IT1312539B1 - Processo per la preparazione del pirlindolo cloridrato. - Google Patents

Processo per la preparazione del pirlindolo cloridrato.

Info

Publication number
IT1312539B1
IT1312539B1 IT1999MI000802A ITMI990802A IT1312539B1 IT 1312539 B1 IT1312539 B1 IT 1312539B1 IT 1999MI000802 A IT1999MI000802 A IT 1999MI000802A IT MI990802 A ITMI990802 A IT MI990802A IT 1312539 B1 IT1312539 B1 IT 1312539B1
Authority
IT
Italy
Prior art keywords
hydrochloride
pyrindol
preparation
methyl
formula
Prior art date
Application number
IT1999MI000802A
Other languages
English (en)
Inventor
Massimo Ferrari
Marcello Ghezzi
Paolo Belotti
Fabrizio Zinetti
Original Assignee
Erregierre Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to IT1999MI000802A priority Critical patent/IT1312539B1/it
Application filed by Erregierre Spa filed Critical Erregierre Spa
Priority to DE60000274T priority patent/DE60000274T2/de
Priority to PT00107836T priority patent/PT1044976E/pt
Priority to AT00107836T priority patent/ATE221070T1/de
Priority to EP00107836A priority patent/EP1044976B1/en
Priority to ES00107836T priority patent/ES2180483T3/es
Priority to PL00339641A priority patent/PL339641A1/xx
Priority to HU0001558A priority patent/HUP0001558A3/hu
Priority to RU2000109633/04A priority patent/RU2249592C2/ru
Publication of ITMI990802A1 publication Critical patent/ITMI990802A1/it
Application granted granted Critical
Publication of IT1312539B1 publication Critical patent/IT1312539B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Saccharide Compounds (AREA)
IT1999MI000802A 1999-04-16 1999-04-16 Processo per la preparazione del pirlindolo cloridrato. IT1312539B1 (it)

Priority Applications (9)

Application Number Priority Date Filing Date Title
IT1999MI000802A IT1312539B1 (it) 1999-04-16 1999-04-16 Processo per la preparazione del pirlindolo cloridrato.
PT00107836T PT1044976E (pt) 1999-04-16 2000-04-12 Processo para a preparacao de cloridrato de pirlindole
AT00107836T ATE221070T1 (de) 1999-04-16 2000-04-12 Verfahren zur herstelung von pirlindolehydrochlorid
EP00107836A EP1044976B1 (en) 1999-04-16 2000-04-12 Process for the preparation of pirlindole hydrochloride
DE60000274T DE60000274T2 (de) 1999-04-16 2000-04-12 Verfahren zur Herstelung von Pirlindolehydrochlorid
ES00107836T ES2180483T3 (es) 1999-04-16 2000-04-12 Proceso mejorado para la elaboracion de clorhidrato de pirlindol.
PL00339641A PL339641A1 (en) 1999-04-16 2000-04-13 Method of obtaining pyridinole hydrochloride
HU0001558A HUP0001558A3 (en) 1999-04-16 2000-04-14 Process for the preparation of pirlindole hydrochloride
RU2000109633/04A RU2249592C2 (ru) 1999-04-16 2000-04-14 Способ получения гидрохлорида пирлиндола

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999MI000802A IT1312539B1 (it) 1999-04-16 1999-04-16 Processo per la preparazione del pirlindolo cloridrato.

Publications (2)

Publication Number Publication Date
ITMI990802A1 ITMI990802A1 (it) 2000-10-16
IT1312539B1 true IT1312539B1 (it) 2002-04-22

Family

ID=11382759

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1999MI000802A IT1312539B1 (it) 1999-04-16 1999-04-16 Processo per la preparazione del pirlindolo cloridrato.

Country Status (9)

Country Link
EP (1) EP1044976B1 (it)
AT (1) ATE221070T1 (it)
DE (1) DE60000274T2 (it)
ES (1) ES2180483T3 (it)
HU (1) HUP0001558A3 (it)
IT (1) IT1312539B1 (it)
PL (1) PL339641A1 (it)
PT (1) PT1044976E (it)
RU (1) RU2249592C2 (it)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9617517B2 (en) 2011-05-02 2017-04-11 National University Corporation Kumamoto University Small chemical compound which promotes induction of differentiation of stem cells into insulin-producing cells and method for inducing differentiation of stem cells into insulin-producing cells using said small chemical compound
CN102952089B (zh) * 2012-10-19 2015-07-08 江苏省农用激素工程技术研究中心有限公司 苯嗪草酮的制备方法
CN104774208A (zh) * 2015-04-24 2015-07-15 南京靖龙药物研发有限公司 一种氘标记吡吲哚盐酸盐的制备方法
EP3392250A1 (en) * 2017-04-21 2018-10-24 Tecnimede-Sociedade Tecnico-Medicinal, S.A. Process for the preparation of piperazine ring for the synthesis of pyrazinocarbazole derivatives
EP3392251A1 (en) * 2017-04-21 2018-10-24 Tecnimede-Sociedade Tecnico-Medicinal, S.A. Process for the preparation of pirlindole enantiomers and its salts
CN110950873A (zh) * 2019-12-10 2020-04-03 河南大学 坡尔吲哚的合成新方法

Also Published As

Publication number Publication date
ATE221070T1 (de) 2002-08-15
DE60000274T2 (de) 2003-03-06
HUP0001558A3 (en) 2003-08-28
HUP0001558A2 (hu) 2001-04-28
PL339641A1 (en) 2000-10-23
HU0001558D0 (en) 2000-06-28
EP1044976A1 (en) 2000-10-18
EP1044976B1 (en) 2002-07-24
ITMI990802A1 (it) 2000-10-16
ES2180483T3 (es) 2003-02-16
DE60000274D1 (de) 2002-08-29
RU2249592C2 (ru) 2005-04-10
PT1044976E (pt) 2002-12-31

Similar Documents

Publication Publication Date Title
MY136270A (en) Processes and intermediates for preparing anti-cancer compounds
NO20053115D0 (no) Fremgangsmate for fremstilling av 2'-forgrenede nukleosider.
AP2002002637A0 (en) Novel piperazine
FI915920A0 (fi) Serotoninantagonister.
RU92004368A (ru) Замещенные пиримидины, способ их получения, фармацевтическая композиция
MXPA03011954A (es) Nuevos derivados de acido sulfonico.
DE69229339D1 (de) Kristallines tiagabinehydrochlorid-monohydrat, seine herstellung und verwendung
PT992509E (pt) Novos derivados macrolidos
BRPI0409376A (pt) derivados de indeno como agentes farmacêuticos
IT1312539B1 (it) Processo per la preparazione del pirlindolo cloridrato.
TR199500956A2 (tr) Benzimidazol türevleri.
IS6914A (is) 2-þíó-útskiptar imídasólafleiður og notkun þeirraí lyfjaiðnaðinum
IT1274997B (it) Procedimento per la produzione di spazzole nonche' macchina per la produzione di spazzole per l'esecuzione del procedimento
IT1319242B1 (it) Processo per la preparazione di maleato di fluvossamina.
AR041116A1 (es) Metodos para tratar pacientes que sufen el sindrome de piernas inquietas o desordenes relacionados
EP0812844A3 (de) Verwendung von Theophyllinderivaten zur Behandlung und Propylaxe von Schockzuständen, neue Xanthinverbindungen und Verfahren zu deren Herstellung
ITMI991731A0 (it) Processo per la preparazione di derivati 3-sostituiti di 4-fenil-piper idine
ITMI991950A0 (it) Procedimento per la sintesi del ritomavir
NO20042729L (no) Heksasykliske forbindelser
ES2063266T3 (es) 4,5,6,11-tetrahidrobenzo(6,7)cicloocta(1,2-b)tiofen-6,11-iminas y 6,11-dihidrobenzo(6,7)cicloocta(1,2-b)tiofen-6,11-iminas.
PT889044E (pt) Derivados do 5-(heteroaril)alquil-3-oxo-pirido-(1,2-a)benzimidazole-4-carboxamida (pbi) uteis no tratamento de perturbacoes do sistema nervoso central
IT1244036B (it) Processo per la preparazione del 4-nitro-benzoato di 4-(2,4- difluorofenil)-fenile
PT952157E (pt) Derivados 9a, 11b-desidro de 9-oxima-3-ceto-6-o-metileritromicina
IT1312551B1 (it) Processo per la sintesi di 5-alchilbenzodiossoli
ATE338759T1 (de) 2-(aminomethyl)tetrahydro-9-oxa-1,3- diazacyclopentaca)naphthalinylderivate mit antipsychotischer wirkung