JP2000500489A5 - - Google Patents

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Publication number
JP2000500489A5
JP2000500489A5 JP1997519726A JP51972697A JP2000500489A5 JP 2000500489 A5 JP2000500489 A5 JP 2000500489A5 JP 1997519726 A JP1997519726 A JP 1997519726A JP 51972697 A JP51972697 A JP 51972697A JP 2000500489 A5 JP2000500489 A5 JP 2000500489A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP1997519726A
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English (en)
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JP2000500489A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1996/017120 external-priority patent/WO1997019089A1/en
Publication of JP2000500489A publication Critical patent/JP2000500489A/ja
Publication of JP2000500489A5 publication Critical patent/JP2000500489A5/ja
Withdrawn legal-status Critical Current

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Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
Figure 2000500489
JP9519726A 1995-11-17 1996-11-05 三環置換基を有するオキサゾリジノン抗菌剤 Withdrawn JP2000500489A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US737195P 1995-11-17 1995-11-17
US60/007,371 1995-11-17
PCT/US1996/017120 WO1997019089A1 (en) 1995-11-17 1996-11-05 Oxazolidinone antibacterial agent with tricyclic substituents

Publications (2)

Publication Number Publication Date
JP2000500489A JP2000500489A (ja) 2000-01-18
JP2000500489A5 true JP2000500489A5 (ja) 2004-08-12

Family

ID=21725778

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9519726A Withdrawn JP2000500489A (ja) 1995-11-17 1996-11-05 三環置換基を有するオキサゾリジノン抗菌剤

Country Status (12)

Country Link
US (2) US5922707A (ja)
EP (1) EP0874852B1 (ja)
JP (1) JP2000500489A (ja)
AT (1) ATE263172T1 (ja)
AU (1) AU7665196A (ja)
DE (1) DE69632074T2 (ja)
DK (1) DK0874852T3 (ja)
ES (1) ES2217329T3 (ja)
PT (1) PT874852E (ja)
TW (1) TW426683B (ja)
WO (1) WO1997019089A1 (ja)
ZA (1) ZA968661B (ja)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA968661B (en) * 1995-11-17 1998-04-14 Upjohn Co Oxazolidinone antibacterial agent with tricyclic substituents.
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) * 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
CN1265660A (zh) * 1997-08-15 2000-09-06 辉瑞产品公司 2-(4-芳基或杂芳基-哌嗪-1-基甲基)-1h-吲哚衍生物
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
DE19802235A1 (de) * 1998-01-22 1999-07-29 Bayer Ag Mit tricyclischen Indolen substituierte Oxazolidinone
DE19802239A1 (de) * 1998-01-22 1999-07-29 Bayer Ag Neue mit Bicyclen substituierte Oxazolidinone
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
NZ505902A (en) 1998-01-23 2003-08-29 Upjohn Co Oxazolidinone compounds useful as antimicrobial agents and combinatorial libraries
DE19805117A1 (de) * 1998-02-09 1999-08-12 Bayer Ag Neue Oxazolidinone mit azolhaltigen Tricyclen
MY122454A (en) * 1998-06-05 2006-04-29 Upjohn Co Use of oxazolidinones for the preparation of a medicament for transdermal delivery
EP1082323A2 (en) 1998-06-05 2001-03-14 AstraZeneca UK Limited Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
EP1122242B1 (en) 1998-09-22 2008-01-16 Astellas Pharma Inc. Cyanophenyl derivatives
JP2002535680A (ja) 1999-01-27 2002-10-22 ファルマシア・アンド・アップジョン・カンパニー 延長因子p活性モジュレーターのアッセイ方法
WO2000073301A1 (en) 1999-05-27 2000-12-07 Pharmacia & Upjohn Company Bicyclic oxazolidinones as antibacterial agent
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
GB0009803D0 (en) * 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
JP2005537301A (ja) 2002-08-12 2005-12-08 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー N−アリール−2−オキサゾリジノン類及びそれらの誘導体
AR042086A1 (es) 2002-11-21 2005-06-08 Upjohn Co N-aril-2- oxazolidinon -5- carboxamidas y sus derivados, usados como agentes antibacterianos
JP2006516991A (ja) * 2003-02-07 2006-07-13 ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー 抗菌剤
US7795267B2 (en) * 2003-08-29 2010-09-14 Takeda Pharmaceutical Company Limited Bicyclic piperazine compound having TGR23 antagonistic activity
AR057828A1 (es) * 2005-09-29 2007-12-19 Astrazeneca Ab Compuestos derivados de azetidina, su preparacion y composicion farmaceuutica
MX2008009475A (es) * 2006-01-23 2008-10-20 Amira Pharmaceuticals Inc Inhibidores triciclicos de 5-lipoxigenasa.
CN110734454B (zh) * 2016-12-12 2021-08-17 石药集团中奇制药技术(石家庄)有限公司 一类含有三环杂芳基的化合物

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883522A (en) * 1974-02-11 1975-05-13 Riker Laboratories Inc Substituted pyrido(1,2,3-de)-1,4-benzoxazines
US4080499A (en) * 1976-12-20 1978-03-21 1 Substituted 7,8-dihydro-6H-(1,2,5)thiadiazolo(3',4'-5,6)pyrazino(2,3-b)(1,4)oxazines
US5039690A (en) * 1987-10-09 1991-08-13 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5225565A (en) * 1988-09-15 1993-07-06 The Upjohn Company Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones
DE68929303T2 (de) * 1988-09-15 2002-05-02 Upjohn Co 3-(Stickstoff substituierte)phenyl-5-beta-amidomethyloxazoliden-2-one
EP0625982B1 (en) * 1992-02-13 2002-06-12 PHARMACIA & UPJOHN COMPANY 4-oxo- and 4h-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
US5668286A (en) * 1994-03-15 1997-09-16 Pharmacia & Upjohn Company Oxazolidinone derivatives and pharmaceutical compositions containing them
US5952324A (en) * 1994-11-15 1999-09-14 Pharmacia & Upjohn Company Bicyclic oxazine and thiazine oxazolidinone antibacterials
ZA968661B (en) * 1995-11-17 1998-04-14 Upjohn Co Oxazolidinone antibacterial agent with tricyclic substituents.

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