JP2006506380A - 月経困難症の治療用トリアゾール化合物 - Google Patents

月経困難症の治療用トリアゾール化合物 Download PDF

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JP2006506380A
JP2006506380A JP2004546268A JP2004546268A JP2006506380A JP 2006506380 A JP2006506380 A JP 2006506380A JP 2004546268 A JP2004546268 A JP 2004546268A JP 2004546268 A JP2004546268 A JP 2004546268A JP 2006506380 A JP2006506380 A JP 2006506380A
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triazol
benzyl
tetrahydro
bipyridinyl
ylmethyl
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JP2006506380A5 (enExample
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ダンカン アーマー，ロバート
ダグラス バクスター，アンドリュー
スティーブン ブライアンス，ジャスティン
ネイル ダック，ケビン
スティーブン ジョンソン，パトリック
アンドリュー ルースウェイト，ラッセル
ニューマン，ジュリー
ジェイムズ ローソン，デイビット
リックマンズ，トーマス
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ファイザー・インク
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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  • Diabetes (AREA)
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  • Pulmonology (AREA)
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  • Obesity (AREA)
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  • Child & Adolescent Psychology (AREA)
  • Dermatology (AREA)
  • Otolaryngology (AREA)
  • Anesthesiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
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JP2004546268A 2002-10-25 2003-10-14 月経困難症の治療用トリアゾール化合物 Withdrawn JP2006506380A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0224919.1A GB0224919D0 (en) 2002-10-25 2002-10-25 Triazole compounds useful in therapy
PCT/IB2003/004587 WO2004037809A1 (en) 2002-10-25 2003-10-14 Triazole compounds for the treatment of dysmenorrhoea

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Publication Number Publication Date
JP2006506380A true JP2006506380A (ja) 2006-02-23
JP2006506380A5 JP2006506380A5 (enExample) 2006-11-30

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JP2004546268A Withdrawn JP2006506380A (ja) 2002-10-25 2003-10-14 月経困難症の治療用トリアゾール化合物

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EP (1) EP1558598B1 (enExample)
JP (1) JP2006506380A (enExample)
AT (1) ATE367386T1 (enExample)
AU (1) AU2003267791A1 (enExample)
BR (1) BR0315676A (enExample)
CA (1) CA2502932A1 (enExample)
DE (1) DE60315062T2 (enExample)
ES (1) ES2287508T3 (enExample)
GB (1) GB0224919D0 (enExample)
MX (1) MXPA05004305A (enExample)
WO (1) WO2004037809A1 (enExample)

Cited By (4)

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JP2010514795A (ja) * 2006-12-28 2010-05-06 メタボレックス， インコーポレイテッド 糖尿病および代謝障害を処置するためのヘテロ環式受容体アゴニスト
JP2015500220A (ja) * 2011-12-02 2015-01-05 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ピペリジン誘導体、その医薬組成物及び使用
JP2017510645A (ja) * 2014-03-28 2017-04-13 アゼヴァン ファーマスーティカルズ，インコーポレイテッド 神経変性疾患を治療するための組成物および方法
US10292983B2 (en) 2016-08-03 2019-05-21 Cymabay Therapeutics, Inc. Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions

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GB0317227D0 (en) * 2003-07-23 2003-08-27 Pfizer Ltd Treatment of male sexual dysfunction
ES2277237T3 (es) * 2003-02-19 2007-07-01 Pfizer Inc. Compuestos de triazol utiles en terapia.
GB0325021D0 (en) * 2003-10-27 2003-12-03 Pfizer Ltd Therapeutic combinations
US7745630B2 (en) 2003-12-22 2010-06-29 Justin Stephen Bryans Triazolyl piperidine arginine vasopressin receptor modulators
CN101084207A (zh) 2004-09-20 2007-12-05 泽农医药公司 杂环衍生物及其作为硬脂酰CoA去饱和酶抑制剂的用途
EP1804799B1 (en) 2004-09-20 2013-08-21 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
AR051094A1 (es) * 2004-09-20 2006-12-20 Xenon Pharmaceuticals Inc Derivados heterociclicos y su uso como inhibidores de la estearoil-coa desaturasa
AP2007004047A0 (en) 2005-01-20 2007-06-30 Pfizer Ltd Substituted triazole derivatives as oxtocin antagonists
WO2006114706A1 (en) * 2005-04-26 2006-11-02 Pfizer Limited Triazole derivatives as vasopressin antagonists
CA2608718A1 (en) 2005-05-18 2006-11-23 Pfizer Limited 1, 2, 4-triazole derivatives as vasopressin antagonists
BRPI0611187A2 (pt) 2005-06-03 2010-08-24 Xenon Pharmaceuticals Inc derivados aminotiazàis como inibidores da estearoil-coa desaturase humana
EP1958631A1 (en) * 2007-02-14 2008-08-20 AEterna Zentaris GmbH Novel triazole derivatives as ligands of G-protein coupled receptors
AU2008279447A1 (en) 2007-07-19 2009-01-29 Metabolex, Inc. N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders
WO2009082526A2 (en) * 2007-10-05 2009-07-02 Pharmacopeia, Inc. Ortho pyrrolidine, benzyl-substituted heterocycle ccr1 antagonists for autoimmune diseases & inflammation
JP5909185B2 (ja) 2009-10-01 2016-04-26 シマベイ セラピューティクス， インコーポレーテッド 置換テトラゾール−１−イルフェノキシメチルチアゾール−２−イルピペリジニルピリミジン塩
CN103037843A (zh) 2010-06-23 2013-04-10 麦它波莱克斯股份有限公司 5-乙基-2-{4-[4-(4-四唑-1-基-苯氧甲基)-噻唑-2-基]-哌啶-1-基}-嘧啶的组合物
US9006450B2 (en) * 2010-07-01 2015-04-14 Boehringer Ingelheim International Gmbh Compounds, pharmaceutical compositions and uses thereof
ES2858499T3 (es) 2010-07-01 2021-09-30 Azevan Pharmaceuticals Inc Compuestos para su uso en el tratamiento de trastorno explosivo intermitente
TW201919625A (zh) 2017-09-15 2019-06-01 美商愛治凡製藥公司 用於治療腦損傷之組合物及方法
CN112055713A (zh) 2018-03-01 2020-12-08 安娜普尔纳生物股份有限公司 用于治疗与apj受体活性有关的疾病的化合物和组合物
WO2020163689A1 (en) 2019-02-08 2020-08-13 University Of Pittsburgh - Of The Commonwealth System Of Higher Education 20-hete formation inhibitors
WO2022018121A1 (en) * 2020-07-23 2022-01-27 F. Hoffmann-La Roche Ag Cyclohexyl substituted triazoles as vasopressin receptor v1 a antagonists
WO2025252661A1 (en) * 2024-06-03 2025-12-11 Immunic Ag Reducing body weight and/or induction of satiety by triazolo compounds

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DE574944C (de) * 1932-02-14 1933-04-21 Schering Kahlbaum Ag Verfahren zur Darstellung von 3, 4, 5-trisubstituierten 1, 2, 4-Triazolen
WO2001058880A1 (en) * 2000-02-08 2001-08-16 Yamanouchi Pharmaceutical Co., Ltd. Novel triazole derivatives
JP3873746B2 (ja) * 2000-05-19 2007-01-24 アステラス製薬株式会社 トリアゾール誘導体

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2010514795A (ja) * 2006-12-28 2010-05-06 メタボレックス， インコーポレイテッド 糖尿病および代謝障害を処置するためのヘテロ環式受容体アゴニスト
US9737537B2 (en) 2006-12-28 2017-08-22 Cymabay Therapeutics, Inc. Heterocyclic receptor agonists for the treatment of diabetes and metabolic disorders
US9925189B2 (en) 2006-12-28 2018-03-27 Cymabay Therapeutics, Inc. Heterocyclic receptor agonists for the treatment of diabetes and metabolic disorders
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AU2003267791A1 (en) 2004-05-13
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