JP2002523446A - 過活動性膀胱の治療のための抗ムスカリン剤としての経皮投与トルテロジン - Google Patents
過活動性膀胱の治療のための抗ムスカリン剤としての経皮投与トルテロジンInfo
- Publication number
- JP2002523446A JP2002523446A JP2000567189A JP2000567189A JP2002523446A JP 2002523446 A JP2002523446 A JP 2002523446A JP 2000567189 A JP2000567189 A JP 2000567189A JP 2000567189 A JP2000567189 A JP 2000567189A JP 2002523446 A JP2002523446 A JP 2002523446A
- Authority
- JP
- Japan
- Prior art keywords
- tolterodine
- transdermal
- type
- transdermal administration
- patch
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A—HUMAN NECESSITIES
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- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A61K9/7061—Polyacrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7069—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9802864-0 | 1998-08-27 | ||
| SE9802864A SE9802864D0 (sv) | 1998-08-27 | 1998-08-27 | Transdermally administered tolterodine as antimuscarinic agent for the treatment of overactive bladder |
| PCT/SE1999/001464 WO2000012070A1 (en) | 1998-08-27 | 1999-08-26 | Transdermally administered tolterodine as anti-muscarinic agent for the treatment of overactive bladder |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002523446A true JP2002523446A (ja) | 2002-07-30 |
| JP2002523446A5 JP2002523446A5 (https=) | 2006-05-25 |
Family
ID=20412370
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000567189A Pending JP2002523446A (ja) | 1998-08-27 | 1999-08-26 | 過活動性膀胱の治療のための抗ムスカリン剤としての経皮投与トルテロジン |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US6517864B1 (https=) |
| EP (1) | EP1105111B1 (https=) |
| JP (1) | JP2002523446A (https=) |
| AT (1) | ATE405254T1 (https=) |
| AU (1) | AU758399B2 (https=) |
| CA (1) | CA2341063C (https=) |
| DE (1) | DE69939382D1 (https=) |
| ES (2) | ES2353765T3 (https=) |
| NZ (1) | NZ509928A (https=) |
| SE (1) | SE9802864D0 (https=) |
| TW (1) | TWI253349B (https=) |
| WO (1) | WO2000012070A1 (https=) |
| ZA (1) | ZA200002488B (https=) |
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPWO2005011683A1 (ja) * | 2003-08-04 | 2007-10-04 | 杏林製薬株式会社 | 経皮吸収型製剤 |
| JP2011512405A (ja) * | 2008-02-20 | 2011-04-21 | エスケー ケミカルズ カンパニー リミテッド | 経皮ドラッグデリバリーシステムとして効果的な安定性を有するトルテロジン酸付加塩 |
| WO2012017892A1 (ja) | 2010-08-03 | 2012-02-09 | 久光製薬株式会社 | 貼付剤及びその粘着力増強方法 |
| JP2012532096A (ja) * | 2009-06-29 | 2012-12-13 | エスケー ケミカルズ カンパニー リミテッド | 保管安定性が向上したトルテロジンを含有する経皮投与組成物 |
| WO2013099835A1 (ja) | 2011-12-27 | 2013-07-04 | 帝國製薬株式会社 | トルテロジン含有貼付剤 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998003067A1 (en) * | 1996-07-19 | 1998-01-29 | Gunnar Aberg | S(-)-tolterodine in the treatment of urinary and gastrointestinal disorders |
| EP0957073A1 (en) * | 1998-05-12 | 1999-11-17 | Schwarz Pharma Ag | Novel derivatives of 3,3-diphenylpropylamines |
| SE9802864D0 (sv) * | 1998-08-27 | 1998-08-27 | Pharmacia & Upjohn Ab | Transdermally administered tolterodine as antimuscarinic agent for the treatment of overactive bladder |
| PT1031346E (pt) | 1999-01-27 | 2002-09-30 | Idea Ag | Vacinacao nao invasiva atraves da pele |
| SI1031347T1 (en) | 1999-01-27 | 2002-10-31 | Idea Ag | Transnasal transport/immunisation with highly adaptable carriers |
| DE19922662C1 (de) | 1999-05-18 | 2000-12-28 | Sanol Arznei Schwarz Gmbh | Transdermales therapeutisches System (TTS) Tolterodin enthaltend |
| WO2001001962A1 (en) * | 1999-07-05 | 2001-01-11 | Idea Ag. | A method for the improvement of transport across adaptable semi-permeable barriers |
| DE19932651A1 (de) * | 1999-07-13 | 2001-01-18 | Hexal Ag | Transdermales therapeutisches System zur Anwendung von Tolterodin |
| JP2005513080A (ja) * | 2001-12-20 | 2005-05-12 | フェムファーマ， インコーポレイテッド | 薬物の膣送達 |
| JP2006515026A (ja) * | 2003-01-02 | 2006-05-18 | フェムファーマ ホールディング カンパニー， インコーポレイテッド | 乳房の疾患および障害の処置のための薬学的調製物 |
| US9173836B2 (en) | 2003-01-02 | 2015-11-03 | FemmeParma Holding Company, Inc. | Pharmaceutical preparations for treatments of diseases and disorders of the breast |
| US20040191345A1 (en) * | 2003-03-26 | 2004-09-30 | Fredrik Nicklasson | New formulations and use thereof |
| DE10315917A1 (de) * | 2003-04-08 | 2004-11-18 | Schwarz Pharma Ag | Hochreine Basen von 3,3-Diphenylpropylaminmonoestern |
| WO2006015299A2 (en) * | 2004-07-30 | 2006-02-09 | Microchips, Inc. | Multi-reservoir device for transdermal drug delivery and sensing |
| WO2006082888A1 (ja) * | 2005-02-03 | 2006-08-10 | Kyorin Pharmaceutical Co., Ltd. | 経皮吸収型製剤 |
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| WO1998003067A1 (en) * | 1996-07-19 | 1998-01-29 | Gunnar Aberg | S(-)-tolterodine in the treatment of urinary and gastrointestinal disorders |
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| US5382600A (en) | 1988-01-22 | 1995-01-17 | Pharmacia Aktiebolag | 3,3-diphenylpropylamines and pharmaceutical compositions thereof |
| ZA933349B (en) * | 1992-05-13 | 1994-06-15 | Alza Corp | Transdermal administration of oxybutynin |
| PT877600E (pt) * | 1996-08-09 | 2004-02-27 | Alcon Mfg Ltd | Sistemas conservantes para composicoes farmaceuticas contendo ciclodextrinas |
| SE9802864D0 (sv) * | 1998-08-27 | 1998-08-27 | Pharmacia & Upjohn Ab | Transdermally administered tolterodine as antimuscarinic agent for the treatment of overactive bladder |
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- 1998-08-27 SE SE9802864A patent/SE9802864D0/xx unknown
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- 1999-08-26 AT AT99946522T patent/ATE405254T1/de not_active IP Right Cessation
- 1999-08-26 NZ NZ509928A patent/NZ509928A/en unknown
- 1999-08-26 US US09/763,654 patent/US6517864B1/en not_active Expired - Fee Related
- 1999-08-26 DE DE69939382T patent/DE69939382D1/de not_active Expired - Lifetime
- 1999-08-26 CA CA002341063A patent/CA2341063C/en not_active Expired - Fee Related
- 1999-08-26 AU AU58919/99A patent/AU758399B2/en not_active Ceased
- 1999-08-26 ES ES99946521T patent/ES2353765T3/es not_active Expired - Lifetime
- 1999-08-26 EP EP99946522A patent/EP1105111B1/en not_active Expired - Lifetime
- 1999-08-26 WO PCT/SE1999/001464 patent/WO2000012070A1/en not_active Ceased
- 1999-08-26 ES ES99946522T patent/ES2310942T3/es not_active Expired - Lifetime
- 1999-08-26 JP JP2000567189A patent/JP2002523446A/ja active Pending
- 1999-08-27 TW TW088114752A patent/TWI253349B/zh not_active IP Right Cessation
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2000
- 2000-05-19 ZA ZA200002488A patent/ZA200002488B/xx unknown
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| WO1998003067A1 (en) * | 1996-07-19 | 1998-01-29 | Gunnar Aberg | S(-)-tolterodine in the treatment of urinary and gastrointestinal disorders |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPWO2005011683A1 (ja) * | 2003-08-04 | 2007-10-04 | 杏林製薬株式会社 | 経皮吸収型製剤 |
| JP2011512405A (ja) * | 2008-02-20 | 2011-04-21 | エスケー ケミカルズ カンパニー リミテッド | 経皮ドラッグデリバリーシステムとして効果的な安定性を有するトルテロジン酸付加塩 |
| JP2012532096A (ja) * | 2009-06-29 | 2012-12-13 | エスケー ケミカルズ カンパニー リミテッド | 保管安定性が向上したトルテロジンを含有する経皮投与組成物 |
| WO2012017892A1 (ja) | 2010-08-03 | 2012-02-09 | 久光製薬株式会社 | 貼付剤及びその粘着力増強方法 |
| WO2013099835A1 (ja) | 2011-12-27 | 2013-07-04 | 帝國製薬株式会社 | トルテロジン含有貼付剤 |
| JPWO2013099835A1 (ja) * | 2011-12-27 | 2015-05-07 | 帝國製薬株式会社 | トルテロジン含有貼付剤 |
| US10195162B2 (en) | 2011-12-27 | 2019-02-05 | Teikoku Seiyaku Co., Ltd. | Tolterodine-containing adhesive patch |
Also Published As
| Publication number | Publication date |
|---|---|
| US20030124179A1 (en) | 2003-07-03 |
| US7008637B2 (en) | 2006-03-07 |
| CA2341063C (en) | 2008-02-12 |
| AU5891999A (en) | 2000-03-21 |
| ZA200002488B (en) | 2001-05-16 |
| ATE405254T1 (de) | 2008-09-15 |
| AU758399B2 (en) | 2003-03-20 |
| CA2341063A1 (en) | 2000-03-09 |
| US6517864B1 (en) | 2003-02-11 |
| WO2000012070A1 (en) | 2000-03-09 |
| EP1105111B1 (en) | 2008-08-20 |
| TWI253349B (en) | 2006-04-21 |
| DE69939382D1 (de) | 2008-10-02 |
| EP1105111A1 (en) | 2001-06-13 |
| SE9802864D0 (sv) | 1998-08-27 |
| NZ509928A (en) | 2003-08-29 |
| ES2353765T3 (es) | 2011-03-04 |
| ES2310942T3 (es) | 2009-01-16 |
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