JP2003510320A5 - - Google Patents
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- Publication number
- JP2003510320A5 JP2003510320A5 JP2001526531A JP2001526531A JP2003510320A5 JP 2003510320 A5 JP2003510320 A5 JP 2003510320A5 JP 2001526531 A JP2001526531 A JP 2001526531A JP 2001526531 A JP2001526531 A JP 2001526531A JP 2003510320 A5 JP2003510320 A5 JP 2003510320A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- alkyl
- sulfonyl
- aryl
- heteroaryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 C*S(N(*)C(*)(*)C(N(*)*)=O)(=O)=O Chemical compound C*S(N(*)C(*)(*)C(N(*)*)=O)(=O)=O 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP99810871.6 | 1999-09-28 | ||
| EP99810871A EP1088815A1 (en) | 1999-09-28 | 1999-09-28 | Pharmaceutically active sulfonyl amino acid derivatives |
| PCT/IB2000/001382 WO2001023379A1 (en) | 1999-09-28 | 2000-09-28 | Pharmaceutically active sulfonyl amino acid derivatives |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012033338A Division JP2012111777A (ja) | 1999-09-28 | 2012-02-17 | 薬剤活性のあるスルホニルアミノ酸誘導体 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2003510320A JP2003510320A (ja) | 2003-03-18 |
| JP2003510320A5 true JP2003510320A5 (cg-RX-API-DMAC7.html) | 2011-09-01 |
| JP5068913B2 JP5068913B2 (ja) | 2012-11-07 |
Family
ID=8243051
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001526531A Expired - Fee Related JP5068913B2 (ja) | 1999-09-28 | 2000-09-28 | 薬剤活性のあるスルホニルアミノ酸誘導体 |
| JP2012033338A Withdrawn JP2012111777A (ja) | 1999-09-28 | 2012-02-17 | 薬剤活性のあるスルホニルアミノ酸誘導体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012033338A Withdrawn JP2012111777A (ja) | 1999-09-28 | 2012-02-17 | 薬剤活性のあるスルホニルアミノ酸誘導体 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US7638538B1 (cg-RX-API-DMAC7.html) |
| EP (2) | EP1088815A1 (cg-RX-API-DMAC7.html) |
| JP (2) | JP5068913B2 (cg-RX-API-DMAC7.html) |
| AT (1) | ATE440838T1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU783651B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2384997A1 (cg-RX-API-DMAC7.html) |
| DE (1) | DE60042831D1 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2332575T3 (cg-RX-API-DMAC7.html) |
| IL (1) | IL148874A0 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2001023379A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1088821A1 (en) * | 1999-09-28 | 2001-04-04 | Applied Research Systems ARS Holding N.V. | Pharmaceutically active sulfonamide derivatives |
| EP1088815A1 (en) * | 1999-09-28 | 2001-04-04 | Applied Research Systems ARS Holding N.V. | Pharmaceutically active sulfonyl amino acid derivatives |
| US6657070B2 (en) | 2000-12-13 | 2003-12-02 | Wyeth | Production of chirally pure α-amino acids and N-sulfonyl α-amino acids |
| EA009035B1 (ru) * | 2000-12-13 | 2007-10-26 | Уиет | Получение гетероциклических сульфонамидных ингибиторов бета-амилоида |
| KR20040007497A (ko) | 2001-04-16 | 2004-01-24 | 에자이 가부시키가이샤 | 신규 1ｈ-인다졸 화합물 |
| AU2002331253B2 (en) * | 2001-07-23 | 2008-04-03 | Laboratoires Serono Sa | Arylsulfonamide derivatives as C-JUN-N-terminal kinases (JNK'S) inhibitors |
| JP4414881B2 (ja) | 2002-05-31 | 2010-02-10 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピラゾール化合物およびこれを含んでなる医薬組成物 |
| IL165265A0 (en) | 2002-06-11 | 2005-12-18 | Wyeth Corp | Substituted phenylsulfonamide inhibitors of beta amyloid production |
| WO2004031123A1 (en) * | 2002-10-02 | 2004-04-15 | Aventis Pharma Deutschland Gmbh | Hydroxyphenylundecane derivatives, a process for their production and their use |
| CL2004000647A1 (es) | 2003-03-31 | 2005-02-04 | Wyeth Corp | Compuestos derivados de heterociclicos de sulfonamida que contienen fluoro y trifluoro alquilo; composicion farmaceutica; kit farmaceutico; procedimiento de preparacion; y su uso como inhibidores de beta amiloides para tratar alzheimer, angiopatia am |
| US7705052B2 (en) | 2003-09-12 | 2010-04-27 | Merck Serono Sa | Sulfonamide derivatives for the treatment of diabetes |
| US7399778B2 (en) | 2004-01-16 | 2008-07-15 | Wyeth | Heterocyclic sulfonamide inhibitors of beta amyloid production containing an azole |
| US20060094753A1 (en) | 2004-10-29 | 2006-05-04 | Alcon, Inc. | Use of inhibitors of Jun N-terminal kinases for the treatment of glaucomatous retinopathy and ocular diseases |
| US7803824B2 (en) | 2004-10-29 | 2010-09-28 | Alcon, Inc. | Use of inhibitors of Jun N-terminal kinases to treat glaucoma |
| US20060223807A1 (en) | 2005-03-29 | 2006-10-05 | University Of Massachusetts Medical School, A Massachusetts Corporation | Therapeutic methods for type I diabetes |
| BRPI0613042A2 (pt) | 2005-07-15 | 2010-12-14 | Serono Lab | inibidores de jnk para o tratamento de endometriose |
| KR20080044836A (ko) | 2005-07-15 | 2008-05-21 | 라보라뚜와르 세로노 에스. 에이. | 자궁내막증 치료용 ｊｎｋ 억제제 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL6509157A (cg-RX-API-DMAC7.html) * | 1964-07-24 | 1966-01-25 | ||
| AU473887B2 (en) * | 1975-05-30 | 1975-07-10 | Kyorin Pharmaceutical Co. Ltd. | Novel pyrazole derivatives |
| JPH09104672A (ja) * | 1995-08-08 | 1997-04-22 | Ono Pharmaceut Co Ltd | ヒドロキサム酸誘導体 |
| PT757984E (pt) * | 1995-08-08 | 2003-02-28 | Ono Pharmaceutical Co | Derivados de acido hidroxamico uteis para inibir a gelatinase |
| NZ333825A (en) * | 1996-07-22 | 2000-10-27 | Monsanto Co | Metalloprotease inhibitors particularly MMP-13 |
| DE69828783T2 (de) * | 1997-03-04 | 2006-01-12 | Pharmacia Corp. | Hydroxamsäure-sulfonamid-derivate mit amidiertem aromatischen ring |
| US6043083A (en) * | 1997-04-28 | 2000-03-28 | Davis; Roger J. | Inhibitors of the JNK signal transduction pathway and methods of use |
| AU758570B2 (en) * | 1997-07-15 | 2003-03-27 | Mediquest Therapeutics, Inc. | Novel polyamine analogues as therapeutic and diagnostic agents |
| US6646149B1 (en) * | 1997-07-15 | 2003-11-11 | Nicolaas M. J. Vermeulin | Polyamine analogues as therapeutic and diagnostic agents |
| SK11692000A3 (sk) * | 1998-02-04 | 2001-02-12 | Novartis Ag | Sulfonylaminoderiváty, ktoré inhibujú metaloproteinázy degradujúce matricu, spôsob ich prípravy a farmaceutická kompozícia, ktorá ich obsahuje |
| JPH11236369A (ja) * | 1998-02-23 | 1999-08-31 | Kotobuki Seiyaku Kk | スルホンアミド誘導体及びその製造法並びにこれを含有する医薬組成物 |
| JPH11246527A (ja) * | 1998-03-02 | 1999-09-14 | Shionogi & Co Ltd | Ｍｍｐ−８阻害剤 |
| CA2318004A1 (en) * | 1999-09-15 | 2001-03-15 | Oridigm Corporation | Novel polyamine analogues as therapeutic and diagnostic agents |
| EP1088815A1 (en) * | 1999-09-28 | 2001-04-04 | Applied Research Systems ARS Holding N.V. | Pharmaceutically active sulfonyl amino acid derivatives |
| WO2001027108A1 (en) * | 1999-10-08 | 2001-04-19 | Bristol-Myers Squibb Pharma Company | AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
-
1999
- 1999-09-28 EP EP99810871A patent/EP1088815A1/en not_active Withdrawn
-
2000
- 2000-09-28 EP EP00960922A patent/EP1218375B1/en not_active Expired - Lifetime
- 2000-09-28 JP JP2001526531A patent/JP5068913B2/ja not_active Expired - Fee Related
- 2000-09-28 ES ES00960922T patent/ES2332575T3/es not_active Expired - Lifetime
- 2000-09-28 DE DE60042831T patent/DE60042831D1/de not_active Expired - Lifetime
- 2000-09-28 AU AU73075/00A patent/AU783651B2/en not_active Ceased
- 2000-09-28 AT AT00960922T patent/ATE440838T1/de not_active IP Right Cessation
- 2000-09-28 CA CA002384997A patent/CA2384997A1/en not_active Abandoned
- 2000-09-28 WO PCT/IB2000/001382 patent/WO2001023379A1/en not_active Ceased
- 2000-09-28 IL IL14887400A patent/IL148874A0/xx unknown
- 2000-09-28 US US10/088,090 patent/US7638538B1/en not_active Expired - Fee Related
-
2012
- 2012-02-17 JP JP2012033338A patent/JP2012111777A/ja not_active Withdrawn
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