JP2005533860A5 - - Google Patents

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Publication number
JP2005533860A5
JP2005533860A5 JP2004524793A JP2004524793A JP2005533860A5 JP 2005533860 A5 JP2005533860 A5 JP 2005533860A5 JP 2004524793 A JP2004524793 A JP 2004524793A JP 2004524793 A JP2004524793 A JP 2004524793A JP 2005533860 A5 JP2005533860 A5 JP 2005533860A5
Authority
JP
Japan
Prior art keywords
composition
pharmaceutical composition
hydroxy
compound according
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2004524793A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005533860A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/023214 external-priority patent/WO2004011416A1/en
Publication of JP2005533860A publication Critical patent/JP2005533860A/ja
Publication of JP2005533860A5 publication Critical patent/JP2005533860A5/ja
Pending legal-status Critical Current

Links

JP2004524793A 2002-07-26 2003-07-25 結晶状β２アドレナリン作用性レセプターアゴニスト Pending JP2005533860A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US39892802P 2002-07-26 2002-07-26
US39867802P 2002-07-26 2002-07-26
PCT/US2003/023214 WO2004011416A1 (en) 2002-07-26 2003-07-25 CRYSTALLINE β2 ADRENERGIC RECEPTOR AGONIST

Publications (2)

Publication Number Publication Date
JP2005533860A JP2005533860A (ja) 2005-11-10
JP2005533860A5 true JP2005533860A5 (enExample) 2006-09-07

Family

ID=31191218

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004524793A Pending JP2005533860A (ja) 2002-07-26 2003-07-25 結晶状β２アドレナリン作用性レセプターアゴニスト

Country Status (11)

Country Link
US (1) US20050075271A1 (enExample)
EP (1) EP1532104A1 (enExample)
JP (1) JP2005533860A (enExample)
CN (1) CN100491342C (enExample)
AR (1) AR040661A1 (enExample)
AU (1) AU2003259229A1 (enExample)
BR (1) BR0312975A (enExample)
CA (1) CA2493128A1 (enExample)
MY (1) MY139296A (enExample)
TW (1) TW200409746A (enExample)
WO (1) WO2004011416A1 (enExample)

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PE20140960A1 (es) 2008-04-03 2014-08-15 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
BRPI0916997A2 (pt) 2008-08-06 2020-12-15 Boehringer Ingelheim International Gmbh Inibidor de dpp-4 e seu uso
AU2009290911A1 (en) 2008-09-10 2010-03-18 Boehringer Ingelheim International Gmbh Combination therapy for the treatment of diabetes and related conditions
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
EP2382216A1 (en) 2008-12-23 2011-11-02 Boehringer Ingelheim International GmbH Salt forms of organic compound
AR074990A1 (es) 2009-01-07 2011-03-02 Boehringer Ingelheim Int Tratamiento de diabetes en pacientes con un control glucemico inadecuado a pesar de la terapia con metformina
EP2228368A1 (en) 2009-03-12 2010-09-15 Almirall, S.A. Process for manufacturing 5-(2-{[6-(2,2-difluoro-2-phenylethoxy) hexyl]amino}-1-hydroxyethyl)-8-hydroxyquinolin-2(1H)-one
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
EA034869B1 (ru) 2009-11-27 2020-03-31 Бёрингер Ингельхайм Интернациональ Гмбх Лечение генотипированных пациентов с диабетом ингибиторами дпп-4, такими как линаглиптин
MX341025B (es) 2010-05-05 2016-08-04 Boehringer Ingelheim Int Gmbh * Terapia de combinacion.
PH12012502524A1 (en) 2010-06-24 2014-02-10 Boehringer Ingelheim Int Diabetes therapy
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US9034883B2 (en) 2010-11-15 2015-05-19 Boehringer Ingelheim International Gmbh Vasoprotective and cardioprotective antidiabetic therapy
EP3517539B1 (en) 2011-07-15 2022-12-14 Boehringer Ingelheim International GmbH Substituted dimeric quinazoline derivative, its preparation and its use in pharmaceutical compositions for the treatment of type i and ii diabetes
EP2578570A1 (en) 2011-10-07 2013-04-10 Almirall, S.A. Novel process for preparing 5-(2-{[6-(2,2-difluoro-2-phenylethoxy)hexyl]amino}-1(r)-hydroxyethyl)-8-hydroxyquinolin-2(1h)-one via novel intermediates of synthesis.
US9555001B2 (en) 2012-03-07 2017-01-31 Boehringer Ingelheim International Gmbh Pharmaceutical composition and uses thereof
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PL3517541T3 (pl) 2012-05-08 2020-12-28 Nicox Ophthalmics, Inc. Postać polimorficzna propionianu flutykazonu
US8765725B2 (en) 2012-05-08 2014-07-01 Aciex Therapeutics, Inc. Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof
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JP6224084B2 (ja) 2012-05-14 2017-11-01 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 糸球体上皮細胞関連障害及び／又はネフローゼ症候群の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体
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TW202140550A (zh) 2020-01-29 2021-11-01 瑞士商諾華公司 使用抗ｔｓｌｐ抗體治療炎性或阻塞性氣道疾病之方法

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