JP2004517069A5 - - Google Patents
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- Publication number
- JP2004517069A5 JP2004517069A5 JP2002543486A JP2002543486A JP2004517069A5 JP 2004517069 A5 JP2004517069 A5 JP 2004517069A5 JP 2002543486 A JP2002543486 A JP 2002543486A JP 2002543486 A JP2002543486 A JP 2002543486A JP 2004517069 A5 JP2004517069 A5 JP 2004517069A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- triazol
- pharmaceutically acceptable
- phenyl
- compound according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0027987.7A GB0027987D0 (en) | 2000-11-16 | 2000-11-16 | Compounds |
| PCT/GB2001/005036 WO2002040476A1 (en) | 2000-11-16 | 2001-11-15 | Pyridyl-substituted triazoles as tgf inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004517069A JP2004517069A (ja) | 2004-06-10 |
| JP2004517069A5 true JP2004517069A5 (https=) | 2005-12-22 |
Family
ID=9903300
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002543486A Withdrawn JP2004517069A (ja) | 2000-11-16 | 2001-11-15 | Ｔｇｆ阻害剤としてのピリジル置換トリアゾール類 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20040152738A1 (https=) |
| EP (1) | EP1335916A1 (https=) |
| JP (1) | JP2004517069A (https=) |
| AU (1) | AU2002214163A1 (https=) |
| GB (1) | GB0027987D0 (https=) |
| WO (1) | WO2002040476A1 (https=) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0127430D0 (en) * | 2001-11-15 | 2002-01-09 | Smithkline Beecham Corp | Compounds |
| GB0127433D0 (en) * | 2001-11-15 | 2002-01-09 | Smithkline Beecham Corp | Compounds |
| AR039241A1 (es) | 2002-04-04 | 2005-02-16 | Biogen Inc | Heteroarilos trisustituidos y metodos para su produccion y uso de los mismos |
| GB0217783D0 (en) * | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | Compounds |
| GB0217780D0 (en) * | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | Compounds |
| GB0217786D0 (en) * | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | Compounds |
| WO2004013135A1 (en) * | 2002-07-31 | 2004-02-12 | Smithkline Beecham Corporation | 2-phenylpyridin-4-yl derivatives as alk5 inhibitors |
| GB0217787D0 (en) * | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | C ompounds |
| UA80295C2 (en) | 2002-09-06 | 2007-09-10 | Biogen Inc | Pyrazolopyridines and using the same |
| PL375973A1 (en) * | 2002-09-18 | 2005-12-12 | Pfizer Products Inc. | Novel isothiazole and isoxazole compounds as transforming growth factor (tgf) inhibitors |
| CA2497971A1 (en) | 2002-09-18 | 2004-04-01 | Pfizer Products Inc. | Triazole derivatives as transforming growth factor (tgf) inhibitors |
| MXPA05002332A (es) * | 2002-09-18 | 2005-06-08 | Pfizer Prod Inc | Nuevos compuestos de oxazol y tiazol como inhibidores del factor de crecimiento transformador (tgf). |
| HRP20050247A2 (en) | 2002-09-18 | 2005-10-31 | Pfizer Products Inc. | Pyrazole derivatives as transforming growth factor (tgf) inhibitors |
| JP4547271B2 (ja) * | 2002-09-18 | 2010-09-22 | ファイザー・プロダクツ・インク | トランスフォーミング増殖因子（ｔｇｆ）阻害剤としての新規イミダゾール化合物 |
| CA2513086A1 (en) * | 2002-12-19 | 2004-07-08 | Scios Inc. | Treatment of obesity and associated conditions with tgf-.beta. inhibitors |
| PA8595001A1 (es) | 2003-03-04 | 2004-09-28 | Pfizer Prod Inc | Nuevos compuestos heteroaromaticos condensados que son inhibidores del factor de crecimiento transforante (tgf) |
| GB0313915D0 (en) * | 2003-06-16 | 2003-07-23 | Smithkline Beecham Corp | Compounds |
| NZ549003A (en) * | 2004-03-05 | 2009-07-31 | Taisho Pharmaceutical Co Ltd | Thiazole derivative as an ALK5 inhibitor |
| JP5149177B2 (ja) | 2005-07-25 | 2013-02-20 | シンタ ファーマシューティカルズ コーポレーション | 増殖性疾患の治療のための、チューブリンポリマー化の１，２，３−トリアゾール系抑制剤 |
| WO2007070866A2 (en) * | 2005-12-16 | 2007-06-21 | Alcon, Inc. | Control of intraocular pressure using alk5 modulation agents |
| US8586581B2 (en) | 2009-12-17 | 2013-11-19 | Hoffmann-La Roche Inc | Ethynyl compounds useful for treatment of CNS disorders |
| CA2874764C (en) | 2012-05-30 | 2022-11-01 | Cornell University | Generation of functional and durable endothelial cells from human amniotic fluid-derived cells |
| WO2014197421A1 (en) | 2013-06-05 | 2014-12-11 | Biotime, Inc. | Compositions and methods for induced tissue regeneration in mammalian species |
| US11078462B2 (en) | 2014-02-18 | 2021-08-03 | ReCyte Therapeutics, Inc. | Perivascular stromal cells from primate pluripotent stem cells |
| RU2688665C2 (ru) | 2014-04-22 | 2019-05-22 | Университет Базель | Новый способ получения производных триазина, пиримидина и пиридина |
| US10240127B2 (en) | 2014-07-03 | 2019-03-26 | ReCyte Therapeutics, Inc. | Exosomes from clonal progenitor cells |
| CA3202332A1 (en) | 2015-12-07 | 2017-06-15 | Agex Therapeutics, Inc. | Methods for the re-derivation of diverse pluripotent stem cell-derived brown fat cells |
| WO2022251359A1 (en) * | 2021-05-26 | 2022-12-01 | Theravance Biopharma R&D Ip, Llc | Bicyclic inhibitors of alk5 and methods of use |
| US12240830B2 (en) * | 2021-08-13 | 2025-03-04 | Bisichem Co., Ltd. | Fused ring heteroaryl compounds and use thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2003525201A (ja) * | 1998-08-20 | 2003-08-26 | スミスクライン・ビーチャム・コーポレイション | 新規な置換トリアゾール化合物 |
-
2000
- 2000-11-16 GB GBGB0027987.7A patent/GB0027987D0/en not_active Ceased
-
2001
- 2001-11-15 JP JP2002543486A patent/JP2004517069A/ja not_active Withdrawn
- 2001-11-15 US US10/416,680 patent/US20040152738A1/en not_active Abandoned
- 2001-11-15 AU AU2002214163A patent/AU2002214163A1/en not_active Abandoned
- 2001-11-15 EP EP01982621A patent/EP1335916A1/en not_active Withdrawn
- 2001-11-15 WO PCT/GB2001/005036 patent/WO2002040476A1/en not_active Ceased
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