JP2003012683A5 - - Google Patents
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- Publication number
- JP2003012683A5 JP2003012683A5 JP2001201316A JP2001201316A JP2003012683A5 JP 2003012683 A5 JP2003012683 A5 JP 2003012683A5 JP 2001201316 A JP2001201316 A JP 2001201316A JP 2001201316 A JP2001201316 A JP 2001201316A JP 2003012683 A5 JP2003012683 A5 JP 2003012683A5
- Authority
- JP
- Japan
- Prior art keywords
- acetyl
- sugar
- metal fluoride
- oxazoline derivative
- tri
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000003504 2-oxazolinyl group Chemical class O1C(=NCC1)* 0.000 description 4
- 238000004519 manufacturing process Methods 0.000 description 3
- -1 N-acetyl chloride-3,4,6-tri-O-acetyl-α-glucosaminyl chloride Chemical compound 0.000 description 2
- 229910001512 metal fluoride Inorganic materials 0.000 description 2
- 150000001271 acylaminosugars Chemical class 0.000 description 1
- 229910001515 alkali metal fluoride Inorganic materials 0.000 description 1
- 238000000034 method Methods 0.000 description 1
- 125000006239 protecting group Chemical group 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
Priority Applications (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001201316A JP4866515B2 (ja) | 2001-07-02 | 2001-07-02 | 糖オキサゾリン誘導体の製造方法 |
| PCT/JP2002/006575 WO2003004508A1 (en) | 2001-07-02 | 2002-06-28 | Process for production of saccharide oxazoline derivatives |
| US10/482,678 US20040176588A1 (en) | 2001-07-02 | 2002-06-28 | Process for production of sugar oxazoline derivatives |
| EP02738865.1A EP1405857B1 (en) | 2001-07-02 | 2002-06-28 | Process for the production of 2-methyl-(3,4,6-tri-O-acetyl-1,2-dideoxy-alpha-glucopyrano)-[2,1-d]-2-oxazoline |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001201316A JP4866515B2 (ja) | 2001-07-02 | 2001-07-02 | 糖オキサゾリン誘導体の製造方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2003012683A JP2003012683A (ja) | 2003-01-15 |
| JP2003012683A5 true JP2003012683A5 (enExample) | 2010-10-07 |
| JP4866515B2 JP4866515B2 (ja) | 2012-02-01 |
Family
ID=19038309
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001201316A Expired - Fee Related JP4866515B2 (ja) | 2001-07-02 | 2001-07-02 | 糖オキサゾリン誘導体の製造方法 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20040176588A1 (enExample) |
| EP (1) | EP1405857B1 (enExample) |
| JP (1) | JP4866515B2 (enExample) |
| WO (1) | WO2003004508A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5380293B2 (ja) * | 2006-08-31 | 2014-01-08 | サイモン・フレーザー・ユニバーシティ | 選択的グリコシダーゼ阻害剤およびその使用 |
| JP5301427B2 (ja) * | 2007-03-09 | 2013-09-25 | 生化学工業株式会社 | 糖オキサゾリン誘導体の製造方法 |
| US9120781B2 (en) | 2010-05-11 | 2015-09-01 | Simon Fraser University | Selective glycosidase inhibitors and uses thereof |
| RU2609210C2 (ru) | 2010-12-23 | 2017-01-31 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| WO2012129651A1 (en) | 2011-03-31 | 2012-10-04 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| RU2625308C2 (ru) | 2011-06-27 | 2017-07-13 | Алектос Терапьютикс Инк. | Селективные ингибиторы гликозидазы и их применение |
| EP2726468B1 (en) | 2011-06-27 | 2017-04-12 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| US9701693B2 (en) | 2011-06-27 | 2017-07-11 | Alectos Therapeutics Inc. | Selective glycosidase inhibitors and uses thereof |
| EP2890675A4 (en) | 2012-08-31 | 2016-01-13 | Alectos Therapeutics Inc | GLYCOSIDASE INHIBITORS AND USES THEREOF |
| EP2890676B1 (en) | 2012-08-31 | 2018-12-05 | Alectos Therapeutics Inc. | Glycosidase inhibitors and uses thereof |
| KR20150079711A (ko) | 2012-10-31 | 2015-07-08 | 알렉토스 테라퓨틱스 인크. | 글리코시다아제 저해제 및 이의 용도 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5382665A (en) * | 1993-03-17 | 1995-01-17 | The United States Of America As Represented By The United States Department Of Energy | Synthesis of oxazolines and oxazines |
| JP3713065B2 (ja) * | 1995-03-10 | 2005-11-02 | 信越化学工業株式会社 | 二糖モノマー及びそのオリゴマーとオリゴマーの製造方法 |
| JPH093088A (ja) | 1995-06-19 | 1997-01-07 | Shin Etsu Chem Co Ltd | アミノ二糖及びキチン又はその類似多糖類の製造方法 |
-
2001
- 2001-07-02 JP JP2001201316A patent/JP4866515B2/ja not_active Expired - Fee Related
-
2002
- 2002-06-28 WO PCT/JP2002/006575 patent/WO2003004508A1/ja not_active Ceased
- 2002-06-28 US US10/482,678 patent/US20040176588A1/en not_active Abandoned
- 2002-06-28 EP EP02738865.1A patent/EP1405857B1/en not_active Expired - Lifetime