JP2005516986A5 - - Google Patents

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Publication number
JP2005516986A5
JP2005516986A5 JP2003565415A JP2003565415A JP2005516986A5 JP 2005516986 A5 JP2005516986 A5 JP 2005516986A5 JP 2003565415 A JP2003565415 A JP 2003565415A JP 2003565415 A JP2003565415 A JP 2003565415A JP 2005516986 A5 JP2005516986 A5 JP 2005516986A5
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JP
Japan
Prior art keywords
phenyl
amino
oxime
carbonyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2003565415A
Other languages
English (en)
Japanese (ja)
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JP2005516986A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2003/003222 external-priority patent/WO2003065989A2/en
Publication of JP2005516986A publication Critical patent/JP2005516986A/ja
Publication of JP2005516986A5 publication Critical patent/JP2005516986A5/ja
Withdrawn legal-status Critical Current

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JP2003565415A 2002-02-08 2003-02-04 (オキシム)カルバモイル脂肪酸アミド加水分解酵素インヒビター Withdrawn JP2005516986A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35530202P 2002-02-08 2002-02-08
PCT/US2003/003222 WO2003065989A2 (en) 2002-02-08 2003-02-04 (oxime)carbamoyl fatty acid amide hydrolase inhibitors

Publications (2)

Publication Number Publication Date
JP2005516986A JP2005516986A (ja) 2005-06-09
JP2005516986A5 true JP2005516986A5 (https=) 2006-02-02

Family

ID=27734499

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003565415A Withdrawn JP2005516986A (ja) 2002-02-08 2003-02-04 (オキシム)カルバモイル脂肪酸アミド加水分解酵素インヒビター

Country Status (6)

Country Link
US (2) US6949574B2 (https=)
EP (1) EP1472215A4 (https=)
JP (1) JP2005516986A (https=)
AU (1) AU2003210824A1 (https=)
PL (1) PL373970A1 (https=)
WO (1) WO2003065989A2 (https=)

Families Citing this family (38)

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AU2002338329B2 (en) 2001-03-27 2006-09-07 The Regents Of The University Of California Methods, compounds, and compositions for reducing body fat and modulating fatty acid metabolism
US20050054730A1 (en) * 2001-03-27 2005-03-10 The Regents Of The University Of California Compounds, compositions and treatment of oleoylethanolamide-like modulators of PPARalpha
AU2002311784B2 (en) * 2001-03-29 2007-11-22 Michael Davis Acute pharmacologic augmentation of psychotherapy with enhancers of learning or conditioning
EP1558591B1 (en) 2002-10-07 2014-05-07 The Regents of The University of California Modulation of anxiety through blockade of anandamide hydrolysis
US7765162B2 (en) * 2002-10-07 2010-07-27 Mastercard International Incorporated Method and system for conducting off-line and on-line pre-authorized payment transactions
FR2850377B1 (fr) * 2003-01-23 2009-02-20 Sanofi Synthelabo Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
FR2860514A1 (fr) * 2003-10-03 2005-04-08 Sanofi Synthelabo Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
JP2007509066A (ja) * 2003-10-16 2007-04-12 ザ・レジェンツ・オブ・ザ・ユニバーシティ・オブ・カリフォルニア 体脂肪を減らし、食欲を抑制し、脂肪酸代謝を調節するための食物および他の組成物、化合物ならびに方法
FR2865205B1 (fr) * 2004-01-16 2006-02-24 Sanofi Synthelabo Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique
US20060084659A1 (en) * 2004-10-19 2006-04-20 Michael Davis Augmentation of psychotherapy with cannabinoid reuptake inhibitors
TW200633990A (en) 2004-11-18 2006-10-01 Takeda Pharmaceuticals Co Amide compound
AR055831A1 (es) 2004-12-30 2007-09-12 Janssen Pharmaceutica Nv Pepirazinilureas y piperidinilureas como moduladores de hidrolasa de amida de acidos grasos
ES2528674T3 (es) 2005-02-17 2015-02-11 Astellas Pharma Inc. Piperidina y carboxilatos de piperacina como inhibidores de FAAH
WO2006116773A2 (en) * 2005-04-28 2006-11-02 The Regents Of The University Of California Methods, compositions, and compounds for modulation of monoacylglycerol lipase, pain, and stress-related disorders
EP1954137A4 (en) * 2005-11-18 2008-12-17 Janssen Pharmaceutica Nv 2-KETO-OXAZOLE AS MODULATORS OF FATTY ACID AMIDHYDROLASE
US20070155707A1 (en) * 2005-12-29 2007-07-05 Kadmus Pharmaceuticals, Inc. Ionizable inhibitors of fatty acid amide hydrolase
US20110172230A1 (en) 2006-08-23 2011-07-14 Takahiro Ishii Urea compound or salt thereof
US20080119549A1 (en) * 2006-11-20 2008-05-22 N.V. Organon Metabolically-stabilized inhibitors of fatty acid amide hydrolase
CA2679741A1 (en) * 2007-03-15 2008-09-18 Sun Pharma Advanced Research Company Ltd. Novel prodrugs
ES2575954T3 (es) * 2007-10-11 2016-07-04 The Regents Of The University Of California Composiciones y métodos de inhibición de la amidasa ácida hidrolizante de la N-aciletanolamina
EP2062578A1 (en) * 2007-11-12 2009-05-27 Institut National De La Sante Et De La Recherche Medicale (Inserm) Novel use of chemical compounds for the treatment of AIDS
TW201006791A (en) * 2008-05-15 2010-02-16 Sigma Tau Ind Farmaceuti Oxime carbamoyl derivatives as modulators of fatty acid amide hydrolase
US8207226B1 (en) 2008-06-03 2012-06-26 Alcon Research, Ltd. Use of FAAH antagonists for treating dry eye and ocular pain
TWI434842B (zh) 2008-07-14 2014-04-21 Astellas Pharma Inc Azole compounds
MX2011004704A (es) 2008-11-06 2011-05-30 Astellas Pharma Inc Compuesto de carbamato o sal del mismo.
WO2011085216A2 (en) 2010-01-08 2011-07-14 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating parkinson's disease and restless legs syndrome
WO2011123719A2 (en) 2010-03-31 2011-10-06 Ironwood Pharmaceuticals, Inc. Use of faah inhibitors for treating abdominal, visceral and pelvic pain
UA108233C2 (uk) 2010-05-03 2015-04-10 Модулятори активності гідролази амідів жирних кислот
EP2632912A4 (en) * 2010-10-28 2014-05-07 Scripps Research Inst ANTI-CANCER-SERINHYDROLASE-INHIBITING CARBAMATE
AU2012340519B2 (en) 2011-11-22 2017-09-14 Fondazione Istituto Italiano Di Tecnologia Disubstituted beta-lactones as inhibitors of N-acylethanolamine acid amidase (NAAA)
EP2931291B1 (en) 2012-12-11 2021-10-20 The McLean Hospital Corporation Xenon treatment as an adjunct to psychotherapy for psychiatric disorders
US9474271B2 (en) 2013-01-18 2016-10-25 Research Foundation Of The City University Of New York Method for enhancing amidohydrolase activity of fatty acid amide hydrolase
WO2014144836A2 (en) 2013-03-15 2014-09-18 The Regents Of The University Of California Carbamate derivatives of lactam based n-acylethanolamine acid amidase (naaa) inhibitors
WO2014144547A2 (en) 2013-03-15 2014-09-18 The Regents Of The University Of California Amide derivatives of lactam based n-acylethanolamine acid amidase (naaa) inhibitors
CN105418460B (zh) * 2014-08-11 2017-04-12 苏州鹏旭医药科技有限公司 匹莫范色林及其类似化合物中间体,其制备方法和制备匹莫范色林及其类似化合物的方法
JP7200261B2 (ja) * 2017-12-05 2023-01-06 スージョウ ポンシュー ファーマテック カンパニー リミテッド エラゴリクスを作製するプロセス
US10414721B1 (en) 2018-06-04 2019-09-17 University Of Bern Inhibitor of endocannabinoid cellular reuptake

Family Cites Families (6)

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GB841141A (en) * 1955-08-29 1960-07-13 Union Carbide Corp Naphthyl esters of n-alkyl-substituted carbamic acids and insecticidal compositions containing the same
NL302370A (https=) * 1962-12-22
DE1232947B (de) * 1963-12-09 1967-01-26 Fahlberg List Chemische Veb Verfahren zur Herstellung von Ketoximcarbanilaten aus Ketoximen und Arylisocyanaten
WO1990001874A1 (en) * 1988-08-24 1990-03-08 Teijin Limited Oxime derivatives and herbicides containing the same as an active ingredient
GB9719530D0 (en) * 1997-09-12 1997-11-19 Smithkline Beecham Plc Novel compounds
MXPA03009850A (es) * 2001-04-27 2004-02-12 Bristol Myers Squibb Co Inhibidores de bisarilimidazolil de hidrolasa de amida del acido graso.

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