JP2005530733A - 乾燥粉末組成物 - Google Patents
乾燥粉末組成物 Download PDFInfo
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- JP2005530733A JP2005530733A JP2003585695A JP2003585695A JP2005530733A JP 2005530733 A JP2005530733 A JP 2005530733A JP 2003585695 A JP2003585695 A JP 2003585695A JP 2003585695 A JP2003585695 A JP 2003585695A JP 2005530733 A JP2005530733 A JP 2005530733A
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- 239000000843 powder Substances 0.000 title claims abstract description 47
- 239000000203 mixture Substances 0.000 title claims description 81
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- 150000001720 carbohydrates Chemical class 0.000 claims description 52
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- RFSUNEUAIZKAJO-ARQDHWQXSA-N Fructose Chemical compound OC[C@H]1O[C@](O)(CO)[C@@H](O)[C@@H]1O RFSUNEUAIZKAJO-ARQDHWQXSA-N 0.000 claims description 3
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- 239000001083 [(2R,3R,4S,5R)-1,2,4,5-tetraacetyloxy-6-oxohexan-3-yl] acetate Substances 0.000 claims description 2
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- 235000019698 starch Nutrition 0.000 description 1
- 229960005322 streptomycin Drugs 0.000 description 1
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- 150000008163 sugars Chemical class 0.000 description 1
- 229940124530 sulfonamide Drugs 0.000 description 1
- 150000003456 sulfonamides Chemical class 0.000 description 1
- 125000000472 sulfonyl group Chemical group *S(*)(=O)=O 0.000 description 1
- 239000003765 sweetening agent Substances 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 229940065721 systemic for obstructive airway disease xanthines Drugs 0.000 description 1
- 239000006068 taste-masking agent Substances 0.000 description 1
- 229960000195 terbutaline Drugs 0.000 description 1
- 235000019364 tetracycline Nutrition 0.000 description 1
- 150000003522 tetracyclines Chemical class 0.000 description 1
- 229940040944 tetracyclines Drugs 0.000 description 1
- 229960000278 theophylline Drugs 0.000 description 1
- LERNTVKEWCAPOY-DZZGSBJMSA-N tiotropium Chemical compound O([C@H]1C[C@@H]2[N+]([C@H](C1)[C@@H]1[C@H]2O1)(C)C)C(=O)C(O)(C=1SC=CC=1)C1=CC=CS1 LERNTVKEWCAPOY-DZZGSBJMSA-N 0.000 description 1
- 229940110309 tiotropium Drugs 0.000 description 1
- 229960005294 triamcinolone Drugs 0.000 description 1
- GFNANZIMVAIWHM-OBYCQNJPSA-N triamcinolone Chemical compound O=C1C=C[C@]2(C)[C@@]3(F)[C@@H](O)C[C@](C)([C@@]([C@H](O)C4)(O)C(=O)CO)[C@@H]4[C@@H]3CCC2=C1 GFNANZIMVAIWHM-OBYCQNJPSA-N 0.000 description 1
- 229960005486 vaccine Drugs 0.000 description 1
- 239000000811 xylitol Substances 0.000 description 1
- 235000010447 xylitol Nutrition 0.000 description 1
- HEBKCHPVOIAQTA-SCDXWVJYSA-N xylitol Chemical compound OC[C@H](O)[C@@H](O)[C@H](O)CO HEBKCHPVOIAQTA-SCDXWVJYSA-N 0.000 description 1
- 229960002675 xylitol Drugs 0.000 description 1
Images
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Pulmonology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Otolaryngology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medical Preparation Storing Or Oral Administration Devices (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| GBGB0208608.0A GB0208608D0 (en) | 2002-04-13 | 2002-04-13 | Composition |
| PCT/GB2003/001542 WO2003088943A1 (en) | 2002-04-13 | 2003-04-10 | Dry powder compositions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005530733A true JP2005530733A (ja) | 2005-10-13 |
| JP2005530733A5 JP2005530733A5 (enExample) | 2006-05-25 |
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| JP2003585695A Pending JP2005530733A (ja) | 2002-04-13 | 2003-04-10 | 乾燥粉末組成物 |
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| EP (1) | EP1494644A1 (enExample) |
| JP (1) | JP2005530733A (enExample) |
| KR (1) | KR20040099436A (enExample) |
| CN (1) | CN1658839A (enExample) |
| AR (1) | AR039409A1 (enExample) |
| AU (1) | AU2003217073A1 (enExample) |
| BR (1) | BR0309114A (enExample) |
| CA (1) | CA2481467A1 (enExample) |
| GB (1) | GB0208608D0 (enExample) |
| IL (1) | IL164420A0 (enExample) |
| IS (1) | IS7500A (enExample) |
| MX (1) | MXPA04010080A (enExample) |
| NO (1) | NO20044497L (enExample) |
| PL (1) | PL373294A1 (enExample) |
| RU (1) | RU2004130439A (enExample) |
| TW (1) | TW200404008A (enExample) |
| WO (1) | WO2003088943A1 (enExample) |
| ZA (1) | ZA200408245B (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009513531A (ja) * | 2003-07-11 | 2009-04-02 | グラクソ グループ リミテッド | 糖エステルを含む吸入可能医薬製剤 |
| JP2013512270A (ja) * | 2009-12-01 | 2013-04-11 | グラクソ グループ リミテッド | ムスカリン受容体拮抗薬およびβ２アドレナリン受容体作動薬の組み合わせ |
| JP2016519123A (ja) * | 2013-04-29 | 2016-06-30 | サノフィ・ソシエテ・アノニム | 吸入可能な医薬組成物およびそれらを収容した吸入器デバイス |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005507881A (ja) | 2001-09-17 | 2005-03-24 | グラクソ グループ リミテッド | 乾燥粉末医薬製剤 |
| SE526509C2 (sv) * | 2003-06-19 | 2005-09-27 | Microdrug Ag | Kombinerade doser av formoterol och budesonid separerade på en gemensam dosbädd |
| JP2009513529A (ja) * | 2003-07-11 | 2009-04-02 | グラクソ グループ リミテッド | ステアリン酸マグネシウムを含む医薬製剤 |
| AR049384A1 (es) | 2004-05-24 | 2006-07-26 | Glaxo Group Ltd | Derivados de purina |
| WO2006066907A1 (en) * | 2004-12-21 | 2006-06-29 | Glaxo Group Limited | Pharmaceutical formulations |
| NZ556709A (en) * | 2005-02-10 | 2009-09-25 | Glaxo Group Ltd | Process for making lactose utilizing pre-classification techniques and pharmaceutical formulations formed therefrom |
| GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
| JP2009545579A (ja) | 2006-08-01 | 2009-12-24 | グラクソ グループ リミテッド | ピラゾロ［３，４−ｂ］ピリジン化合物、及びｐｄｅ４阻害薬としてのその使用 |
| AU2015296024A1 (en) * | 2014-08-01 | 2017-03-23 | Luxena Pharmaceuticals, Inc. | Palonosetron formulations and uses thereof |
| PT109030B (pt) * | 2015-12-15 | 2019-09-25 | Hovione Farmaciência, S.A. | Preparação de partículas inaláveis de zafirlucaste |
| CN110237373B (zh) * | 2018-03-08 | 2023-06-02 | 润生药业有限公司 | 一种生产用于联合用药的药物载体的装置及方法 |
Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH04220268A (ja) * | 1990-12-19 | 1992-08-11 | Olympus Optical Co Ltd | バルーンカテーテル |
| WO2000028979A1 (de) * | 1998-11-13 | 2000-05-25 | Jago Research Ag | Trockenpulver zur inhalation |
| WO2001003673A1 (en) * | 1999-07-12 | 2001-01-18 | Quadrant Healthcare (Uk) Limited | Dry powder compositions |
| JP2001507357A (ja) * | 1996-12-31 | 2001-06-05 | クアドラント ホールディングス ケンブリッジ リミテッド | 粘膜送達用の生物活性物質の生物学的利用性を改良するための方法および組成物 |
| JP2001527087A (ja) * | 1997-12-23 | 2001-12-25 | クアドラント ホールディングス ケンブリッジ リミテッド | 固体輸送系において有用な炭水化物 |
| WO2002000198A1 (en) * | 2000-06-29 | 2002-01-03 | Glaxo Group Limited | Process for preparing and harvesting crystalline particles |
| WO2002015876A2 (en) * | 2000-08-21 | 2002-02-28 | Quadrant Healthcare (Uk) Limited | Amorphous carrier materials for drug delivery |
| JP2002510316A (ja) * | 1997-07-03 | 2002-04-02 | クアドラント ホールディングス ケンブリッジ リミテッド | 修飾グリコシド、これを含む組成物およびその使用方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR8007911A (pt) * | 1979-12-06 | 1981-06-16 | Glaxo Group Ltd | Inalador aperfeicoado |
| SE448277B (sv) * | 1985-04-12 | 1987-02-09 | Draco Ab | Indikeringsanordning vid en doseringsanordning for lekemedel |
| FI88112C (fi) * | 1985-07-30 | 1993-04-13 | Glaxo Group Ltd | Anordning foer administrering av laekemedel till patienter |
| GB9004781D0 (en) * | 1990-03-02 | 1990-04-25 | Glaxo Group Ltd | Device |
| WO2002043750A2 (en) * | 2000-12-01 | 2002-06-06 | Battelle Memorial Institute | Method for the stabilizing of biomolecules (e.g. insulin) in liquid formulations |
| GB0103630D0 (en) * | 2001-02-14 | 2001-03-28 | Glaxo Group Ltd | Chemical compounds |
-
2002
- 2002-04-13 GB GBGB0208608.0A patent/GB0208608D0/en not_active Ceased
-
2003
- 2003-04-10 AU AU2003217073A patent/AU2003217073A1/en not_active Abandoned
- 2003-04-10 RU RU2004130439/15A patent/RU2004130439A/ru not_active Application Discontinuation
- 2003-04-10 PL PL03373294A patent/PL373294A1/xx not_active Application Discontinuation
- 2003-04-10 EP EP03712461A patent/EP1494644A1/en not_active Withdrawn
- 2003-04-10 WO PCT/GB2003/001542 patent/WO2003088943A1/en not_active Ceased
- 2003-04-10 JP JP2003585695A patent/JP2005530733A/ja active Pending
- 2003-04-10 CA CA002481467A patent/CA2481467A1/en not_active Abandoned
- 2003-04-10 BR BR0309114-7A patent/BR0309114A/pt not_active IP Right Cessation
- 2003-04-10 US US10/511,042 patent/US20050244340A1/en not_active Abandoned
- 2003-04-10 CN CN038137194A patent/CN1658839A/zh active Pending
- 2003-04-10 KR KR10-2004-7016302A patent/KR20040099436A/ko not_active Withdrawn
- 2003-04-10 MX MXPA04010080A patent/MXPA04010080A/es unknown
- 2003-04-11 TW TW092108394A patent/TW200404008A/zh unknown
- 2003-04-11 AR ARP030101280A patent/AR039409A1/es not_active Application Discontinuation
-
2004
- 2004-10-05 IL IL16442004A patent/IL164420A0/xx unknown
- 2004-10-11 IS IS7500A patent/IS7500A/is unknown
- 2004-10-12 ZA ZA200408245A patent/ZA200408245B/xx unknown
- 2004-10-21 NO NO20044497A patent/NO20044497L/no not_active Application Discontinuation
Patent Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH04220268A (ja) * | 1990-12-19 | 1992-08-11 | Olympus Optical Co Ltd | バルーンカテーテル |
| JP2001507357A (ja) * | 1996-12-31 | 2001-06-05 | クアドラント ホールディングス ケンブリッジ リミテッド | 粘膜送達用の生物活性物質の生物学的利用性を改良するための方法および組成物 |
| JP2002510316A (ja) * | 1997-07-03 | 2002-04-02 | クアドラント ホールディングス ケンブリッジ リミテッド | 修飾グリコシド、これを含む組成物およびその使用方法 |
| JP2001527087A (ja) * | 1997-12-23 | 2001-12-25 | クアドラント ホールディングス ケンブリッジ リミテッド | 固体輸送系において有用な炭水化物 |
| WO2000028979A1 (de) * | 1998-11-13 | 2000-05-25 | Jago Research Ag | Trockenpulver zur inhalation |
| WO2001003673A1 (en) * | 1999-07-12 | 2001-01-18 | Quadrant Healthcare (Uk) Limited | Dry powder compositions |
| WO2002000198A1 (en) * | 2000-06-29 | 2002-01-03 | Glaxo Group Limited | Process for preparing and harvesting crystalline particles |
| WO2002015876A2 (en) * | 2000-08-21 | 2002-02-28 | Quadrant Healthcare (Uk) Limited | Amorphous carrier materials for drug delivery |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009513531A (ja) * | 2003-07-11 | 2009-04-02 | グラクソ グループ リミテッド | 糖エステルを含む吸入可能医薬製剤 |
| JP2013512270A (ja) * | 2009-12-01 | 2013-04-11 | グラクソ グループ リミテッド | ムスカリン受容体拮抗薬およびβ２アドレナリン受容体作動薬の組み合わせ |
| JP2016519123A (ja) * | 2013-04-29 | 2016-06-30 | サノフィ・ソシエテ・アノニム | 吸入可能な医薬組成物およびそれらを収容した吸入器デバイス |
Also Published As
| Publication number | Publication date |
|---|---|
| CN1658839A (zh) | 2005-08-24 |
| US20050244340A1 (en) | 2005-11-03 |
| RU2004130439A (ru) | 2005-06-10 |
| KR20040099436A (ko) | 2004-11-26 |
| IL164420A0 (en) | 2005-12-18 |
| IS7500A (is) | 2004-10-11 |
| GB0208608D0 (en) | 2002-05-22 |
| CA2481467A1 (en) | 2003-10-30 |
| WO2003088943A1 (en) | 2003-10-30 |
| AR039409A1 (es) | 2005-02-16 |
| AU2003217073A1 (en) | 2003-11-03 |
| EP1494644A1 (en) | 2005-01-12 |
| BR0309114A (pt) | 2005-02-01 |
| NO20044497L (no) | 2004-11-15 |
| ZA200408245B (en) | 2007-03-28 |
| TW200404008A (en) | 2004-03-16 |
| PL373294A1 (en) | 2005-08-22 |
| MXPA04010080A (es) | 2004-12-13 |
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