JP2005525300A5 - - Google Patents
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- Publication number
- JP2005525300A5 JP2005525300A5 JP2003537793A JP2003537793A JP2005525300A5 JP 2005525300 A5 JP2005525300 A5 JP 2005525300A5 JP 2003537793 A JP2003537793 A JP 2003537793A JP 2003537793 A JP2003537793 A JP 2003537793A JP 2005525300 A5 JP2005525300 A5 JP 2005525300A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- solvate
- salt
- compound
- yloxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000003839 salts Chemical class 0.000 claims 10
- 239000012453 solvate Substances 0.000 claims 10
- 150000001875 compounds Chemical class 0.000 claims 6
- 239000002253 acid Substances 0.000 claims 4
- 125000003709 fluoroalkyl group Chemical group 0.000 claims 4
- 239000008249 pharmaceutical aerosol Substances 0.000 claims 3
- 239000003380 propellant Substances 0.000 claims 3
- -1 7,10,13,16-tetraoxaheptadec-1-yloxy Chemical group 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 2
- 239000000203 mixture Substances 0.000 claims 2
- 125000006545 (C1-C9) alkyl group Chemical group 0.000 claims 1
- OBRNDARFFFHCGE-PERKLWIXSA-N (S,S)-formoterol fumarate Chemical compound OC(=O)\C=C\C(O)=O.C1=CC(OC)=CC=C1C[C@H](C)NC[C@@H](O)C1=CC=C(O)C(NC=O)=C1.C1=CC(OC)=CC=C1C[C@H](C)NC[C@@H](O)C1=CC=C(O)C(NC=O)=C1 OBRNDARFFFHCGE-PERKLWIXSA-N 0.000 claims 1
- YFMFNYKEUDLDTL-UHFFFAOYSA-N 1,1,1,2,3,3,3-heptafluoropropane Chemical compound FC(F)(F)C(F)C(F)(F)F YFMFNYKEUDLDTL-UHFFFAOYSA-N 0.000 claims 1
- LVGUZGTVOIAKKC-UHFFFAOYSA-N 1,1,1,2-tetrafluoroethane Chemical group FCC(F)(F)F LVGUZGTVOIAKKC-UHFFFAOYSA-N 0.000 claims 1
- KUVIULQEHSCUHY-XYWKZLDCSA-N Beclometasone Chemical compound C1CC2=CC(=O)C=C[C@]2(C)[C@]2(Cl)[C@@H]1[C@@H]1C[C@H](C)[C@@](C(=O)COC(=O)CC)(OC(=O)CC)[C@@]1(C)C[C@@H]2O KUVIULQEHSCUHY-XYWKZLDCSA-N 0.000 claims 1
- VOVIALXJUBGFJZ-KWVAZRHASA-N Budesonide Chemical compound C1CC2=CC(=O)C=C[C@]2(C)[C@@H]2[C@@H]1[C@@H]1C[C@H]3OC(CCC)O[C@@]3(C(=O)CO)[C@@]1(C)C[C@@H]2O VOVIALXJUBGFJZ-KWVAZRHASA-N 0.000 claims 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 1
- GIIZNNXWQWCKIB-UHFFFAOYSA-N Serevent Chemical compound C1=C(O)C(CO)=CC(C(O)CNCCCCCCOCCCCC=2C=CC=CC=2)=C1 GIIZNNXWQWCKIB-UHFFFAOYSA-N 0.000 claims 1
- NDAUXUAQIAJITI-UHFFFAOYSA-N albuterol Chemical compound CC(C)(C)NCC(O)C1=CC=C(O)C(CO)=C1 NDAUXUAQIAJITI-UHFFFAOYSA-N 0.000 claims 1
- 229950000210 beclometasone dipropionate Drugs 0.000 claims 1
- 229960004436 budesonide Drugs 0.000 claims 1
- KYKAJFCTULSVSH-UHFFFAOYSA-N chloro(fluoro)methane Chemical compound F[C]Cl KYKAJFCTULSVSH-UHFFFAOYSA-N 0.000 claims 1
- 229910052731 fluorine Inorganic materials 0.000 claims 1
- 125000001153 fluoro group Chemical group F* 0.000 claims 1
- NBVXSUQYWXRMNV-UHFFFAOYSA-N fluoromethane Chemical compound FC NBVXSUQYWXRMNV-UHFFFAOYSA-N 0.000 claims 1
- 229960000289 fluticasone propionate Drugs 0.000 claims 1
- WMWTYOKRWGGJOA-CENSZEJFSA-N fluticasone propionate Chemical compound C1([C@@H](F)C2)=CC(=O)C=C[C@]1(C)[C@]1(F)[C@@H]2[C@@H]2C[C@@H](C)[C@@](C(=O)SCF)(OC(=O)CC)[C@@]2(C)C[C@@H]1O WMWTYOKRWGGJOA-CENSZEJFSA-N 0.000 claims 1
- 229960000193 formoterol fumarate Drugs 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- OEXHQOGQTVQTAT-JRNQLAHRSA-N ipratropium Chemical compound O([C@H]1C[C@H]2CC[C@@H](C1)[N@@+]2(C)C(C)C)C(=O)C(CO)C1=CC=CC=C1 OEXHQOGQTVQTAT-JRNQLAHRSA-N 0.000 claims 1
- 229960001888 ipratropium Drugs 0.000 claims 1
- 239000011859 microparticle Substances 0.000 claims 1
- SONNWYBIRXJNDC-VIFPVBQESA-N phenylephrine Chemical compound CNC[C@H](O)C1=CC=CC(O)=C1 SONNWYBIRXJNDC-VIFPVBQESA-N 0.000 claims 1
- 229960001802 phenylephrine Drugs 0.000 claims 1
- 229960002052 salbutamol Drugs 0.000 claims 1
- 229960005018 salmeterol xinafoate Drugs 0.000 claims 1
- TXEYQDLBPFQVAA-UHFFFAOYSA-N tetrafluoromethane Chemical group FC(F)(F)F TXEYQDLBPFQVAA-UHFFFAOYSA-N 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0125127.1A GB0125127D0 (en) | 2001-10-19 | 2001-10-19 | Compounds |
| PCT/EP2002/011635 WO2003035237A2 (en) | 2001-10-19 | 2002-10-17 | Compounds for use as surfactants |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005525300A JP2005525300A (ja) | 2005-08-25 |
| JP2005525300A5 true JP2005525300A5 (https=) | 2006-01-05 |
| JP4223954B2 JP4223954B2 (ja) | 2009-02-12 |
Family
ID=9924153
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003537793A Expired - Fee Related JP4223954B2 (ja) | 2001-10-19 | 2002-10-17 | 界面活性剤として使用するための化合物 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7321059B2 (https=) |
| EP (1) | EP1436007B1 (https=) |
| JP (1) | JP4223954B2 (https=) |
| AT (1) | ATE291928T1 (https=) |
| AU (1) | AU2002340578A1 (https=) |
| DE (1) | DE60203528T2 (https=) |
| ES (1) | ES2238606T3 (https=) |
| GB (1) | GB0125127D0 (https=) |
| WO (1) | WO2003035237A2 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60231428D1 (de) | 2001-12-21 | 2009-04-16 | 3M Innovative Properties Co | Medizinische aerosolzusammensetzungen mit einem funktionalisierten polyethylenglykol-hilfsstoff |
| KR20040086370A (ko) | 2002-02-13 | 2004-10-08 | 글락소 그룹 리미티드 | 계면활성제로서 사용되는 카르복실산 화합물 |
| CN102416179B (zh) | 2010-09-28 | 2014-05-07 | 益得生物科技股份有限公司 | 用于哮喘的吸入性复方组合物 |
| US10745606B2 (en) | 2017-08-15 | 2020-08-18 | Saudi Arabian Oil Company | Oil-based drilling fluid compositions which include layered double hydroxides as rheology modifiers |
| US10876039B2 (en) | 2017-08-15 | 2020-12-29 | Saudi Arabian Oil Company | Thermally stable surfactants for oil based drilling fluids |
| US10647903B2 (en) | 2017-08-15 | 2020-05-12 | Saudi Arabian Oil Company | Oil-based drilling fluid compositions which include layered double hydroxides as rheology modifiers and amino amides as emulsifiers |
| US10640696B2 (en) | 2017-08-15 | 2020-05-05 | Saudi Arabian Oil Company | Oil-based drilling fluids for high pressure and high temperature drilling operations |
| US10793762B2 (en) | 2017-08-15 | 2020-10-06 | Saudi Arabian Oil Company | Layered double hydroxides for oil-based drilling fluids |
| US10988659B2 (en) | 2017-08-15 | 2021-04-27 | Saudi Arabian Oil Company | Layered double hydroxides for oil-based drilling fluids |
| US10676658B2 (en) | 2017-08-15 | 2020-06-09 | Saudi Arabian Oil Company | Oil-based drilling fluids for high pressure and high temperature drilling operations |
| US10870788B2 (en) | 2017-08-15 | 2020-12-22 | Saudi Arabian Oil Company | Thermally stable surfactants for oil based drilling fluids |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4352789A (en) * | 1980-03-17 | 1982-10-05 | Minnesota Mining And Manufacturing Company | Aerosol compositions containing finely divided solid materials |
| DE3903663C1 (https=) * | 1989-02-08 | 1990-09-27 | Huels Ag, 4370 Marl, De | |
| IL97065A (en) | 1990-02-02 | 1994-01-25 | Fisons Plc | Repellent preparations for aerosol |
| AU654813B2 (en) * | 1990-03-23 | 1994-11-24 | Minnesota Mining And Manufacturing Company | The use of soluble fluorosurfactants for the preparation of metered-dose aerosol formulations |
| DE69101639T2 (de) | 1990-06-27 | 1994-10-06 | Minnesota Mining & Mfg | Anwendung von löslichen fluorhaltigen tensiden zur herstellung von aerosol-präparaten mit dosierter abgabe. |
| US5126123A (en) * | 1990-06-28 | 1992-06-30 | Glaxo, Inc. | Aerosol drug formulations |
| CA2085884C (en) | 1990-06-29 | 2001-12-04 | Asit Somani | Pressurized hydrofluorocarbon aerosol compositions |
| US5376359A (en) * | 1992-07-07 | 1994-12-27 | Glaxo, Inc. | Method of stabilizing aerosol formulations |
| GB9419536D0 (en) | 1994-09-28 | 1994-11-16 | Glaxo Inc | Medicaments |
| US6451287B1 (en) * | 2000-05-26 | 2002-09-17 | Smithkline Beecham Corporation | Fluorinated copolymer surfactants and use thereof in aerosol compositions |
| US7217409B2 (en) | 2000-09-22 | 2007-05-15 | Smithkline Beecham Corporation | Alkanoic acid derivatives |
| WO2003013610A2 (en) * | 2001-08-03 | 2003-02-20 | Glaxo Group Limited | Surfactant compounds and uses thereof |
-
2001
- 2001-10-19 GB GBGB0125127.1A patent/GB0125127D0/en not_active Ceased
-
2002
- 2002-10-17 JP JP2003537793A patent/JP4223954B2/ja not_active Expired - Fee Related
- 2002-10-17 AT AT02774728T patent/ATE291928T1/de not_active IP Right Cessation
- 2002-10-17 AU AU2002340578A patent/AU2002340578A1/en not_active Abandoned
- 2002-10-17 ES ES02774728T patent/ES2238606T3/es not_active Expired - Lifetime
- 2002-10-17 DE DE60203528T patent/DE60203528T2/de not_active Expired - Fee Related
- 2002-10-17 EP EP02774728A patent/EP1436007B1/en not_active Expired - Lifetime
- 2002-10-17 WO PCT/EP2002/011635 patent/WO2003035237A2/en not_active Ceased
- 2002-10-17 US US10/492,606 patent/US7321059B2/en not_active Expired - Fee Related
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