthon B.V. Crystalline aripiprazole solvates
EP1812397A1 (en) * 2004-11-18 2007-08-01 Synthon B.V. Process of making crystalline aripiprazole
EP1686117A1 (en) * 2005-01-27 2006-08-02 Sandoz AG Polymorph and solvates of aripiprazole
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EP1919453A2 (en) * 2005-12-22 2008-05-14 Teva Pharmaceutical Industries Ltd Processes for reducing particle size of aripiprazole
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EP1880714A1 (en) * 2006-07-20 2008-01-23 Helm AG Amorphous Aripiprazole and Process for the Preparation thereof

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