JP2004510749A - No阻害またはtnf阻害に関連した疾病の治療におけるpparデルタ活性化因子の使用 - Google Patents

No阻害またはtnf阻害に関連した疾病の治療におけるpparデルタ活性化因子の使用 Download PDF

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JP2004510749A
JP2004510749A JP2002532257A JP2002532257A JP2004510749A JP 2004510749 A JP2004510749 A JP 2004510749A JP 2002532257 A JP2002532257 A JP 2002532257A JP 2002532257 A JP2002532257 A JP 2002532257A JP 2004510749 A JP2004510749 A JP 2004510749A
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ppardelta
tnf
synthase
methyl
disease
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JP2002532257A
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JP2004510749A5 (enExample
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バカン,ケヴィン,ウィリアム
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Glaxo Group Ltd
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Glaxo Group Ltd
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/4211,3-Oxazoles, e.g. pemoline, trimethadione
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
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JP2002532257A 2000-10-05 2001-10-02 No阻害またはtnf阻害に関連した疾病の治療におけるpparデルタ活性化因子の使用 Pending JP2004510749A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0024362.6A GB0024362D0 (en) 2000-10-05 2000-10-05 Medicaments
PCT/GB2001/004370 WO2002028433A2 (en) 2000-10-05 2001-10-02 Use of a ppar delta activator in the treatment of diseases related to no inhibit ion or tnf inhibition

Publications (2)

Publication Number Publication Date
JP2004510749A true JP2004510749A (ja) 2004-04-08
JP2004510749A5 JP2004510749A5 (enExample) 2005-12-22

Family

ID=9900710

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002532257A Pending JP2004510749A (ja) 2000-10-05 2001-10-02 No阻害またはtnf阻害に関連した疾病の治療におけるpparデルタ活性化因子の使用

Country Status (6)

Country Link
US (1) US20040029938A1 (enExample)
EP (1) EP1324773A2 (enExample)
JP (1) JP2004510749A (enExample)
AU (1) AU2001292044A1 (enExample)
GB (1) GB0024362D0 (enExample)
WO (1) WO2002028433A2 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20040063897A (ko) 2001-09-14 2004-07-14 툴라릭, 인코포레이티드 링크된 바이아릴 화합물
EP1637161A4 (en) * 2003-04-22 2007-06-27 Astellas Pharma Inc MEANS FOR THE TREATMENT OF NEURODEGENERATIVE ILLNESSES OF THE BRAIN WITH PPAR [delta] AGONIST
KR100849747B1 (ko) * 2003-05-20 2008-07-31 노파르티스 아게 과산화소체 증식체-활성화 수용체의 리간드로서의 n-아실질소 헤테로환
KR20060018241A (ko) * 2003-06-06 2006-02-28 에프. 호프만-라 로슈 아게 아닐린 유도체
RU2344135C2 (ru) 2003-07-02 2009-01-20 Ф.Хоффманн-Ля Рош Аг Тиазолзамещенные индолилпроизводные и их применение в качестве модуляторов ppar
SG138623A1 (en) * 2004-04-01 2008-01-28 Aventis Pharmaceuticals Inc Us Use of ppr delta agonists for treating demyelinating diseases
US7126825B2 (en) * 2004-12-07 2006-10-24 Cleavage Enterprise Co., Ltd. Combined chip/heat-dissipating metal plate and method for manufacturing the same
RU2012109545A (ru) * 2009-08-14 2013-09-20 Серенис Терапьютикс С.А. Использование лигандов ppar дельта для лечения или предотвращения воспалений или заболеваний, связанных с метаболизмом/выработкой энергии

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997028149A1 (en) * 1996-02-02 1997-08-07 Merck & Co., Inc. Method for raising hdl cholesterol levels
JP4427825B2 (ja) * 1997-07-24 2010-03-10 アステラス製薬株式会社 コレステロール低下作用を有する医薬組成物
GB9914977D0 (en) * 1999-06-25 1999-08-25 Glaxo Group Ltd Chemical compounds
EP1170008A1 (en) * 2000-07-07 2002-01-09 Chemotherapeutisches Forschungsinstitut Georg-Speyer-Haus Valproic acid and derivatives thereof as histone deacetylase inhibitors

Also Published As

Publication number Publication date
EP1324773A2 (en) 2003-07-09
GB0024362D0 (en) 2000-11-22
AU2001292044A1 (en) 2002-04-15
WO2002028433A3 (en) 2002-08-15
WO2002028433A2 (en) 2002-04-11
US20040029938A1 (en) 2004-02-12

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