JP2003523325A5 - - Google Patents

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Publication number
JP2003523325A5
JP2003523325A5 JP2001548102A JP2001548102A JP2003523325A5 JP 2003523325 A5 JP2003523325 A5 JP 2003523325A5 JP 2001548102 A JP2001548102 A JP 2001548102A JP 2001548102 A JP2001548102 A JP 2001548102A JP 2003523325 A5 JP2003523325 A5 JP 2003523325A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
abl
pdgf
acceptable salt
tyrosine kinase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001548102A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003523325A (ja
Filing date
Publication date
Priority claimed from IT1999MI002711A external-priority patent/ITMI992711A1/it
Application filed filed Critical
Publication of JP2003523325A publication Critical patent/JP2003523325A/ja
Publication of JP2003523325A5 publication Critical patent/JP2003523325A5/ja
Pending legal-status Critical Current

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JP2001548102A 1999-12-27 2000-12-22 受容体チロシンキナーゼ阻害剤とα１−酸性糖タンパク質結合性有機化合物との組合せ Pending JP2003523325A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IT99A002711 1999-12-27
IT1999MI002711A ITMI992711A1 (it) 1999-12-27 1999-12-27 Composti organici
PCT/EP2000/013161 WO2001047507A2 (en) 1999-12-27 2000-12-22 Combinations of receptor tyrosine kinase inhibitor with an a1-acidic glycoprotein binding compound

Publications (2)

Publication Number Publication Date
JP2003523325A JP2003523325A (ja) 2003-08-05
JP2003523325A5 true JP2003523325A5 (https=) 2008-02-14

Family

ID=11384195

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001548102A Pending JP2003523325A (ja) 1999-12-27 2000-12-22 受容体チロシンキナーゼ阻害剤とα１−酸性糖タンパク質結合性有機化合物との組合せ

Country Status (18)

Country Link
US (2) US20030125343A1 (https=)
EP (1) EP1250140B1 (https=)
JP (1) JP2003523325A (https=)
CN (1) CN1304005C (https=)
AR (1) AR030179A1 (https=)
AT (1) ATE432069T1 (https=)
AU (1) AU2171901A (https=)
BR (1) BR0016817A (https=)
CA (1) CA2394944A1 (https=)
CO (1) CO5271710A1 (https=)
DE (1) DE60042283D1 (https=)
ES (1) ES2326307T3 (https=)
HK (1) HK1050993A1 (https=)
IT (1) ITMI992711A1 (https=)
PE (1) PE20010991A1 (https=)
PT (1) PT1250140E (https=)
TW (1) TWI246917B (https=)
WO (1) WO2001047507A2 (https=)

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US20060052387A1 (en) * 2002-06-26 2006-03-09 Marsh Clay B Organic compounds
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CA2538523A1 (en) * 2003-09-19 2005-03-31 Novartis Ag Treatment of gastrointestinal stromal tumors with imatinib and midostaurin
TW200517114A (en) * 2003-10-15 2005-06-01 Combinatorx Inc Methods and reagents for the treatment of immunoinflammatory disorders
US8048883B2 (en) † 2004-02-11 2011-11-01 Natco Pharma Limited Polymorphic form of imatinib mesylate and a process for its preparation
EP1768982A2 (en) 2004-06-29 2007-04-04 Amgen Inc. Pyrolo [2,3-d] pyrimidines that modulate ack1 and lck activity
BRPI0514094A (pt) * 2004-08-02 2008-05-27 Osi Pharm Inc composto, composição, e, método de tratamento de distúrbio hiperproliferativo
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US20060275365A1 (en) * 2005-06-07 2006-12-07 Thomas Backensfeld Immediate-release and high-drug-load pharmaceutical formulations of micronised (4-chlorophenyl) [4-(4-pyridylmethyl)phthalazin-1-yl] and salts thereof
US20070059359A1 (en) * 2005-06-07 2007-03-15 Thomas Backensfeld Immediate-release and high-drug-load pharmaceutical formulations of non-micronised (4-chlorophenyl)[4-(4-pyridylmethyl)phthalazin-1-yl] and salts thereof
DE602006015994D1 (de) * 2005-06-23 2010-09-16 Novartis Ag Verfahren zur behandlung von soliden tumoren einschliesslich der verabreichung einer kombination mit imatinib und einem effluxpumpenhemmer
ATE475660T1 (de) 2005-12-21 2010-08-15 Abbott Lab Antivirale verbindungen
US7915411B2 (en) 2005-12-21 2011-03-29 Abbott Laboratories Anti-viral compounds
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EA016611B1 (ru) * 2006-04-20 2012-06-29 Янссен Фармацевтика Н.В. Способ лечения мастоцитоза
EP2043651A2 (en) * 2006-07-05 2009-04-08 Exelixis, Inc. Methods of using igf1r and abl kinase modulators
US8236950B2 (en) 2006-12-20 2012-08-07 Abbott Laboratories Anti-viral compounds
JP5571387B2 (ja) 2007-01-11 2014-08-13 クリティカル・アウトカム・テクノロジーズ・インコーポレイテッド 癌の治療のための化合物および方法
US20080248548A1 (en) * 2007-04-09 2008-10-09 Flynn Daniel L Modulation of protein functionalities
BRPI0817946A2 (pt) * 2007-09-25 2015-05-05 Teva Pharma Composições de imatinibe estável
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US9273077B2 (en) 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
PT2300013T (pt) 2008-05-21 2017-10-31 Ariad Pharma Inc Derivados de fósforo como inibidores de cinases
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AR083797A1 (es) 2010-11-10 2013-03-20 Novartis Ag Succinato de dimetil-amida del acido 7-ciclopentil-2-(5-piperazin-1-il-piridin-2-il-amino)-7h-pirrolo-[2,3-d]pirimidin-6-carboxilico, proceso para prepararla, intermediarios de dicha sintesis y proceso de preparacion de los mismos
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KR102529049B1 (ko) 2013-08-14 2023-05-08 노파르티스 아게 암의 치료를 위한 조합 요법
WO2017078647A1 (en) 2015-11-05 2017-05-11 Koçak Farma Ilaç Ve Kimya Sanayi Anonim Şirketi Pharmaceutical compositions of imatinib
EP3257499A1 (en) 2016-06-17 2017-12-20 Vipharm S.A. Process for preparation of imatinib methanesulfonate capsules
AU2020211071A1 (en) 2019-01-23 2021-07-15 Novartis Ag New crystalline forms of a succinate salt of 7-Cyclopentyl-2-(5-piperazin-1-yl-pyridin-2-ylamino)-7H-pyrrolo[2,3-d]pyrimidine -6-carboxylic acid dimethylamide

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US5587459A (en) * 1994-08-19 1996-12-24 Regents Of The University Of Minnesota Immunoconjugates comprising tyrosine kinase inhibitors
US5750493A (en) * 1995-08-30 1998-05-12 Raymond F. Schinazi Method to improve the biological and antiviral activity of protease inhibitors
US20030069174A1 (en) * 1997-03-10 2003-04-10 Ludwig Pichler Use of human alpha1-acid glycoprotein for producing a pharmaceutical preparation
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EP1201668A4 (en) * 1999-07-13 2003-05-21 Kyowa Hakko Kogyo Kk Staurosporine DERIVATIVES
EP1382339B1 (en) * 1999-12-10 2007-12-05 Pfizer Products Inc. Compositions containing pyrrolo ¬2,3-d pyrimidine derivatives

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