JP2002538106A - イソバレルアミド、イソ吉草酸、または関連化合物を用いてｃｎｓ活性の調節に影響を与えることによる、痙縮および痙攣を含む様々な病状の治療 - Google Patents
イソバレルアミド、イソ吉草酸、または関連化合物を用いてｃｎｓ活性の調節に影響を与えることによる、痙縮および痙攣を含む様々な病状の治療Info
- Publication number
- JP2002538106A JP2002538106A JP2000602054A JP2000602054A JP2002538106A JP 2002538106 A JP2002538106 A JP 2002538106A JP 2000602054 A JP2000602054 A JP 2000602054A JP 2000602054 A JP2000602054 A JP 2000602054A JP 2002538106 A JP2002538106 A JP 2002538106A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- isovaleramide
- condition
- isovaleric acid
- dimethylisovaleramide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
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- Physical Education & Sports Medicine (AREA)
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- Orthopedic Medicine & Surgery (AREA)
- Addiction (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/258,882 | 1999-03-01 | ||
| US09/258,882 US6589994B1 (en) | 1996-08-30 | 1999-03-01 | Treating a variety of pathological conditions, including spasticity and convulsions, by effecting a modulation of CNS activity with isovaleramide, isovaleric acid, or a related compound |
| PCT/US2000/005324 WO2000051586A2 (en) | 1999-03-01 | 2000-03-01 | Treating a variety of pathological conditions, including spasticity and convulsions, by effecting modulation of cns activity with isovaleramide, isovaleric acid, or a related compound |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002538106A true JP2002538106A (ja) | 2002-11-12 |
| JP2002538106A5 JP2002538106A5 (https=) | 2007-04-26 |
Family
ID=22982536
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000602054A Pending JP2002538106A (ja) | 1999-03-01 | 2000-03-01 | イソバレルアミド、イソ吉草酸、または関連化合物を用いてｃｎｓ活性の調節に影響を与えることによる、痙縮および痙攣を含む様々な病状の治療 |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US6589994B1 (https=) |
| EP (1) | EP1176953A2 (https=) |
| JP (1) | JP2002538106A (https=) |
| AU (1) | AU779418B2 (https=) |
| CA (1) | CA2366038A1 (https=) |
| WO (1) | WO2000051586A2 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007530493A (ja) * | 2004-03-26 | 2007-11-01 | シュバルツ ファルマ アクチェンゲゼルシャフト | 痛みのある糖尿病性神経障害における疼痛を治療するためのペプチド化合物の新規使用 |
| KR20180054381A (ko) * | 2016-11-15 | 2018-05-24 | 경희대학교 산학협력단 | 쥐오줌풀 추출물을 유효성분으로 포함하는 측두엽 뇌전증 예방 또는 치료용 약학적 조성물 |
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| US20040115290A1 (en) * | 2001-06-20 | 2004-06-17 | Tripp Matthew L. | Modulation of inflammation by hops fractions and derivatives |
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| RU2010142655A (ru) | 2008-03-19 | 2012-04-27 | Ауриммед Фарма, Инк. (Us) | Соединение, пригодное для лечения болезней и нарушений центральной нервной системы, и способ его получения |
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| US9212155B2 (en) | 2008-03-19 | 2015-12-15 | Aurimmed Pharma, Inc. | Compounds advantageous in the treatment of central nervous system diseases and disorders |
| EP2268600A4 (en) * | 2008-04-02 | 2012-03-21 | Metaproteomics Llc | SUBSTITUTED 1,3-CYCLOPENTADION-ENHANCED ENDOTHELIAL IGNITION AND ENDOTHELIAL MONOCYTE INTERACTIONS |
| US9808434B2 (en) | 2011-01-27 | 2017-11-07 | City Of Hope | Compound for treating cancer and diabetes |
| WO2012103523A2 (en) | 2011-01-27 | 2012-08-02 | Samuel Rahbar | Novel modulators of development of adipocyte and cancer cells |
| EP2675297A4 (en) * | 2011-02-16 | 2014-10-01 | Wellbemed Sweden Ab | FOOD WITH AN EXTRACT MIXTURE |
| WO2017150903A1 (en) | 2016-02-29 | 2017-09-08 | Bio-Pharm Solutions Co., Ltd. | Sulfamate derivative compounds, processes for preparing them and their uses |
| US11670410B1 (en) * | 2022-04-13 | 2023-06-06 | Green Sky Creations LLC | Systems and methods to automatically administer a psychoactive substance to an airway of a user based on a detected event or condition |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JPH09501908A (ja) * | 1993-06-11 | 1997-02-25 | エヌピーエス ファーマシューティカルズ，インク． | 穏和不安緩解薬および穏和鎮静薬としてのイソバレラマイドの使用 |
| WO1998008498A1 (en) * | 1996-08-30 | 1998-03-05 | Nps Pharmaceuticals, Inc. | Treatment of spasticity, convulsions by isovaleric acid derivatives cns depressants |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1617555C3 (de) | 1966-04-19 | 1974-09-19 | Kali-Chemie Ag, 3000 Hannover | Verfahren zur Isolierung von therapeutisch wertvollen Isovaleriansäureestern aus Valeriana- und Kentranthus-Extrakten |
| US6107499A (en) * | 1988-02-26 | 2000-08-22 | Neuromedica, Inc. | Dopamine analog amide |
| US4939174A (en) * | 1988-02-26 | 1990-07-03 | Shashoua Victor E | Appetite suppression with dopamine-fatty acid conjugates |
| US4933324A (en) * | 1988-02-26 | 1990-06-12 | Shashoua Victor E | Fatty acid-neuroactive drug conjugate as a prodrug |
| US5994392A (en) * | 1988-02-26 | 1999-11-30 | Neuromedica, Inc. | Antipsychotic prodrugs comprising an antipsychotic agent coupled to an unsaturated fatty acid |
| IT1283951B1 (it) | 1996-03-15 | 1998-05-07 | Mendes Srl | Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi di |
| US6589994B1 (en) * | 1996-08-30 | 2003-07-08 | Nps Pharmaceuticals, Inc. | Treating a variety of pathological conditions, including spasticity and convulsions, by effecting a modulation of CNS activity with isovaleramide, isovaleric acid, or a related compound |
| AU2894599A (en) | 1998-03-04 | 1999-09-20 | Nps Pharmaceuticals, Inc. | Compositions comprising valerian extracts, isovaleric acid or derivatives thereof with a nsaid |
| AU780505B2 (en) | 1999-10-19 | 2005-03-24 | Nps Pharmaceuticals, Inc. | Sustained-release formulations for treating CNS-mediated disorders |
-
1999
- 1999-03-01 US US09/258,882 patent/US6589994B1/en not_active Expired - Fee Related
-
2000
- 2000-03-01 JP JP2000602054A patent/JP2002538106A/ja active Pending
- 2000-03-01 CA CA002366038A patent/CA2366038A1/en not_active Abandoned
- 2000-03-01 AU AU32483/00A patent/AU779418B2/en not_active Ceased
- 2000-03-01 WO PCT/US2000/005324 patent/WO2000051586A2/en not_active Ceased
- 2000-03-01 EP EP00910383A patent/EP1176953A2/en not_active Withdrawn
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2003
- 2003-07-08 US US10/614,344 patent/US7265155B2/en not_active Expired - Fee Related
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH09501908A (ja) * | 1993-06-11 | 1997-02-25 | エヌピーエス ファーマシューティカルズ，インク． | 穏和不安緩解薬および穏和鎮静薬としてのイソバレラマイドの使用 |
| WO1998008498A1 (en) * | 1996-08-30 | 1998-03-05 | Nps Pharmaceuticals, Inc. | Treatment of spasticity, convulsions by isovaleric acid derivatives cns depressants |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007530493A (ja) * | 2004-03-26 | 2007-11-01 | シュバルツ ファルマ アクチェンゲゼルシャフト | 痛みのある糖尿病性神経障害における疼痛を治療するためのペプチド化合物の新規使用 |
| KR20180054381A (ko) * | 2016-11-15 | 2018-05-24 | 경희대학교 산학협력단 | 쥐오줌풀 추출물을 유효성분으로 포함하는 측두엽 뇌전증 예방 또는 치료용 약학적 조성물 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2000051586A3 (en) | 2001-11-29 |
| AU3248300A (en) | 2000-09-21 |
| EP1176953A2 (en) | 2002-02-06 |
| US20040072900A1 (en) | 2004-04-15 |
| US7265155B2 (en) | 2007-09-04 |
| AU779418B2 (en) | 2005-01-20 |
| CA2366038A1 (en) | 2000-09-08 |
| WO2000051586A2 (en) | 2000-09-08 |
| US6589994B1 (en) | 2003-07-08 |
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