JP2006505533A5 - - Google Patents

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Publication number
JP2006505533A5
JP2006505533A5 JP2004537065A JP2004537065A JP2006505533A5 JP 2006505533 A5 JP2006505533 A5 JP 2006505533A5 JP 2004537065 A JP2004537065 A JP 2004537065A JP 2004537065 A JP2004537065 A JP 2004537065A JP 2006505533 A5 JP2006505533 A5 JP 2006505533A5
Authority
JP
Japan
Prior art keywords
pyrrolidin
urea
methyl
quinolin
diphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
JP2004537065A
Other languages
English (en)
Japanese (ja)
Other versions
JP2006505533A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2003/010154 external-priority patent/WO2004026836A2/en
Publication of JP2006505533A publication Critical patent/JP2006505533A/ja
Publication of JP2006505533A5 publication Critical patent/JP2006505533A5/ja
Abandoned legal-status Critical Current

Links

JP2004537065A 2002-09-17 2003-09-12 1−ピリジン−4−イル−尿素誘導体 Abandoned JP2006505533A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP0210417 2002-09-17
PCT/EP2003/010154 WO2004026836A2 (en) 2002-09-17 2003-09-12 1-pyridin-4-yl-urea derivatives

Publications (2)

Publication Number Publication Date
JP2006505533A JP2006505533A (ja) 2006-02-16
JP2006505533A5 true JP2006505533A5 (https=) 2006-10-19

Family

ID=32010909

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004537065A Abandoned JP2006505533A (ja) 2002-09-17 2003-09-12 1−ピリジン−4−イル−尿素誘導体

Country Status (13)

Country Link
US (1) US20060094716A1 (https=)
EP (1) EP1554249A2 (https=)
JP (1) JP2006505533A (https=)
KR (1) KR20050043967A (https=)
CN (1) CN1681789A (https=)
AU (1) AU2003270186A1 (https=)
BR (1) BR0314353A (https=)
CA (1) CA2496624A1 (https=)
MX (1) MXPA05002839A (https=)
NO (1) NO20050932L (https=)
RU (1) RU2005111589A (https=)
WO (1) WO2004026836A2 (https=)
ZA (1) ZA200502009B (https=)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1565436B1 (en) 2002-11-27 2012-04-25 Incyte Corporation 3-aminopyrrolidine derivatives as modulators of chemokine receptors
US7288538B2 (en) 2003-02-20 2007-10-30 Encysive Pharmaceuticals, Inc. Phenylenediamine urotensin-II receptor antagonists and CCR-9 antagonists
US7319111B2 (en) 2003-02-20 2008-01-15 Encysive Pharmaceuticals, Inc. Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists
US7320989B2 (en) 2003-02-28 2008-01-22 Encysive Pharmaceuticals, Inc. Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-II receptor antagonists
WO2004078114A2 (en) 2003-02-28 2004-09-16 Encysive Pharmaceuticals Inc. Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-ii receptor antagonists.
ATE440835T1 (de) 2003-03-06 2009-09-15 Glaxo Group Ltd Heterozyklische harnstoff-derivate für die behandlung von schmerzen.
EP1601665A2 (en) 2003-03-07 2005-12-07 Glaxo Group Limited Urea derivatives
GB0305426D0 (en) * 2003-03-08 2003-04-16 Glaxo Group Ltd Novel compounds
WO2005089380A2 (en) 2004-03-16 2005-09-29 The Regents Of The University Of California Reducing nephropathy with inhibitors of soluble epoxide hydrolase and epoxyeicosanoids
US20050026844A1 (en) 2003-04-03 2005-02-03 Regents Of The University Of California Inhibitors for the soluble epoxide hydrolase
AU2004275488A1 (en) * 2003-09-26 2005-04-07 Actelion Pharmaceuticals Ltd Pyridine derivatives and use thereof as urotensin II antagonists
BRPI0515979A (pt) * 2004-10-12 2008-08-12 Actelion Pharmaceuticals Ltd composto, processo para a preparação do mesmo, composições, uso de um ou mais compostos, e, método de tratamento de um paciente sofrendo de um distúrbio
JP2008517072A (ja) 2004-10-20 2008-05-22 ザ レジェンツ オブ ザ ユニバーシティー オブ カリフォルニア 可溶性エポキシド加水分解酵素の改良された阻害剤
JP4221447B1 (ja) 2005-09-21 2009-02-12 ファイザー・リミテッド ムスカリン様受容体アンタゴニストとしてのカルボキサミド誘導体
AR059826A1 (es) 2006-03-13 2008-04-30 Univ California Inhibidores de urea conformacionalmente restringidos de epoxido hidrolasa soluble
US8258301B2 (en) * 2007-05-15 2012-09-04 Boehringer Ingelheim International Gmbh Urotensin II receptor antagonists
MX2010012855A (es) * 2008-06-03 2010-12-21 Actelion Pharmaceuticals Ltd Derivados de [4-(1-amino-etil)-ciclohexil]-metil-amina y [6-(1-amino-etil)-tetrahidro-piran-3-il]-metil-amina como antibacterianos.
WO2012054093A2 (en) 2010-01-29 2012-04-26 The Regents Of The University Of California Acyl piperidine inhibitors of soluble epoxide hydrolase
RU2012146246A (ru) * 2010-03-31 2014-05-10 Актелион Фармасьютиклз Лтд Антибактериальные производные изохинолин-3-илмочевины
CN110015962B (zh) * 2011-01-28 2022-03-15 肯塔基大学研究基金会 茋类似物和治疗癌症的方法
CA2974784A1 (en) 2015-01-23 2016-07-28 Gvk Biosciences Private Limited Inhibitors of trka kinase
CN107056673B (zh) * 2016-09-09 2019-10-29 南京工业大学 一种3,4-二芳基马来酰亚胺衍生物及其制备方法与应用
CN106432039B (zh) * 2016-09-27 2019-02-22 南京工业大学 3,4-二芳基马来酰亚胺衍生物及其制备方法与应用
CN110862398B (zh) * 2018-08-27 2021-04-06 北京赛特明强医药科技有限公司 脲取代的芳环连二噁烷并喹唑啉或喹啉类化合物、组合物及其应用
HRP20241159T1 (hr) 2020-02-07 2024-12-06 Gasherbrum Bio, Inc. Heterociklički agonisti za glp-1
CN116368140A (zh) 2020-09-10 2023-06-30 加舒布鲁姆生物公司 杂环glp-1激动剂
CN120957993A (zh) 2023-02-16 2025-11-14 加舒布鲁姆生物公司 杂环glp-1激动剂
CN119219821A (zh) * 2024-12-03 2024-12-31 江苏金杉新材料有限公司 用于湿法冶金的苯乙烯系阴离子树脂及其制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR016817A1 (es) * 1997-08-14 2001-08-01 Smithkline Beecham Plc Derivados de fenilurea o feniltiourea, procedimiento para su preparacion, coleccion de compuestos, compuestos intermediarios, composicion farmaceutica,metodo de tratamiento y uso de dichos compuestos para la manufactura de un medicamento
AUPP003197A0 (en) * 1997-09-03 1997-11-20 Fujisawa Pharmaceutical Co., Ltd. New heterocyclic compounds
EP1150977B1 (en) * 1999-02-12 2004-08-25 SmithKline Beecham plc Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
IL157093A0 (en) * 2001-03-27 2004-02-08 Actelion Pharmaceuticals Ltd 1,2,3,4-tetrahydroisoquinolines derivatives as urotensin ii receptor antagonists
CA2473892C (en) * 2001-12-04 2010-09-21 Actelion Pharmaceuticals Ltd Novel quinoline derivatives

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