JP2004504399A5 - - Google Patents
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- Publication number
- JP2004504399A5 JP2004504399A5 JP2002514137A JP2002514137A JP2004504399A5 JP 2004504399 A5 JP2004504399 A5 JP 2004504399A5 JP 2002514137 A JP2002514137 A JP 2002514137A JP 2002514137 A JP2002514137 A JP 2002514137A JP 2004504399 A5 JP2004504399 A5 JP 2004504399A5
- Authority
- JP
- Japan
- Prior art keywords
- branched
- straight
- substituents
- carbon atoms
- saturated alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000001424 substituent group Chemical group 0.000 description 25
- 125000000217 alkyl group Chemical group 0.000 description 22
- 125000003118 aryl group Chemical group 0.000 description 20
- 125000004432 carbon atom Chemical group C* 0.000 description 20
- 125000004417 unsaturated alkyl group Chemical group 0.000 description 18
- 150000001875 compounds Chemical class 0.000 description 13
- 125000004043 oxo group Chemical group O=* 0.000 description 12
- 150000003839 salts Chemical class 0.000 description 9
- 239000008194 pharmaceutical composition Substances 0.000 description 3
- -1 amino, hydroxyl Chemical group 0.000 description 2
- 125000004093 cyano group Chemical group *C#N 0.000 description 2
- 125000006841 cyclic skeleton Chemical group 0.000 description 2
- 229910052736 halogen Inorganic materials 0.000 description 2
- 125000005843 halogen group Chemical group 0.000 description 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 description 2
- 125000000446 sulfanediyl group Chemical group *S* 0.000 description 2
- 239000003814 drug Substances 0.000 description 1
- 150000002148 esters Chemical group 0.000 description 1
- 230000005764 inhibitory process Effects 0.000 description 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 description 1
- 229910052757 nitrogen Inorganic materials 0.000 description 1
- 125000004433 nitrogen atom Chemical group N* 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22027000P | 2000-07-24 | 2000-07-24 | |
| US60/220,270 | 2000-07-24 | ||
| PCT/US2001/023633 WO2002008231A2 (en) | 2000-07-24 | 2001-07-24 | Biologically active macrolides, compositions, and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2004504399A JP2004504399A (ja) | 2004-02-12 |
| JP2004504399A5 true JP2004504399A5 (enExample) | 2008-09-04 |
| JP4980542B2 JP4980542B2 (ja) | 2012-07-18 |
Family
ID=22822844
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002514137A Expired - Fee Related JP4980542B2 (ja) | 2000-07-24 | 2001-07-24 | 生物活性マクロライド、組成物、及びそれらの使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (5) | US7144918B2 (enExample) |
| EP (1) | EP1303522B1 (enExample) |
| JP (1) | JP4980542B2 (enExample) |
| AT (1) | ATE504589T1 (enExample) |
| AU (2) | AU8083401A (enExample) |
| CA (1) | CA2415611C (enExample) |
| DE (1) | DE60144376D1 (enExample) |
| WO (1) | WO2002008231A2 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU8083401A (en) * | 2000-07-24 | 2002-02-05 | Us Health | Biologically active macrolides, compositions, and uses thereof |
| WO2004009079A1 (en) | 2002-07-24 | 2004-01-29 | The Government Of The United States Of America, Represented By The Secretary, Dept. Of Health And Human Services | Chondropsin-class antitumor v-atpase inhibitor compounds, compositions and methods of use thereof |
| WO2010144611A2 (en) * | 2009-06-10 | 2010-12-16 | 3-V Biosciences, Inc. | Antivirals that target transporters, carriers, and ion channels |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1000053B1 (en) * | 1997-07-25 | 2004-06-30 | THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES | Macrocyclic lactones, compositions, and methods of use |
| US7381744B1 (en) | 1999-03-05 | 2008-06-03 | The United States Of America As Represented By The Department Of Health And Human Services | Method of treating osteoporosis comprising vacuolar-type (H+)-ATPase-inhibiting compounds |
| AU8083401A (en) * | 2000-07-24 | 2002-02-05 | Us Health | Biologically active macrolides, compositions, and uses thereof |
-
2001
- 2001-07-24 AU AU8083401A patent/AU8083401A/xx active Pending
- 2001-07-24 JP JP2002514137A patent/JP4980542B2/ja not_active Expired - Fee Related
- 2001-07-24 WO PCT/US2001/023633 patent/WO2002008231A2/en not_active Ceased
- 2001-07-24 DE DE60144376T patent/DE60144376D1/de not_active Expired - Lifetime
- 2001-07-24 AT AT01959257T patent/ATE504589T1/de not_active IP Right Cessation
- 2001-07-24 US US10/333,710 patent/US7144918B2/en not_active Expired - Lifetime
- 2001-07-24 AU AU2001280834A patent/AU2001280834B2/en not_active Ceased
- 2001-07-24 EP EP20010959257 patent/EP1303522B1/en not_active Expired - Lifetime
- 2001-07-24 CA CA 2415611 patent/CA2415611C/en not_active Expired - Fee Related
-
2006
- 2006-05-16 US US11/435,189 patent/US7790764B2/en not_active Expired - Fee Related
-
2010
- 2010-08-06 US US12/851,691 patent/US8741947B2/en not_active Expired - Fee Related
-
2014
- 2014-05-12 US US14/275,336 patent/US9139595B2/en not_active Expired - Fee Related
-
2015
- 2015-09-10 US US14/849,798 patent/US9820965B2/en not_active Expired - Fee Related
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