JP2000504014A - ファルネシル―タンパク質転移酵素の阻害剤 - Google Patents
ファルネシル―タンパク質転移酵素の阻害剤Info
- Publication number
- JP2000504014A JP2000504014A JP9527779A JP52777997A JP2000504014A JP 2000504014 A JP2000504014 A JP 2000504014A JP 9527779 A JP9527779 A JP 9527779A JP 52777997 A JP52777997 A JP 52777997A JP 2000504014 A JP2000504014 A JP 2000504014A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- hydrogen
- unsubstituted
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1079896P | 1996-01-30 | 1996-01-30 | |
| GBGB9605708.8A GB9605708D0 (en) | 1996-03-19 | 1996-03-19 | Inhibitors of farnesyl-protein transferase |
| GB60/010,798 | 1996-03-19 | ||
| GB9605708.8 | 1996-03-19 | ||
| PCT/US1997/001354 WO1997027852A1 (en) | 1996-01-30 | 1997-01-27 | Inhibitors of farnesyl-protein transferase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JP2000504014A true JP2000504014A (ja) | 2000-04-04 |
Family
ID=26308955
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP9527779A Pending JP2000504014A (ja) | 1996-01-30 | 1997-01-27 | ファルネシル―タンパク質転移酵素の阻害剤 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US6066738A (OSRAM) |
| EP (1) | EP0944387A1 (OSRAM) |
| JP (1) | JP2000504014A (OSRAM) |
| AU (1) | AU703203B2 (OSRAM) |
| WO (1) | WO1997027852A1 (OSRAM) |
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| AU7997600A (en) | 1999-10-08 | 2001-04-23 | Du Pont Pharmaceuticals Company | Amino lactam sulfonamides as inhibitors of abeta protein production |
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| AU706008B2 (en) * | 1995-03-29 | 1999-06-03 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| CN1219174A (zh) * | 1996-05-22 | 1999-06-09 | 沃尼尔·朗伯公司 | 蛋白质法呢基转移酶的抑制剂 |
-
1997
- 1997-01-27 US US09/117,260 patent/US6066738A/en not_active Expired - Fee Related
- 1997-01-27 WO PCT/US1997/001354 patent/WO1997027852A1/en not_active Ceased
- 1997-01-27 JP JP9527779A patent/JP2000504014A/ja active Pending
- 1997-01-27 AU AU18444/97A patent/AU703203B2/en not_active Ceased
- 1997-01-27 EP EP97904037A patent/EP0944387A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| US6066738A (en) | 2000-05-23 |
| AU1844497A (en) | 1997-08-22 |
| WO1997027852A1 (en) | 1997-08-07 |
| AU703203B2 (en) | 1999-03-18 |
| EP0944387A4 (OSRAM) | 1999-09-29 |
| EP0944387A1 (en) | 1999-09-29 |
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