JP2003501443A - ニューロメジンｂおよびソマトスタチンレセプターアゴニスト - Google Patents
ニューロメジンｂおよびソマトスタチンレセプターアゴニストInfo
- Publication number
- JP2003501443A JP2003501443A JP2001502467A JP2001502467A JP2003501443A JP 2003501443 A JP2003501443 A JP 2003501443A JP 2001502467 A JP2001502467 A JP 2001502467A JP 2001502467 A JP2001502467 A JP 2001502467A JP 2003501443 A JP2003501443 A JP 2003501443A
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- Prior art keywords
- cys
- trp
- lys
- bzl
- tyr
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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| US13765599P | 1999-06-04 | 1999-06-04 | |
| US60/137,655 | 1999-06-04 | ||
| PCT/US2000/015396 WO2000075186A1 (en) | 1999-06-04 | 2000-06-05 | Neuromedin b and somatostatin receptor agonists |
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| JP2011264477A Expired - Fee Related JP5519622B2 (ja) | 1999-06-04 | 2011-12-02 | ニューロメジンｂおよびソマトスタチンレセプターアゴニスト |
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| US20040198653A1 (en) * | 2001-06-25 | 2004-10-07 | Culler Michael De Witt | Pharmaceutical compositions which inhibit proliferation of pituitary adenomas and method of use thereof |
| AU2002359359A1 (en) | 2001-12-28 | 2003-07-24 | Somatocor Pharmaceuticals, Inc. | Imidazolidin-2,4-dione derivatives as non-peptide somatostatin receptor ligands |
| AU2003240469A1 (en) * | 2002-05-02 | 2003-11-17 | Bayer Aktiengesellschaft | Diagnostics and therapeutics for diseases associated with neuromedin b receptor (nmb) |
| CA2647986C (en) | 2006-03-31 | 2014-07-08 | Erasmus University Medical Center Rotterdam | Compositions for tumor growth control |
| NZ571862A (en) * | 2006-04-13 | 2011-10-28 | Ipsen Pharma Sas | Pharmaceutical composition comprising HGLP-1, a zinc divalent metal ion and a solvent |
| KR101642363B1 (ko) | 2008-06-12 | 2016-07-25 | 입센 바이오이노베이션 리미티드 | 신경내분비계 질환의 억제 |
| CN107446053A (zh) | 2008-06-12 | 2017-12-08 | 益普生生物创新有限公司 | 癌症的抑制 |
| GB0820970D0 (en) | 2008-11-17 | 2008-12-24 | Syntaxin Ltd | Suppression of cancer |
| US20120008318A1 (en) | 2009-04-27 | 2012-01-12 | Kabushiki Kaisha Toshiba | Lighting apparatus |
| CN108659100A (zh) * | 2017-03-28 | 2018-10-16 | 上海新生源医药集团有限公司 | 具有镇痛作用的多肽及其应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4505897A (en) * | 1983-04-18 | 1985-03-19 | The Administrators Of The Tulane Educational Fund | Cyclic pentapeptides displaying somatostatin antagonism and method of treatment of mammals therewith |
| EP0478101B1 (en) * | 1990-09-24 | 2001-08-29 | W.R. Grace & Co.-Conn. | Therapeutic use of peptides having thrombospondin-like activity |
| HU207104B (en) * | 1991-01-25 | 1993-03-01 | Biosignal Kutato Fejlesztoe Kf | Process for producing new somatostatin analogs inhibiting tumour growth and pharmaceutical compositions comprising such compounds |
| DE69225597T2 (de) * | 1991-08-09 | 1998-11-26 | Kolbeck, Winfried, 81247 Muenchen | Peptide mit einer lanthionin-brücke |
| US5462926A (en) * | 1992-07-27 | 1995-10-31 | Biomeasure, Inc. | Neuromedin B receptor antagonists which demonstrate selectivity |
| CA2144180A1 (en) * | 1992-09-08 | 1994-03-17 | George A. Heavner | Peptide inhibitors of cellular adhesion |
| RU2128055C1 (ru) * | 1992-12-07 | 1999-03-27 | Такеда Кемикал Индастриз Лтд. | Фармацевтическая композиция замедленного высвобождения и способ ее получения |
| CA2274144C (en) * | 1996-12-04 | 2004-03-30 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A. (A.S.) | Somatostatin antagonists |
| AU8019898A (en) * | 1997-05-13 | 1998-12-08 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Somatostatin and somatostatin agonists for treating insulin insensitivity and syndrome |
| EP1033372A4 (en) * | 1997-11-18 | 2000-10-04 | Chugai Pharmaceutical Co Ltd | COMPOSITIONS WITH ANTI-TUMOR ACTIVITY |
-
2000
- 2000-06-05 JP JP2001502467A patent/JP2003501443A/ja active Pending
- 2000-06-05 PL PL00352968A patent/PL352968A1/xx not_active Application Discontinuation
- 2000-06-05 AR ARP000102776A patent/AR020862A1/es not_active Application Discontinuation
- 2000-06-05 AU AU54633/00A patent/AU774096B2/en not_active Ceased
- 2000-06-05 IL IL14688400A patent/IL146884A0/xx unknown
- 2000-06-05 CZ CZ20014297A patent/CZ20014297A3/cs unknown
- 2000-06-05 BR BR0011680-7A patent/BR0011680A/pt not_active Application Discontinuation
- 2000-06-05 CN CN00811215A patent/CN1367793A/zh active Pending
- 2000-06-05 ES ES00939563T patent/ES2401096T3/es not_active Expired - Lifetime
- 2000-06-05 WO PCT/US2000/015396 patent/WO2000075186A1/en not_active Ceased
- 2000-06-05 EP EP00939563A patent/EP1189941B1/en not_active Expired - Lifetime
- 2000-06-05 CA CA2376506A patent/CA2376506C/en not_active Expired - Fee Related
- 2000-06-05 RU RU2002100069/04A patent/RU2263680C2/ru not_active IP Right Cessation
- 2000-06-05 HU HU0202022A patent/HUP0202022A3/hu unknown
- 2000-06-29 TW TW089110978A patent/TWI243177B/zh active
-
2005
- 2005-05-19 RU RU2005115448/04A patent/RU2005115448A/ru not_active Application Discontinuation
- 2005-05-19 RU RU2005115449/04A patent/RU2005115449A/ru not_active Application Discontinuation
-
2008
- 2008-11-12 JP JP2008290079A patent/JP5165537B2/ja not_active Expired - Fee Related
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2011
- 2011-12-02 JP JP2011264477A patent/JP5519622B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2009108078A (ja) | 2009-05-21 |
| RU2263680C2 (ru) | 2005-11-10 |
| AU5463300A (en) | 2000-12-28 |
| BR0011680A (pt) | 2002-04-30 |
| WO2000075186A1 (en) | 2000-12-14 |
| CZ20014297A3 (cs) | 2002-06-12 |
| JP5165537B2 (ja) | 2013-03-21 |
| AR020862A1 (es) | 2002-05-29 |
| IL146884A0 (en) | 2002-08-14 |
| ES2401096T3 (es) | 2013-04-16 |
| CA2376506A1 (en) | 2000-12-14 |
| TWI243177B (en) | 2005-11-11 |
| EP1189941B1 (en) | 2013-01-09 |
| CA2376506C (en) | 2014-07-22 |
| HUP0202022A3 (en) | 2003-10-28 |
| AU774096B2 (en) | 2004-06-17 |
| EP1189941A1 (en) | 2002-03-27 |
| RU2005115449A (ru) | 2006-11-20 |
| CN1367793A (zh) | 2002-09-04 |
| RU2005115448A (ru) | 2006-11-20 |
| JP2012102103A (ja) | 2012-05-31 |
| JP5519622B2 (ja) | 2014-06-11 |
| PL352968A1 (en) | 2003-09-22 |
| HUP0202022A2 (en) | 2002-10-28 |
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