JP2004532828A5 - - Google Patents

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Publication number
JP2004532828A5
JP2004532828A5 JP2002572952A JP2002572952A JP2004532828A5 JP 2004532828 A5 JP2004532828 A5 JP 2004532828A5 JP 2002572952 A JP2002572952 A JP 2002572952A JP 2002572952 A JP2002572952 A JP 2002572952A JP 2004532828 A5 JP2004532828 A5 JP 2004532828A5
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JP
Japan
Prior art keywords
tramadol
pharmaceutical composition
milligrams
cis
composition according
Prior art date
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JP2002572952A
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English (en)
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JP2004532828A (ja
JP4377585B2 (ja
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Priority claimed from PCT/US2002/007928 external-priority patent/WO2002074241A2/en
Publication of JP2004532828A publication Critical patent/JP2004532828A/ja
Publication of JP2004532828A5 publication Critical patent/JP2004532828A5/ja
Application granted granted Critical
Publication of JP4377585B2 publication Critical patent/JP4377585B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Claims (14)

  1. 効量のトラマドール物質を含んでなる射精遅延のための医薬組成物
  2. 前記トラマドール物質はトラマドール又は医薬として許容可能なトラマドールの塩である請求項1に記載の医薬組成物
  3. 前記トラマドール物質は(±)シス‐トラマドール又は医薬として許容可能な(±)シス‐トラマドールの塩である請求項2に記載の医薬組成物
  4. 約10ミリグラムから約50ミリグラムの量の前記トラマドール又は前記医薬として許容可能な(±)シス‐トラマドールの塩を含んでなる請求項3に記載の医薬組成物
  5. 約15ミリグラムから約35ミリグラムの量の前記トラマドール又は前記医薬として許容可能な(±)シス‐トラマドールの塩を含んでなる請求項4に記載の医薬組成物
  6. 約25ミリグラムの量の前記トラマドール又は前記医薬として許容可能な(±)シス‐トラマドールの塩を含んでなる請求項5に記載の医薬組成物
  7. 前記シス‐トラマドールの、又は前記医薬として許容可能なシス‐トラマドールの塩の(+)光学異性体を含んでなる請求項3に記載の医薬組成物
  8. 前記シス‐トラマドールの、又は前記医薬として許容可能なシス‐トラマドールの塩の(−)光学異性体を含んでなる請求項3に記載の医薬組成物
  9. 前記トラマドール物質は塩酸(±)シス‐トラマドールである請求項3に記載の医薬組成物
  10. 約10ミリグラムから約50ミリグラムの量の前記塩酸トラマドールを含んでなる請求項9に記載の医薬組成物
  11. 約15ミリグラムから約35ミリグラムの量の前記塩酸トラマドールを含んでなる請求
    項10に記載の医薬組成物
  12. 約25ミリグラムの量の前記塩酸トラマドールを含んでなる請求項11に記載の医薬組成物
  13. 経口投与されることを特徴とする請求項1乃至請求項12のいずれか1項に記載の医薬組成物
  14. 早漏を治療するための請求項1乃至請求項13のいずれか1項に記載の医薬組成物
JP2002572952A 2001-03-16 2002-03-15 射精遅延の方法 Expired - Fee Related JP4377585B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27680601P 2001-03-16 2001-03-16
PCT/US2002/007928 WO2002074241A2 (en) 2001-03-16 2002-03-15 Method of delaying ejaculation

Publications (3)

Publication Number Publication Date
JP2004532828A JP2004532828A (ja) 2004-10-28
JP2004532828A5 true JP2004532828A5 (ja) 2006-01-05
JP4377585B2 JP4377585B2 (ja) 2009-12-02

Family

ID=23058139

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002572952A Expired - Fee Related JP4377585B2 (ja) 2001-03-16 2002-03-15 射精遅延の方法

Country Status (18)

Country Link
US (2) US6974839B2 (ja)
EP (1) EP1397126B9 (ja)
JP (1) JP4377585B2 (ja)
KR (1) KR100908350B1 (ja)
CN (1) CN1289071C (ja)
AT (1) ATE326957T1 (ja)
AU (1) AU2002252361C1 (ja)
CA (2) CA2758923A1 (ja)
CY (1) CY1107478T1 (ja)
DE (1) DE60211689T2 (ja)
DK (1) DK1397126T5 (ja)
ES (1) ES2265495T3 (ja)
HK (1) HK1068549A1 (ja)
MX (1) MXPA03008372A (ja)
NZ (1) NZ528935A (ja)
PT (1) PT1397126E (ja)
WO (1) WO2002074241A2 (ja)
ZA (1) ZA200308067B (ja)

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WO2004078143A2 (en) * 2003-03-05 2004-09-16 The Brigham And Women's Hospital Inc. Methods for identification and uses of anti-inflammatory receptors for eicosapentaenoic acid analogs
US8841345B2 (en) 2003-03-21 2014-09-23 Nexmed Holdings, Inc. Compositions and methods for treatment of premature ejaculation
AU2003903597A0 (en) * 2003-07-11 2003-07-24 Jakov Vaisman Treatment of premature ejaculation
US8604082B2 (en) * 2005-12-13 2013-12-10 Trinity Laboratories, Inc. Method to treat premature ejaculation in humans
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US20100120780A1 (en) * 2007-04-19 2010-05-13 Chandra Ulagaraj Singh Treatments for premature ejaculation in humans
US20090005319A1 (en) * 2007-07-01 2009-01-01 Barone Jr Frank V Topical compositions for delaying ejaculation and methods of using the same
KR101103118B1 (ko) * 2007-11-02 2012-01-04 동아제약주식회사 신규한 1,3-디히드로-5-이소벤조퓨란카르보니트릴 유도체 화합물 및 이를 함유하는 조루증 치료용 약학조성물
US8147848B2 (en) 2009-08-26 2012-04-03 Allergan, Inc. Method for treating premature ejaculation with a botulinum neurotoxin
GR1007315B (el) * 2010-04-19 2011-06-14 Uni-Pharma Κλεων Τσετης Φαρμακευτικα Εργαστηρια Αβεε Με Δ.Τ. Uni-Pharma Abee, Υγρομορφη παρεντερικης χορηγησης συνθεση που περιλαμβανει τραμαδολη hci και παρακεταμολη
US10702485B2 (en) 2011-07-09 2020-07-07 Syntrix Biosystems Inc. Compositions and methods for overcoming resistance to tramadol
US20180071269A1 (en) 2015-08-12 2018-03-15 Tianxin Wang Therapeutical methods, formulations and nutraceutical formulations
US11000488B2 (en) 2019-03-22 2021-05-11 Syntrix Biosystems Inc. Treating pain using desmetramadol

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