CA2376506C - Neuromedin b and somatostatin receptor agonists - Google Patents
Neuromedin b and somatostatin receptor agonists Download PDFInfo
- Publication number
- CA2376506C CA2376506C CA2376506A CA2376506A CA2376506C CA 2376506 C CA2376506 C CA 2376506C CA 2376506 A CA2376506 A CA 2376506A CA 2376506 A CA2376506 A CA 2376506A CA 2376506 C CA2376506 C CA 2376506C
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- Prior art keywords
- cys
- trp
- lys
- tyr
- cyclo
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US13765599P | 1999-06-04 | 1999-06-04 | |
| US60/137,655 | 1999-06-04 | ||
| PCT/US2000/015396 WO2000075186A1 (en) | 1999-06-04 | 2000-06-05 | Neuromedin b and somatostatin receptor agonists |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2376506A1 CA2376506A1 (en) | 2000-12-14 |
| CA2376506C true CA2376506C (en) | 2014-07-22 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2376506A Expired - Fee Related CA2376506C (en) | 1999-06-04 | 2000-06-05 | Neuromedin b and somatostatin receptor agonists |
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|---|---|
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| JP (3) | JP2003501443A (enExample) |
| CN (1) | CN1367793A (enExample) |
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| WO (1) | WO2000075186A1 (enExample) |
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| CA2433785C (en) * | 2001-01-12 | 2009-08-04 | Michael Dewitt Culler | Pharmaceutical compositions which inhibit vascular proliferation and method of use thereof |
| CA2450446A1 (en) * | 2001-06-25 | 2003-01-03 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R | Pharmaceutical compositions which inhibit proliferation of pituitary adenomas and method of use thereof |
| US7189856B2 (en) | 2001-12-28 | 2007-03-13 | Gideon Shapiro | Non-peptide somatostatin receptor ligands |
| WO2003093830A1 (en) * | 2002-05-02 | 2003-11-13 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with neuromedin b receptor (nmb) |
| CA2647986C (en) | 2006-03-31 | 2014-07-08 | Erasmus University Medical Center Rotterdam | Compositions for tumor growth control |
| MX2008013168A (es) * | 2006-04-13 | 2008-10-27 | Sod Conseils Rech Applic | Composiciones faramaceuticas del peptido 1 similar al glucagon humano, exendina-4 y análogos de los mismos. |
| CN102083451A (zh) | 2008-06-12 | 2011-06-01 | 赛恩泰新公司 | 癌症的抑制 |
| CA2727082C (en) | 2008-06-12 | 2019-02-26 | Syntaxin Limited | Fusion proteins for use in suppression of acromegaly |
| GB0820970D0 (en) | 2008-11-17 | 2008-12-24 | Syntaxin Ltd | Suppression of cancer |
| CN102341925A (zh) | 2009-04-27 | 2012-02-01 | 东芝照明技术株式会社 | 照明装置 |
| CN108659100A (zh) * | 2017-03-28 | 2018-10-16 | 上海新生源医药集团有限公司 | 具有镇痛作用的多肽及其应用 |
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| US4505897A (en) * | 1983-04-18 | 1985-03-19 | The Administrators Of The Tulane Educational Fund | Cyclic pentapeptides displaying somatostatin antagonism and method of treatment of mammals therewith |
| EP0478101B1 (en) * | 1990-09-24 | 2001-08-29 | W.R. Grace & Co.-Conn. | Therapeutic use of peptides having thrombospondin-like activity |
| HU207104B (en) * | 1991-01-25 | 1993-03-01 | Biosignal Kutato Fejlesztoe Kf | Process for producing new somatostatin analogs inhibiting tumour growth and pharmaceutical compositions comprising such compounds |
| WO1993003056A1 (en) * | 1991-08-09 | 1993-02-18 | Winfried Kolbeck | Lanthionine bridged peptides |
| US5462926A (en) * | 1992-07-27 | 1995-10-31 | Biomeasure, Inc. | Neuromedin B receptor antagonists which demonstrate selectivity |
| WO1994005310A1 (en) * | 1992-09-08 | 1994-03-17 | Centocor, Inc. | Peptide inhibitors of cellular adhesion |
| RU2128055C1 (ru) * | 1992-12-07 | 1999-03-27 | Такеда Кемикал Индастриз Лтд. | Фармацевтическая композиция замедленного высвобождения и способ ее получения |
| ATE330966T1 (de) * | 1996-12-04 | 2006-07-15 | Sod Conseils Rech Applic | Somatostatin-antagonisten |
| CA2289499C (en) * | 1997-05-13 | 2010-02-23 | Michael Anthony Cawthorne | Somatostatin and somatostatin agonists for treating insulin insensitivity and syndrome x |
| WO1999025729A1 (fr) * | 1997-11-18 | 1999-05-27 | Chugai Seiyaku Kabushiki Kaisha | Composes possedant une activite antitumorale |
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2000
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- 2000-06-05 HU HU0202022A patent/HUP0202022A3/hu unknown
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2005
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2008
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2011
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Also Published As
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|---|---|
| HUP0202022A2 (en) | 2002-10-28 |
| JP5519622B2 (ja) | 2014-06-11 |
| TWI243177B (en) | 2005-11-11 |
| CA2376506A1 (en) | 2000-12-14 |
| CN1367793A (zh) | 2002-09-04 |
| BR0011680A (pt) | 2002-04-30 |
| ES2401096T3 (es) | 2013-04-16 |
| JP2009108078A (ja) | 2009-05-21 |
| AU5463300A (en) | 2000-12-28 |
| PL352968A1 (en) | 2003-09-22 |
| RU2005115449A (ru) | 2006-11-20 |
| IL146884A0 (en) | 2002-08-14 |
| EP1189941A1 (en) | 2002-03-27 |
| CZ20014297A3 (cs) | 2002-06-12 |
| RU2263680C2 (ru) | 2005-11-10 |
| JP2003501443A (ja) | 2003-01-14 |
| HUP0202022A3 (en) | 2003-10-28 |
| EP1189941B1 (en) | 2013-01-09 |
| WO2000075186A1 (en) | 2000-12-14 |
| JP2012102103A (ja) | 2012-05-31 |
| AU774096B2 (en) | 2004-06-17 |
| RU2005115448A (ru) | 2006-11-20 |
| AR020862A1 (es) | 2002-05-29 |
| JP5165537B2 (ja) | 2013-03-21 |
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