JP2001520634A5 - - Google Patents

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Publication number
JP2001520634A5
JP2001520634A5 JP1997509507A JP50950797A JP2001520634A5 JP 2001520634 A5 JP2001520634 A5 JP 2001520634A5 JP 1997509507 A JP1997509507 A JP 1997509507A JP 50950797 A JP50950797 A JP 50950797A JP 2001520634 A5 JP2001520634 A5 JP 2001520634A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1997509507A
Other languages
English (en)
Japanese (ja)
Other versions
JP2001520634A (ja
JP3868494B2 (ja
Filing date
Publication date
Priority claimed from US08/514,451 external-priority patent/US5837809A/en
Priority claimed from US08/553,058 external-priority patent/US5821219A/en
Application filed filed Critical
Publication of JP2001520634A publication Critical patent/JP2001520634A/ja
Publication of JP2001520634A5 publication Critical patent/JP2001520634A5/ja
Application granted granted Critical
Publication of JP3868494B2 publication Critical patent/JP3868494B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

JP50950797A 1995-08-11 1996-08-12 オピオイドアンタゴニストおよびそれらの使用方法 Expired - Lifetime JP3868494B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US08/514,451 US5837809A (en) 1995-08-11 1995-08-11 Mammalian opioid receptor ligand and uses
US08/514,451 1995-08-11
US08/553,058 1995-11-03
US08/553,058 US5821219A (en) 1995-08-11 1995-11-03 Opioid antagonists and methods of their use
PCT/US1996/013305 WO1997007212A1 (en) 1995-08-11 1996-08-12 Opioid antagonists and methods of their use

Publications (3)

Publication Number Publication Date
JP2001520634A JP2001520634A (ja) 2001-10-30
JP2001520634A5 true JP2001520634A5 (enExample) 2004-09-09
JP3868494B2 JP3868494B2 (ja) 2007-01-17

Family

ID=27058205

Family Applications (1)

Application Number Title Priority Date Filing Date
JP50950797A Expired - Lifetime JP3868494B2 (ja) 1995-08-11 1996-08-12 オピオイドアンタゴニストおよびそれらの使用方法

Country Status (8)

Country Link
US (1) US5821219A (enExample)
EP (1) EP0843726B1 (enExample)
JP (1) JP3868494B2 (enExample)
AT (1) ATE323160T1 (enExample)
AU (1) AU728001B2 (enExample)
CA (1) CA2229126A1 (enExample)
DE (1) DE69636037D1 (enExample)
WO (1) WO1997007212A1 (enExample)

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EP0813065A3 (en) * 1996-06-13 1998-07-22 F. Hoffmann-La Roche Ag Modulation of LC132 (opioid-like) receptor function
CA2206192A1 (en) 1996-06-13 1997-12-13 F. Hoffmann-La Roche Ag Modulation of lc132 (opioid-like) receptor function
AU8333998A (en) * 1997-07-15 1999-02-10 Novo Nordisk A/S New use of nociceptin
WO1999003880A1 (en) * 1997-07-15 1999-01-28 Novo Nordisk A/S Nociceptin analogues
US5929035A (en) * 1998-04-14 1999-07-27 Regents Of The University Of Michigan Methods of treating intestinal disorders
GB9815618D0 (en) * 1998-07-18 1998-09-16 Univ Manchester Treatment of dyskinesia
MA26659A1 (fr) 1998-08-06 2004-12-20 Pfizer Dérivés de benzimidazole nouveaux, compositions pharmaceutiques les contenant et procédé pour leur préparation.
US6582457B2 (en) * 2001-02-15 2003-06-24 Radiant Medical, Inc. Method of controlling body temperature while reducing shivering
US6849449B2 (en) * 2001-03-01 2005-02-01 Regents Of The University Of Michigan Orphanin FQ receptor nucleic acids
US20030040479A1 (en) * 2001-07-02 2003-02-27 Omeros Corporation Rotational intrathecal analgesia method and device
EP1406629A1 (en) * 2001-07-02 2004-04-14 Omeros Corporation Method for inducing analgesia comprising administration alternatively of an opioid receptor agonist and an opioid receptor like receptor 1 agonist for and an implantable infusion pump
WO2003030828A2 (en) * 2001-10-09 2003-04-17 Synvax, Inc. Nociceptin-based analgesics
ES2348604T3 (es) * 2002-04-29 2010-12-09 Euro-Celtique S.A. Péptidos conformacionalmente restringidos que se unen al receptor orl-1.
AU2003257111A1 (en) * 2002-08-02 2004-02-23 Incyte Corporation Extracellular messengers
EA009369B1 (ru) 2002-09-09 2007-12-28 Янссен Фармацевтика, Н.В. Производные гидроксизамещенного 1,3,8-триазинспиро[4,5]декан-4-она, полезные для лечения расстройств, опосредованных orl-рецептором
BRPI0409133B8 (pt) 2003-04-08 2021-05-25 Progenics Pharm Inc preparações farmacêuticas estavéis compreendendo metilnaltrexona
US7173010B2 (en) * 2003-05-19 2007-02-06 Regents Of The University Of Michigan Orphanin FQ receptor
US8524731B2 (en) 2005-03-07 2013-09-03 The University Of Chicago Use of opioid antagonists to attenuate endothelial cell proliferation and migration
BRPI0608818A2 (pt) 2005-03-07 2010-01-26 Univ Chicago uso de antagonista opióides para atenuação de proliferação e migração de células endoteliais
US8518962B2 (en) 2005-03-07 2013-08-27 The University Of Chicago Use of opioid antagonists
US9662325B2 (en) 2005-03-07 2017-05-30 The University Of Chicago Use of opioid antagonists to attenuate endothelial cell proliferation and migration
AR057325A1 (es) 2005-05-25 2007-11-28 Progenics Pharm Inc Sintesis de (s)-n-metilnaltrexona, composiciones farmaceuticas y usos
AR057035A1 (es) 2005-05-25 2007-11-14 Progenics Pharm Inc SíNTESIS DE (R)-N-METILNALTREXONA, COMPOSICIONES FARMACÉUTICAS Y USOS
WO2006130416A2 (en) 2005-06-02 2006-12-07 Janssen Pharmaceutica, N.V. Novel 3-spirocyclic indolyl derivatives useful as orl-1 receptor modulators
TWI489984B (zh) 2006-08-04 2015-07-01 Wyeth Corp 用於非經腸道傳輸化合物之配方及其用途
MX2009005641A (es) 2006-11-28 2009-06-05 Janssen Pharmaceutica Nv Sales de 3-(3-amino-2-(r)-hidroxi-propil)-1-(4-fluoro-fenil)-8-(8- metil-naftalen-1-ilmetil)-1,3,8-triaza-espiro[4,5]deca n-4-ona.
EP2134718A2 (en) 2007-03-29 2009-12-23 Progenics Pharmaceuticals, Inc. Crystal forms of (r)-n-methylnaltrexone bromide and uses thereof
PT2139890E (pt) 2007-03-29 2014-09-03 Wyeth Llc Antagonistas do receptor opióide periférico e respectivas utilizações
CA2682125C (en) 2007-03-29 2015-06-16 Progenics Pharmaceuticals, Inc. Peripheral opioid receptor antagonists and uses thereof
CN101679430B (zh) 2007-04-09 2013-12-25 詹森药业有限公司 用于治疗焦虑和抑郁症的作为orl-1受体的配体的1,3,8-三取代-1,3,8-三氮杂-螺[4.5]癸-4-酮衍生物
JP2010527980A (ja) 2007-05-22 2010-08-19 プロシディオン・リミテッド 代謝障害を治療するための二環状アリールおよびヘテロアリール化合物
US8063247B2 (en) 2007-09-07 2011-11-22 Prosidion Limited Bicyclic aryl and heteroaryl receptor modulators
CA2713568C (en) 2008-02-06 2016-09-20 Progenics Pharmaceuticals, Inc. Preparation and use of (r),(r)-2,2'-bis-methylnaltrexone
AU2009225434B2 (en) 2008-03-21 2014-05-22 The University Of Chicago Treatment with opioid antagonists and mTOR inhibitors
CA2676881C (en) 2008-09-30 2017-04-25 Wyeth Peripheral opioid receptor antagonists and uses thereof
RU2492482C1 (ru) * 2012-10-08 2013-09-10 Игорь Петрович Папышев Способ диагностики причины смерти от интоксикации наркотическими веществами группы опиатов

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US4582820A (en) * 1982-12-23 1986-04-15 Research Corporation Orally administered biologically active peptides and proteins
US4683195A (en) * 1986-01-30 1987-07-28 Cetus Corporation Process for amplifying, detecting, and/or-cloning nucleic acid sequences
US4683202A (en) * 1985-03-28 1987-07-28 Cetus Corporation Process for amplifying nucleic acid sequences
US5017689A (en) * 1989-07-06 1991-05-21 Arizona Technology Development Corporation Dynorphin analogs specific for kappa opioid receptors
US5512578A (en) * 1992-09-21 1996-04-30 Albert Einstein College Of Medicine Of Yeshiva University, A Division Of Yeshiva University Method of simultaneously enhancing analgesic potency and attenuating dependence liability caused by exogenous and endogenous opiod agonists
US6235496B1 (en) * 1993-03-08 2001-05-22 Advanced Research & Technology Institute Nucleic acid encoding mammalian mu opioid receptor

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