JP2005520795A5 - - Google Patents

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Publication number
JP2005520795A5
JP2005520795A5 JP2003551316A JP2003551316A JP2005520795A5 JP 2005520795 A5 JP2005520795 A5 JP 2005520795A5 JP 2003551316 A JP2003551316 A JP 2003551316A JP 2003551316 A JP2003551316 A JP 2003551316A JP 2005520795 A5 JP2005520795 A5 JP 2005520795A5
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JP
Japan
Prior art keywords
hsp90
high affinity
assay
compound
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003551316A
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English (en)
Japanese (ja)
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JP2005520795A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/039993 external-priority patent/WO2003050295A2/en
Publication of JP2005520795A publication Critical patent/JP2005520795A/ja
Publication of JP2005520795A5 publication Critical patent/JP2005520795A5/ja
Pending legal-status Critical Current

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JP2003551316A 2001-12-12 2002-12-12 Hsp90阻害活性を有するプリン類似体 Pending JP2005520795A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34076201P 2001-12-12 2001-12-12
PCT/US2002/039993 WO2003050295A2 (en) 2001-12-12 2002-12-12 Assays and implements for determining and modulating hsp90 binding activity

Publications (2)

Publication Number Publication Date
JP2005520795A JP2005520795A (ja) 2005-07-14
JP2005520795A5 true JP2005520795A5 (https=) 2006-02-02

Family

ID=23334832

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003551316A Pending JP2005520795A (ja) 2001-12-12 2002-12-12 Hsp90阻害活性を有するプリン類似体

Country Status (6)

Country Link
US (2) US20050074457A1 (https=)
EP (1) EP1519735A4 (https=)
JP (1) JP2005520795A (https=)
AU (1) AU2002364566B2 (https=)
CA (1) CA2468202A1 (https=)
WO (1) WO2003050295A2 (https=)

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CN103539769B (zh) * 2006-08-11 2016-03-16 斯特拉斯堡大学 用作激酶抑制剂和hsp90抑制剂的大环化合物
CN104127878A (zh) 2007-03-14 2014-11-05 恩多塞特公司 结合配体连接的微管溶素递药缀合物
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WO2001072779A1 (en) * 2000-03-24 2001-10-04 Duke University Characterization of grp94-ligand interactions and purification, screening, and therapeutic methods relating thereto

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