JP2005529160A - 糖尿病及び糖尿病−関連障害の処置のための化合物及び組成物 - Google Patents
糖尿病及び糖尿病−関連障害の処置のための化合物及び組成物 Download PDFInfo
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- JP2005529160A JP2005529160A JP2004509679A JP2004509679A JP2005529160A JP 2005529160 A JP2005529160 A JP 2005529160A JP 2004509679 A JP2004509679 A JP 2004509679A JP 2004509679 A JP2004509679 A JP 2004509679A JP 2005529160 A JP2005529160 A JP 2005529160A
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- 150000003505 terpenes Chemical class 0.000 description 1
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- 125000000999 tert-butyl group Chemical group [H]C([H])([H])C(*)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
- WROMPOXWARCANT-UHFFFAOYSA-N tfa trifluoroacetic acid Chemical compound OC(=O)C(F)(F)F.OC(=O)C(F)(F)F WROMPOXWARCANT-UHFFFAOYSA-N 0.000 description 1
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- RTKIYNMVFMVABJ-UHFFFAOYSA-L thimerosal Chemical compound [Na+].CC[Hg]SC1=CC=CC=C1C([O-])=O RTKIYNMVFMVABJ-UHFFFAOYSA-L 0.000 description 1
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- 150000003626 triacylglycerols Chemical class 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- BSVBQGMMJUBVOD-UHFFFAOYSA-N trisodium borate Chemical compound [Na+].[Na+].[Na+].[O-]B([O-])[O-] BSVBQGMMJUBVOD-UHFFFAOYSA-N 0.000 description 1
- RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 description 1
- 150000003672 ureas Chemical class 0.000 description 1
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- 239000011701 zinc Substances 0.000 description 1
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- 235000016804 zinc Nutrition 0.000 description 1
- XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical compound [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38459502P | 2002-05-31 | 2002-05-31 | |
| PCT/US2003/017193 WO2003101988A2 (en) | 2002-05-31 | 2003-05-30 | Compounds and compositions for the treatment of diabetes and diabetes-related disorders |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005529160A true JP2005529160A (ja) | 2005-09-29 |
| JP2005529160A5 JP2005529160A5 (https=) | 2006-06-29 |
Family
ID=29712061
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004509679A Withdrawn JP2005529160A (ja) | 2002-05-31 | 2003-05-30 | 糖尿病及び糖尿病−関連障害の処置のための化合物及び組成物 |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1513840B1 (https=) |
| JP (1) | JP2005529160A (https=) |
| AU (1) | AU2003273192A1 (https=) |
| CA (1) | CA2482345A1 (https=) |
| DE (1) | DE60308862T2 (https=) |
| ES (1) | ES2274268T3 (https=) |
| WO (1) | WO2003101988A2 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2007004781A (es) * | 2004-10-20 | 2007-05-11 | Applied Research Systems | Derivados de 3-arilamino piridina. |
| WO2013178320A1 (en) * | 2012-05-30 | 2013-12-05 | Merck Patent Gmbh | Solid state forms of n-((s)-2,3-dihydroxy-propyl)-3-(2-fluoro-4-iodo-phenylamino)-isonicotinamide |
| JOP20190086A1 (ar) | 2016-10-21 | 2019-04-18 | Novartis Ag | مشتقات نافثيريدينون جديدة واستخدامها في معالجة عدم انتظام ضربات القلب |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1022214A (en) * | 1963-01-31 | 1966-03-09 | Sterling Drug Inc | Novel 1,3-disubstituted-1,4-dihydro-4-oxo-1,7-naphthyridines and their preparation |
| JP3242792B2 (ja) * | 1994-08-05 | 2001-12-25 | 日本臓器製薬株式会社 | ナフチリジニウム誘導体 |
| KR100567649B1 (ko) * | 1996-09-25 | 2006-04-05 | 아스트라제네카 유케이 리미티드 | 혈관 내피 성장 인자와 같은 성장 인자의 효과를 억제하는 퀴놀린 유도체 |
-
2003
- 2003-05-30 ES ES03756326T patent/ES2274268T3/es not_active Expired - Lifetime
- 2003-05-30 CA CA002482345A patent/CA2482345A1/en not_active Abandoned
- 2003-05-30 EP EP03756326A patent/EP1513840B1/en not_active Expired - Lifetime
- 2003-05-30 JP JP2004509679A patent/JP2005529160A/ja not_active Withdrawn
- 2003-05-30 WO PCT/US2003/017193 patent/WO2003101988A2/en not_active Ceased
- 2003-05-30 AU AU2003273192A patent/AU2003273192A1/en not_active Abandoned
- 2003-05-30 DE DE60308862T patent/DE60308862T2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ES2274268T3 (es) | 2007-05-16 |
| WO2003101988A2 (en) | 2003-12-11 |
| DE60308862D1 (de) | 2006-11-16 |
| AU2003273192A8 (en) | 2003-12-19 |
| WO2003101988A3 (en) | 2004-04-15 |
| DE60308862T2 (de) | 2007-04-19 |
| EP1513840A2 (en) | 2005-03-16 |
| AU2003273192A1 (en) | 2003-12-19 |
| EP1513840B1 (en) | 2006-10-04 |
| CA2482345A1 (en) | 2003-12-11 |
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