JP2002503674A5 - - Google Patents
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- Publication number
- JP2002503674A5 JP2002503674A5 JP2000531467A JP2000531467A JP2002503674A5 JP 2002503674 A5 JP2002503674 A5 JP 2002503674A5 JP 2000531467 A JP2000531467 A JP 2000531467A JP 2000531467 A JP2000531467 A JP 2000531467A JP 2002503674 A5 JP2002503674 A5 JP 2002503674A5
- Authority
- JP
- Japan
- Prior art keywords
- chemical
- compound according
- nrr
- ring
- nhr
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US1998/002891 WO1999041276A1 (en) | 1998-02-12 | 1998-02-12 | β-SHEET MIMETICS AND METHODS RELATING TO THE USE THEREOF |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002503674A JP2002503674A (ja) | 2002-02-05 |
| JP2002503674A5 true JP2002503674A5 (enExample) | 2005-12-22 |
Family
ID=22266392
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000531467A Pending JP2002503674A (ja) | 1998-02-12 | 1998-02-12 | βシート模倣物およびその使用に関する方法 |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1053246B1 (enExample) |
| JP (1) | JP2002503674A (enExample) |
| KR (1) | KR20010040939A (enExample) |
| AT (1) | ATE230414T1 (enExample) |
| AU (1) | AU748887B2 (enExample) |
| CA (1) | CA2319766A1 (enExample) |
| DE (1) | DE69810513T2 (enExample) |
| ES (1) | ES2192764T3 (enExample) |
| WO (1) | WO1999041276A1 (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001064678A2 (en) * | 2000-02-29 | 2001-09-07 | Bristol-Myers Squibb Pharma Company | Inhibitors of hepatitis c virus ns3 protease |
| US6534651B2 (en) * | 2000-04-06 | 2003-03-18 | Inotek Pharmaceuticals Corp. | 7-Substituted isoindolinone inhibitors of inflammation and reperfusion injury and methods of use thereof |
| US7122679B2 (en) | 2000-05-09 | 2006-10-17 | Cephalon, Inc. | Multicyclic compounds and the use thereof |
| US20060276497A1 (en) | 2000-05-09 | 2006-12-07 | Cephalon, Inc. | Novel multicyclic compounds and the use thereof |
| CN1642550A (zh) * | 2002-02-14 | 2005-07-20 | 美瑞德生物工程公司 | β-折叠模拟物和组合物及其有关方法 |
| WO2009158369A1 (en) | 2008-06-25 | 2009-12-30 | Schering Corporation | Synthesis and use of heterocyclic antibacterial agents |
| WO2016057413A2 (en) | 2014-10-06 | 2016-04-14 | Cortexyme, Inc. | Inhibitors of lysine gingipain |
| CA3004095A1 (en) | 2015-11-09 | 2017-05-18 | Cortexyme, Inc. | Inhibitors of arginine gingipain |
| AU2017317988B2 (en) | 2016-08-31 | 2020-12-24 | Jiangsu Hengrui Medicine Co., Ltd. | Oxopicolinamide derivative, preparation method therefor and pharmaceutical use thereof |
| EP4480541A3 (en) | 2016-09-16 | 2025-04-30 | Lighthouse Pharmaceuticals, Inc. | Ketone inhibitors of lysine gingipain |
| JP2021529201A (ja) | 2018-07-02 | 2021-10-28 | 江▲蘇▼恒瑞医▲薬▼股▲フン▼有限公司Jiangsu Hengrui Medicine Co., Ltd. | オキシピリジンアミド誘導体の結晶形およびその調製方法 |
| JP7450024B2 (ja) | 2019-09-27 | 2024-03-14 | シェンヅェン サルブリス ファーマシューティカルズ カンパニー リミテッド | FXIa阻害剤及びその調製方法と医薬用途 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU220596B1 (hu) * | 1992-02-14 | 2002-03-28 | Merrell Dow Pharmaceuticals Inc. | 7-Szubsztituált pirido-benzazepin-karbonsav-származékok, ezeket tartalmazó gyógyszerkészítmények és eljárás előállításukra |
| HU223663B1 (hu) * | 1992-05-15 | 2004-11-29 | Merrel Dow Pharmaceuticals Inc. | Enkefalináz és ACE gátló hatású 9-[(2-acetil-tio-3-fenil)-propanoil-amino]-piridazo[1,2-a][1,2]diazepin-származékok, eljárás előállításukra, alkalmazásuk és az ezeket tartalmazó gyógyszerkészítmények |
| EP0618223A3 (en) * | 1993-03-08 | 1996-06-12 | Sandoz Ltd | Peptides, the release of Interleukin 1-Bêta, useful as anti-inflammatory agents. |
| WO1996019483A1 (en) * | 1994-12-22 | 1996-06-27 | Biochem Pharma Inc. | Low molecular weight bicyclic thrombin inhibitors |
| WO1996030396A1 (en) * | 1995-03-24 | 1996-10-03 | Molecumetics Ltd. | β-SHEET MIMETICS AND USE THEREOF AS PROTEASE INHIBITORS |
| AU713530B2 (en) * | 1995-03-24 | 1999-12-02 | Molecumetics, Ltd. | Beta-sheet mimetics and use thereof as protease inhibitors |
| US5877313A (en) * | 1995-05-17 | 1999-03-02 | Bristol-Myers Squibb | Benzo-fused azepinone and piperidinone compounds useful in the inhibition of ACE and NEP |
| IT1277405B1 (it) * | 1995-08-01 | 1997-11-10 | Menarini Farma Ind | Derivati di lattami biciclici come inibitori della trombina |
| ES2262184T3 (es) * | 1996-08-05 | 2006-11-16 | Myriad Genetics, Inc. | Utilizacion de mimeticos de hojas beta como inhibidores de proteasa y de kinasa o como inhibidores de factores de transcripcion. |
-
1998
- 1998-02-12 WO PCT/US1998/002891 patent/WO1999041276A1/en not_active Ceased
- 1998-02-12 AU AU66557/98A patent/AU748887B2/en not_active Ceased
- 1998-02-12 EP EP98908551A patent/EP1053246B1/en not_active Expired - Lifetime
- 1998-02-12 KR KR1020007008856A patent/KR20010040939A/ko not_active Ceased
- 1998-02-12 CA CA002319766A patent/CA2319766A1/en not_active Abandoned
- 1998-02-12 AT AT98908551T patent/ATE230414T1/de not_active IP Right Cessation
- 1998-02-12 DE DE69810513T patent/DE69810513T2/de not_active Expired - Lifetime
- 1998-02-12 JP JP2000531467A patent/JP2002503674A/ja active Pending
- 1998-02-12 ES ES98908551T patent/ES2192764T3/es not_active Expired - Lifetime
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