JP2002012595A5 - - Google Patents
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- Publication number
- JP2002012595A5 JP2002012595A5 JP2001130982A JP2001130982A JP2002012595A5 JP 2002012595 A5 JP2002012595 A5 JP 2002012595A5 JP 2001130982 A JP2001130982 A JP 2001130982A JP 2001130982 A JP2001130982 A JP 2001130982A JP 2002012595 A5 JP2002012595 A5 JP 2002012595A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- atom
- substituted
- nitrogen atom
- pharmaceutically
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
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- 229910052757 nitrogen Inorganic materials 0.000 description 47
- 125000004433 nitrogen atom Chemical group N* 0.000 description 47
- -1 methoxyacetyl group Chemical group 0.000 description 35
- 125000004432 carbon atom Chemical group C* 0.000 description 34
- 150000003839 salts Chemical class 0.000 description 29
- 125000004435 hydrogen atom Chemical group [H]* 0.000 description 28
- 125000001424 substituent group Chemical group 0.000 description 24
- 125000005843 halogen group Chemical group 0.000 description 22
- FXWHFKOXMBTCMP-WMEDONTMSA-N milbemycin Natural products COC1C2OCC3=C/C=C/C(C)CC(=CCC4CC(CC5(O4)OC(C)C(C)C(OC(=O)C(C)CC(C)C)C5O)OC(=O)C(C=C1C)C23O)C FXWHFKOXMBTCMP-WMEDONTMSA-N 0.000 description 22
- 125000003277 amino group Chemical group 0.000 description 19
- 150000001875 compounds Chemical class 0.000 description 19
- 125000004430 oxygen atom Chemical group O* 0.000 description 17
- 125000004429 atom Chemical group 0.000 description 16
- 229910052799 carbon Inorganic materials 0.000 description 16
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 description 16
- 229910052717 sulfur Inorganic materials 0.000 description 16
- 125000004434 sulfur atom Chemical group 0.000 description 16
- 125000004043 oxo group Chemical group O=* 0.000 description 15
- 125000003545 alkoxy group Chemical group 0.000 description 14
- 125000004453 alkoxycarbonyl group Chemical group 0.000 description 13
- 125000001511 cyclopentyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 description 13
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 description 13
- 125000000623 heterocyclic group Chemical group 0.000 description 13
- 125000004093 cyano group Chemical group *C#N 0.000 description 12
- 125000002887 hydroxy group Chemical group [H]O* 0.000 description 12
- 125000002861 (C1-C4) alkanoyl group Chemical group 0.000 description 10
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 description 8
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 description 8
- 238000000034 method Methods 0.000 description 8
- 125000004122 cyclic group Chemical group 0.000 description 7
- 125000004455 (C1-C3) alkylthio group Chemical group 0.000 description 6
- 241000490513 Ctenocephalides canis Species 0.000 description 6
- 241000258924 Ctenocephalides felis Species 0.000 description 6
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 description 6
- 125000004390 alkyl sulfonyl group Chemical group 0.000 description 6
- 125000001995 cyclobutyl group Chemical group [H]C1([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 description 6
- 241000238631 Hexapoda Species 0.000 description 5
- 125000000217 alkyl group Chemical group 0.000 description 5
- 244000000053 intestinal parasite Species 0.000 description 5
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 description 4
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 description 4
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 description 4
- 241000238876 Acari Species 0.000 description 4
- 241000124008 Mammalia Species 0.000 description 4
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 description 4
- 239000000203 mixture Substances 0.000 description 4
- 244000045947 parasite Species 0.000 description 4
- 125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 description 4
- 241001465754 Metazoa Species 0.000 description 3
- 125000002252 acyl group Chemical group 0.000 description 3
- 125000000350 glycoloyl group Chemical group O=C([*])C([H])([H])O[H] 0.000 description 3
- 238000003898 horticulture Methods 0.000 description 3
- 230000003071 parasitic effect Effects 0.000 description 3
- 125000004044 trifluoroacetyl group Chemical group FC(C(=O)*)(F)F 0.000 description 3
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 description 2
- 125000004423 acyloxy group Chemical group 0.000 description 2
- 125000004414 alkyl thio group Chemical group 0.000 description 2
- 230000000507 anthelmentic effect Effects 0.000 description 2
- 125000000753 cycloalkyl group Chemical group 0.000 description 2
- 230000000749 insecticidal effect Effects 0.000 description 2
- 239000000126 substance Substances 0.000 description 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 description 1
- 239000013543 active substance Substances 0.000 description 1
- UKJLNMAFNRKWGR-UHFFFAOYSA-N cyclohexatrienamine Chemical group NC1=CC=C=C[CH]1 UKJLNMAFNRKWGR-UHFFFAOYSA-N 0.000 description 1
- 229940079593 drug Drugs 0.000 description 1
- 239000003814 drug Substances 0.000 description 1
- 229910052736 halogen Inorganic materials 0.000 description 1
- 125000005842 heteroatom Chemical group 0.000 description 1
- 239000002917 insecticide Substances 0.000 description 1
- 230000000361 pesticidal effect Effects 0.000 description 1
- 239000008177 pharmaceutical agent Substances 0.000 description 1
- 239000000546 pharmaceutical excipient Substances 0.000 description 1
- 239000000825 pharmaceutical preparation Substances 0.000 description 1
- 229940127557 pharmaceutical product Drugs 0.000 description 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 description 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001130982A JP2002012595A (ja) | 2000-04-27 | 2001-04-27 | ミルベマイシン誘導体 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000-127209 | 2000-04-27 | ||
| JP2000127209 | 2000-04-27 | ||
| JP2001130982A JP2002012595A (ja) | 2000-04-27 | 2001-04-27 | ミルベマイシン誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002012595A JP2002012595A (ja) | 2002-01-15 |
| JP2002012595A5 true JP2002012595A5 (enExample) | 2008-06-05 |
Family
ID=26590940
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001130982A Withdrawn JP2002012595A (ja) | 2000-04-27 | 2001-04-27 | ミルベマイシン誘導体 |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JP2002012595A (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6663876B2 (en) * | 2002-04-29 | 2003-12-16 | Piedmont Pharmaceuticals, Llc | Methods and compositions for treating ectoparasite infestation |
-
2001
- 2001-04-27 JP JP2001130982A patent/JP2002012595A/ja not_active Withdrawn
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