JP2000513334A - 一種以上の抗膣炎薬および一種以上の局部麻酔剤を含む局部使用用抗膣炎組成物 - Google Patents
一種以上の抗膣炎薬および一種以上の局部麻酔剤を含む局部使用用抗膣炎組成物Info
- Publication number
- JP2000513334A JP2000513334A JP09541785A JP54178597A JP2000513334A JP 2000513334 A JP2000513334 A JP 2000513334A JP 09541785 A JP09541785 A JP 09541785A JP 54178597 A JP54178597 A JP 54178597A JP 2000513334 A JP2000513334 A JP 2000513334A
- Authority
- JP
- Japan
- Prior art keywords
- lidocaine
- vaginitis
- composition
- pessary
- anesthetic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Gynecology & Obstetrics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Reproductive Health (AREA)
- Organic Chemistry (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Description
Claims (1)
- 【特許請求の範囲】 1.一種以上の抗膣炎薬と一種以上の局部麻酔剤を含む、膣炎の治療における局 部投与のための医薬組成物。 2.上記薬剤(複数でもよい)および/または局部麻酔剤(複数でもよい)の、 急速または遅延(持続)放出、或いはその両方のための処方である請求項1記載 の組成物。 3.遊離塩基形態および塩形態の両方の麻酔剤を用いることにより、局部麻酔剤 の急速および遅延放出がもたらされる請求項2記載の組成物。 4.急速放出のための、上記一種以上の薬剤および上記一種以上の局部麻酔剤を 含有するクリームまたはペッサリー基剤と、一種以上の局部麻酔剤の遅延放出の ための上記基剤中に分散された多孔性粒子とからなる請求項2記載の組成物。 5.上記一種以上の薬剤の遅延放出のための多孔性粒子を含む請求項2〜4の何 れかに記載の組成物。 6.上記薬剤が、メトロニダゾールおよびミコナゾールである上記請求項の何れ かに記載の組成物。 7.上記局部麻酔剤が、リドカインまたはベンゾカインである上記請求項の何 れかに記載の組成物。 8.界面活性剤を含む上記請求項の何れかに記載の組成物。 9.ペッサリーの形態である上記請求項の何れかに記載の組成物。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9610359.3 | 1996-05-17 | ||
GBGB9610359.3A GB9610359D0 (en) | 1996-05-17 | 1996-05-17 | Pharmaceutical compositions |
PCT/GB1997/001355 WO1997044032A1 (en) | 1996-05-17 | 1997-05-16 | Anti-vaginitis composition for topical use comprising one or more anti-vaginitis medicaments and one or more local anaesthetics |
Publications (1)
Publication Number | Publication Date |
---|---|
JP2000513334A true JP2000513334A (ja) | 2000-10-10 |
Family
ID=10793879
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP09541785A Pending JP2000513334A (ja) | 1996-05-17 | 1997-05-16 | 一種以上の抗膣炎薬および一種以上の局部麻酔剤を含む局部使用用抗膣炎組成物 |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0910377A1 (ja) |
JP (1) | JP2000513334A (ja) |
CN (1) | CN1127338C (ja) |
AU (1) | AU2905597A (ja) |
BR (1) | BR9709316A (ja) |
GB (1) | GB9610359D0 (ja) |
ID (1) | ID16929A (ja) |
MY (1) | MY127711A (ja) |
RU (1) | RU2195281C2 (ja) |
TR (1) | TR199802351T2 (ja) |
WO (1) | WO1997044032A1 (ja) |
ZA (1) | ZA974266B (ja) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007518797A (ja) * | 2004-01-22 | 2007-07-12 | アルパリス エセ.アー. デー セ.ウーベ. | 膣感染症の処置のための、フルコナゾール−チニダゾールの組み合わせ、ならびに、その組成物、調製プロセスおよび使用 |
JP4865792B2 (ja) * | 2005-07-12 | 2012-02-01 | 赴朝 李 | 局所麻酔薬の効果増強・時間延長剤 |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2777783A1 (fr) * | 1998-04-24 | 1999-10-29 | Innothera Lab Sa | Association pharmaceutique d'imidazoles pour le traitement local des vulvo-vaginites infectieuses et des vaginoses |
US5993836A (en) * | 1998-04-28 | 1999-11-30 | Castillo; James G. | Topical anesthetic formulation |
TWI232111B (en) * | 1999-08-06 | 2005-05-11 | Upjohn Co | Intravaginal clindamycin ovule composition |
US20030114394A1 (en) * | 2001-10-29 | 2003-06-19 | Levine Howard L. | Vaginally administered anti-dysrhythmic agents for treating pelvic pain |
US8425892B2 (en) | 2001-10-29 | 2013-04-23 | Columbia Laboratories, Inc. | Extended, controlled-release pharmaceutical compositions using charged polymers |
BRPI0414500A (pt) | 2003-09-19 | 2006-11-07 | Drugtech Corp | formulação farmacêutica composição para tratar uma infecção vaginal, e, métodos para tratar uma infecção vaginal, para estabilizar uma formulação de clindamicina, para tratar ou prevenir uma recorrência de uma infecção vaginal em uma paciente e para tratar condições vaginais |
GB0405406D0 (en) * | 2004-03-10 | 2004-04-21 | Edko Pazarlama Tanitim Ltd Sti | Anti-vaginitis compositions |
AU2006244260A1 (en) * | 2005-05-09 | 2006-11-16 | Drugtech Corporation | Modified-release pharmaceutical compositions |
CA2635994A1 (en) * | 2006-01-05 | 2007-07-12 | Drugtech Corporation | Drug delivery system for bioadhesion to a vulvovaginal surface |
EA200870153A1 (ru) * | 2006-01-05 | 2008-12-30 | Драгтек Корпорейшн | Композиция и способ ее использования |
RU2603490C1 (ru) * | 2015-11-30 | 2016-11-27 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Курский государственный медицинский университет" Министерства здравоохранения Российской Федерации | Средство для лечения гнойно-воспалительных процессов мягких тканей и слизистых оболочек |
RU2605343C1 (ru) * | 2015-11-30 | 2016-12-20 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Курский государственный медицинский университет" Министерства здравоохранения Российской Федерации | Средство для лечения гнойно-воспалительных процессов мягких тканей и слизистых оболочек |
KR20190026686A (ko) | 2016-07-08 | 2019-03-13 | 아지엔드 키미쉐 리유나이트 안젤리니 프란체스코 에이.씨.알.에이.에프. 에스.피.에이 | 벤지다민을 포함하는 약학적 조성물 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8830405D0 (en) * | 1988-12-30 | 1989-03-01 | Embil Koral | Pharmaceutical formulation |
-
1996
- 1996-05-17 GB GBGB9610359.3A patent/GB9610359D0/en active Pending
-
1997
- 1997-05-15 MY MYPI97002126A patent/MY127711A/en unknown
- 1997-05-16 BR BR9709316-5A patent/BR9709316A/pt not_active Application Discontinuation
- 1997-05-16 WO PCT/GB1997/001355 patent/WO1997044032A1/en not_active Application Discontinuation
- 1997-05-16 ZA ZA974266A patent/ZA974266B/xx unknown
- 1997-05-16 EP EP97923187A patent/EP0910377A1/en not_active Withdrawn
- 1997-05-16 CN CN97195988A patent/CN1127338C/zh not_active Expired - Fee Related
- 1997-05-16 AU AU29055/97A patent/AU2905597A/en not_active Abandoned
- 1997-05-16 TR TR1998/02351T patent/TR199802351T2/xx unknown
- 1997-05-16 RU RU98122669/14A patent/RU2195281C2/ru not_active IP Right Cessation
- 1997-05-16 JP JP09541785A patent/JP2000513334A/ja active Pending
- 1997-05-19 ID IDP971652A patent/ID16929A/id unknown
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007518797A (ja) * | 2004-01-22 | 2007-07-12 | アルパリス エセ.アー. デー セ.ウーベ. | 膣感染症の処置のための、フルコナゾール−チニダゾールの組み合わせ、ならびに、その組成物、調製プロセスおよび使用 |
JP4865792B2 (ja) * | 2005-07-12 | 2012-02-01 | 赴朝 李 | 局所麻酔薬の効果増強・時間延長剤 |
Also Published As
Publication number | Publication date |
---|---|
TR199802351T2 (xx) | 1999-03-22 |
CN1223581A (zh) | 1999-07-21 |
ID16929A (id) | 1997-11-20 |
GB9610359D0 (en) | 1996-07-24 |
WO1997044032A1 (en) | 1997-11-27 |
RU2195281C2 (ru) | 2002-12-27 |
CN1127338C (zh) | 2003-11-12 |
EP0910377A1 (en) | 1999-04-28 |
AU2905597A (en) | 1997-12-09 |
ZA974266B (en) | 1998-11-16 |
MY127711A (en) | 2006-12-29 |
BR9709316A (pt) | 2000-05-02 |
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Legal Events
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