JP2006527184A - 口腔内分散性多層錠剤 - Google Patents
口腔内分散性多層錠剤 Download PDFInfo
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- JP2006527184A JP2006527184A JP2006508358A JP2006508358A JP2006527184A JP 2006527184 A JP2006527184 A JP 2006527184A JP 2006508358 A JP2006508358 A JP 2006508358A JP 2006508358 A JP2006508358 A JP 2006508358A JP 2006527184 A JP2006527184 A JP 2006527184A
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- ITVGXXMINPYUHD-CUVHLRMHSA-N neohesperidin dihydrochalcone Chemical compound C1=C(O)C(OC)=CC=C1CCC(=O)C(C(=C1)O)=C(O)C=C1O[C@H]1[C@H](O[C@H]2[C@@H]([C@H](O)[C@@H](O)[C@H](C)O2)O)[C@@H](O)[C@H](O)[C@@H](CO)O1 ITVGXXMINPYUHD-CUVHLRMHSA-N 0.000 description 1
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- 150000003242 quaternary ammonium salts Chemical class 0.000 description 1
- IUVKMZGDUIUOCP-BTNSXGMBSA-N quinbolone Chemical compound O([C@H]1CC[C@H]2[C@H]3[C@@H]([C@]4(C=CC(=O)C=C4CC3)C)CC[C@@]21C)C1=CCCC1 IUVKMZGDUIUOCP-BTNSXGMBSA-N 0.000 description 1
- VMXUWOKSQNHOCA-LCYFTJDESA-N ranitidine Chemical compound [O-][N+](=O)/C=C(/NC)NCCSCC1=CC=C(CN(C)C)O1 VMXUWOKSQNHOCA-LCYFTJDESA-N 0.000 description 1
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- 235000017550 sodium carbonate Nutrition 0.000 description 1
- 235000002639 sodium chloride Nutrition 0.000 description 1
- SUKJFIGYRHOWBL-UHFFFAOYSA-N sodium hypochlorite Chemical compound [Na+].Cl[O-] SUKJFIGYRHOWBL-UHFFFAOYSA-N 0.000 description 1
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- 229940079832 sodium starch glycolate Drugs 0.000 description 1
- YKLJGMBLPUQQOI-UHFFFAOYSA-M sodium;oxidooxy(oxo)borane Chemical compound [Na+].[O-]OB=O YKLJGMBLPUQQOI-UHFFFAOYSA-M 0.000 description 1
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- DPJRMOMPQZCRJU-UHFFFAOYSA-M thiamine hydrochloride Chemical compound Cl.[Cl-].CC1=C(CCO)SC=[N+]1CC1=CN=C(C)N=C1N DPJRMOMPQZCRJU-UHFFFAOYSA-M 0.000 description 1
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- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Zoology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Medicinal Preparation (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0306900A FR2855756B1 (fr) | 2003-06-06 | 2003-06-06 | Comprime orodispersible multicouche |
| US10/610,668 US20040247677A1 (en) | 2003-06-06 | 2003-06-30 | Multilayer orodispersible tablet |
| PCT/FR2004/001400 WO2004110411A2 (fr) | 2003-06-06 | 2004-06-04 | Comprime orodispersible multicouche |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2011243534A Division JP5572616B2 (ja) | 2003-06-06 | 2011-11-07 | 口腔内分散性多層錠剤 |
Publications (2)
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| JP2006527184A true JP2006527184A (ja) | 2006-11-30 |
| JP2006527184A5 JP2006527184A5 (https=) | 2012-01-12 |
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| JP2006508358A Pending JP2006527184A (ja) | 2003-06-06 | 2004-06-04 | 口腔内分散性多層錠剤 |
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| Country | Link |
|---|---|
| US (1) | US8263126B2 (https=) |
| EP (1) | EP1631263B1 (https=) |
| JP (1) | JP2006527184A (https=) |
| KR (1) | KR101125268B1 (https=) |
| AU (1) | AU2004246837B2 (https=) |
| BR (1) | BRPI0411039A (https=) |
| CA (1) | CA2528249C (https=) |
| IS (1) | IS8197A (https=) |
| MX (1) | MXPA05013202A (https=) |
| NO (1) | NO337922B1 (https=) |
| WO (1) | WO2004110411A2 (https=) |
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| WO2008149440A1 (ja) * | 2007-06-07 | 2008-12-11 | Sato Pharmaceutical Co., Ltd. | 速溶性及び可撓性を有するフィルム製剤 |
| JP2009545561A (ja) * | 2006-08-04 | 2009-12-24 | エチファーム | 多層口腔内崩壊錠剤 |
| JP2010516789A (ja) * | 2007-01-29 | 2010-05-20 | ユーロファルマ・ラボラトリオス・エルティーディーエー． | トラマドールおよびケトプロフェンを組合せて含む薬学的組成物 |
| JP2010532367A (ja) * | 2007-06-29 | 2010-10-07 | マクニール−ピーピーシー・インコーポレーテツド | ２部分からなるロゼンジ剤形 |
| JP2013510131A (ja) * | 2009-11-05 | 2013-03-21 | サノフイ | 抗マラリア剤の組み合わせを含有する水中に分散できる多層医薬組成物 |
| JP2016506394A (ja) * | 2012-12-17 | 2016-03-03 | エティファーム | 圧縮成形によって得られる口腔分散性錠剤 |
| JP2016519064A (ja) * | 2013-03-14 | 2016-06-30 | スリー イン ワン デンタル ピーエルエルシー３ ｉｎ １ Ｄｅｎｔａｌ ＰＬＬＣ | 口腔乾燥症の治療及び歯の治療のための組成物 |
| WO2017146106A1 (ja) * | 2016-02-25 | 2017-08-31 | 久光製薬株式会社 | 口腔内貼付剤の製造方法 |
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| DE10232113A1 (de) | 2002-07-16 | 2004-01-29 | Bayer Ag | Vardenafil Hydrochlorid Trihydrat enthaltende Arzneimittel |
| MXPA05007016A (es) * | 2003-01-14 | 2005-09-12 | Gilead Sciences Inc | Composiciones y metodos para terapia antiviral de combinacion. |
| DE102005009240A1 (de) | 2005-03-01 | 2006-09-07 | Bayer Healthcare Ag | Arzneiformen mit verbesserten pharmakokinetischen Eigenschaften |
| US20080187581A1 (en) * | 2005-03-16 | 2008-08-07 | Subhash Pandurang Gore | Delivery System For Mulitple Drugs |
| TWI375560B (en) | 2005-06-13 | 2012-11-01 | Gilead Sciences Inc | Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same |
| TWI471145B (zh) | 2005-06-13 | 2015-02-01 | Bristol Myers Squibb & Gilead Sciences Llc | 單一式藥學劑量型 |
| EP1993518A4 (en) * | 2006-03-06 | 2012-12-12 | Pozen Inc | DOSAGE FORMS FOR THE ADMINISTRATION OF MEDICINAL COMBINATIONS |
| US9265732B2 (en) | 2006-03-06 | 2016-02-23 | Pozen Inc. | Dosage forms for administering combinations of drugs |
| US20070286900A1 (en) * | 2006-06-09 | 2007-12-13 | Catherine Herry | Low dose tablets of opioid analgesics and preparation process |
| KR100816064B1 (ko) * | 2006-08-16 | 2008-03-24 | 주식회사 케이티앤지 | 홍삼이 함유된 다중 정제 및 이의 제조방법 |
| EP2124556B1 (en) | 2006-10-09 | 2014-09-03 | Charleston Laboratories, Inc. | Pharmaceutical compositions |
| ES2620672T3 (es) | 2008-01-09 | 2017-06-29 | Charleston Laboratories, Inc. | Comprimidos de doble capa que comprenden oxicodona y prometazina |
| AU2009240586A1 (en) * | 2008-04-24 | 2009-10-29 | Evestra, Inc. | Oral contraceptive dosage forms comprising a progestogen dispersed in an enteric polymer and further comprising an estrogen |
| JP2012521393A (ja) * | 2009-03-26 | 2012-09-13 | ロイヤル カレッジ オブ サージェオンズ イン アイルランド | 口腔内分散性錠剤 |
| EP2418861A4 (en) * | 2009-04-14 | 2013-01-09 | Panasonic Corp | VIDEO DISPLAY DEVICE, GLASS FOR VIEWING VIDEO AND A VIDEO DISPLAY DEVICE AND GLASS FOR VIDEO LISTENING SYSTEM |
| JP5845172B2 (ja) * | 2009-05-01 | 2016-01-20 | アデア ファーマスーティカルズ，インコーポレイテッド | 高および低用量薬物の組み合わせを含む口腔内崩壊錠組成物 |
| WO2011006012A1 (en) | 2009-07-08 | 2011-01-13 | Charleston Laboratories Inc. | Pharmaceutical compositions |
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| JPH01110622A (ja) * | 1987-10-21 | 1989-04-27 | Teikoku Seiyaku Kk | 薬物断続放出性口腔内適用製剤 |
| JPH08501544A (ja) * | 1992-09-24 | 1996-02-20 | ヤゴテック アーゲー | １種以上の薬剤を異なった放出速度で放出することのできる薬用錠剤 |
| JP2000336027A (ja) * | 1999-05-26 | 2000-12-05 | Lion Corp | 多層錠の剥離抑制方法 |
| JP2003506316A (ja) * | 1999-03-01 | 2003-02-18 | エティファーム | 低破砕性の口内散乱型錠剤及びその調製方法 |
| WO2003017985A1 (en) * | 2001-08-23 | 2003-03-06 | Cimex Ag | Bilayered dispersible tablet formulation comprising amoxycillin and clavulanate in separate layers |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JPH0830005B2 (ja) * | 1985-09-25 | 1996-03-27 | ゲルゲリイ、ゲルハルト | 崩壊性錠剤とその製造方法 |
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| FR2855756B1 (fr) * | 2003-06-06 | 2005-08-26 | Ethypharm Sa | Comprime orodispersible multicouche |
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2004
- 2004-06-04 AU AU2004246837A patent/AU2004246837B2/en not_active Ceased
- 2004-06-04 CA CA2528249A patent/CA2528249C/fr not_active Expired - Fee Related
- 2004-06-04 MX MXPA05013202A patent/MXPA05013202A/es active IP Right Grant
- 2004-06-04 US US10/559,350 patent/US8263126B2/en active Active
- 2004-06-04 JP JP2006508358A patent/JP2006527184A/ja active Pending
- 2004-06-04 WO PCT/FR2004/001400 patent/WO2004110411A2/fr not_active Ceased
- 2004-06-04 BR BRPI0411039-0A patent/BRPI0411039A/pt not_active Application Discontinuation
- 2004-06-04 EP EP04767267.0A patent/EP1631263B1/fr not_active Expired - Lifetime
- 2004-06-04 KR KR1020057023476A patent/KR101125268B1/ko not_active Expired - Lifetime
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2005
- 2005-12-19 NO NO20056046A patent/NO337922B1/no not_active IP Right Cessation
- 2005-12-22 IS IS8197A patent/IS8197A/is unknown
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| JP2003506316A (ja) * | 1999-03-01 | 2003-02-18 | エティファーム | 低破砕性の口内散乱型錠剤及びその調製方法 |
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| WO2003017985A1 (en) * | 2001-08-23 | 2003-03-06 | Cimex Ag | Bilayered dispersible tablet formulation comprising amoxycillin and clavulanate in separate layers |
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009545561A (ja) * | 2006-08-04 | 2009-12-24 | エチファーム | 多層口腔内崩壊錠剤 |
| JP2010516789A (ja) * | 2007-01-29 | 2010-05-20 | ユーロファルマ・ラボラトリオス・エルティーディーエー． | トラマドールおよびケトプロフェンを組合せて含む薬学的組成物 |
| WO2008149440A1 (ja) * | 2007-06-07 | 2008-12-11 | Sato Pharmaceutical Co., Ltd. | 速溶性及び可撓性を有するフィルム製剤 |
| US9125836B2 (en) | 2007-06-07 | 2015-09-08 | Sato Pharmaceutical Co., Ltd. | Film preparation with rapidly dissolving property and flexibility |
| JP2010532367A (ja) * | 2007-06-29 | 2010-10-07 | マクニール−ピーピーシー・インコーポレーテツド | ２部分からなるロゼンジ剤形 |
| JP2013510131A (ja) * | 2009-11-05 | 2013-03-21 | サノフイ | 抗マラリア剤の組み合わせを含有する水中に分散できる多層医薬組成物 |
| JP2016506394A (ja) * | 2012-12-17 | 2016-03-03 | エティファーム | 圧縮成形によって得られる口腔分散性錠剤 |
| JP2016519064A (ja) * | 2013-03-14 | 2016-06-30 | スリー イン ワン デンタル ピーエルエルシー３ ｉｎ １ Ｄｅｎｔａｌ ＰＬＬＣ | 口腔乾燥症の治療及び歯の治療のための組成物 |
| WO2017146106A1 (ja) * | 2016-02-25 | 2017-08-31 | 久光製薬株式会社 | 口腔内貼付剤の製造方法 |
| JPWO2017146106A1 (ja) * | 2016-02-25 | 2018-09-20 | 久光製薬株式会社 | 口腔内貼付剤の製造方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1631263A2 (fr) | 2006-03-08 |
| KR20060028767A (ko) | 2006-04-03 |
| BRPI0411039A (pt) | 2006-07-11 |
| CA2528249A1 (fr) | 2004-12-23 |
| CA2528249C (fr) | 2013-03-05 |
| NO20056046L (no) | 2005-12-19 |
| IS8197A (is) | 2005-12-22 |
| WO2004110411A2 (fr) | 2004-12-23 |
| US8263126B2 (en) | 2012-09-11 |
| NO337922B1 (no) | 2016-07-11 |
| KR101125268B1 (ko) | 2012-04-23 |
| AU2004246837A1 (en) | 2004-12-23 |
| WO2004110411A3 (fr) | 2005-08-18 |
| AU2004246837B2 (en) | 2009-07-16 |
| MXPA05013202A (es) | 2006-03-09 |
| US20070036861A1 (en) | 2007-02-15 |
| EP1631263B1 (fr) | 2014-02-26 |
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