JP2005532359A5 - - Google Patents
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- Publication number
- JP2005532359A5 JP2005532359A5 JP2004511289A JP2004511289A JP2005532359A5 JP 2005532359 A5 JP2005532359 A5 JP 2005532359A5 JP 2004511289 A JP2004511289 A JP 2004511289A JP 2004511289 A JP2004511289 A JP 2004511289A JP 2005532359 A5 JP2005532359 A5 JP 2005532359A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- conh
- csnh
- aryl
- heteroaryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 125000000217 alkyl group Chemical group 0.000 claims 2
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 claims 2
- 150000001875 compounds Chemical class 0.000 claims 2
- 125000001255 4-fluorophenyl group Chemical group [H]C1=C([H])C(*)=C([H])C([H])=C1F 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- 125000001072 heteroaryl group Chemical group 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38655702P | 2002-06-06 | 2002-06-06 | |
| PCT/US2003/016876 WO2003104219A1 (en) | 2002-06-06 | 2003-05-29 | Nf-kb inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005532359A JP2005532359A (ja) | 2005-10-27 |
| JP2005532359A5 true JP2005532359A5 (https=) | 2006-07-20 |
Family
ID=29736178
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004511289A Withdrawn JP2005532359A (ja) | 2002-06-06 | 2003-05-29 | ＮＦ−κＢ阻害剤 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US7300952B2 (https=) |
| EP (1) | EP1532135B1 (https=) |
| JP (1) | JP2005532359A (https=) |
| AT (1) | ATE358673T1 (https=) |
| AU (1) | AU2003240935A1 (https=) |
| DE (1) | DE60312997T2 (https=) |
| ES (1) | ES2285125T3 (https=) |
| WO (1) | WO2003104219A1 (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006512313A (ja) | 2002-10-31 | 2006-04-13 | アムジェン インコーポレイテッド | 抗炎症剤 |
| US7696244B2 (en) | 2003-05-16 | 2010-04-13 | The Regents Of The University Of California | Compounds having activity in increasing ion transport by mutant-CFTR and uses thereof |
| KR100796965B1 (ko) * | 2004-05-04 | 2008-01-22 | 에프. 호프만-라 로슈 아게 | Ｉｋｋ 저해제로서의 티에노피리딘 |
| KR100822681B1 (ko) * | 2004-05-04 | 2008-04-17 | 에프. 호프만-라 로슈 아게 | Ｉｋｋ 억제제로서의 티에노피리다진 |
| EP1989203A2 (en) | 2006-02-16 | 2008-11-12 | Millennium Pharmaceuticals, Inc. | Alpha carbolines and uses thereof |
| WO2008069102A1 (ja) * | 2006-12-06 | 2008-06-12 | Calpis Co., Ltd. | 炎症性腸疾患予防治療剤 |
| CN102171204B (zh) | 2008-10-02 | 2014-08-20 | 旭化成制药株式会社 | 8位取代异喹啉衍生物及其用途 |
| WO2013118842A1 (ja) * | 2012-02-09 | 2013-08-15 | 国立大学法人東京医科歯科大学 | ベンゾチオフェン化合物、該化合物を有効成分とするオルタナティブオートファジー誘導剤及び抗癌剤、並びに抗癌活性を有する化合物をスクリーニングするための方法 |
| WO2016041972A1 (en) * | 2014-09-15 | 2016-03-24 | Ecole Polytechnique Federale De Lausanne (Epfl) | Benzothiophene, benzyloxybenzylidene and indoline derivatives useful for the treatment of tuberculosis |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4782080A (en) | 1985-09-16 | 1988-11-01 | Merck & Co., Inc. | N-alkenyl-2-hydroxybenzo(b)thiophene-3-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors |
| US6545027B1 (en) | 1995-06-07 | 2003-04-08 | Eli Lilly And Company | Methods of modulating NF-kB transcription factor |
| AU7261498A (en) | 1997-04-30 | 1998-11-24 | Eli Lilly And Company | Intermediates and processes for preparing benzo{b}thiophenes |
| EP1324759A4 (en) | 2000-10-12 | 2004-05-12 | Smithkline Beecham Corp | NF - G (K) B INHIBITORS |
-
2003
- 2003-05-29 AU AU2003240935A patent/AU2003240935A1/en not_active Abandoned
- 2003-05-29 DE DE60312997T patent/DE60312997T2/de not_active Expired - Fee Related
- 2003-05-29 JP JP2004511289A patent/JP2005532359A/ja not_active Withdrawn
- 2003-05-29 EP EP03731435A patent/EP1532135B1/en not_active Expired - Lifetime
- 2003-05-29 US US10/517,111 patent/US7300952B2/en not_active Expired - Fee Related
- 2003-05-29 ES ES03731435T patent/ES2285125T3/es not_active Expired - Lifetime
- 2003-05-29 WO PCT/US2003/016876 patent/WO2003104219A1/en not_active Ceased
- 2003-05-29 AT AT03731435T patent/ATE358673T1/de not_active IP Right Cessation