IT1251114B - Forme farmaceutiche antivirali per applicazione vaginale - Google Patents

Forme farmaceutiche antivirali per applicazione vaginale

Info

Publication number
IT1251114B
IT1251114B ITMI912071A ITMI912071A IT1251114B IT 1251114 B IT1251114 B IT 1251114B IT MI912071 A ITMI912071 A IT MI912071A IT MI912071 A ITMI912071 A IT MI912071A IT 1251114 B IT1251114 B IT 1251114B
Authority
IT
Italy
Prior art keywords
tablets
effervescent
vaginal
pharmaceutical forms
preparation
Prior art date
Application number
ITMI912071A
Other languages
English (en)
Inventor
Ubaldo Conte
Lauretta Maggi
Original Assignee
Farcon Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farcon Ag filed Critical Farcon Ag
Publication of ITMI912071A0 publication Critical patent/ITMI912071A0/it
Priority to ITMI912071A priority Critical patent/IT1251114B/it
Priority to DK92915980.4T priority patent/DK0596935T3/da
Priority to DE69205579T priority patent/DE69205579T2/de
Priority to PCT/EP1992/001655 priority patent/WO1993002662A1/en
Priority to EP92915980A priority patent/EP0596935B1/en
Priority to JP5503217A priority patent/JPH06509348A/ja
Priority to AU23454/92A priority patent/AU2345492A/en
Priority to AT92915980T priority patent/ATE129149T1/de
Priority to CA002114216A priority patent/CA2114216A1/en
Priority to CN92111077A priority patent/CN1082894A/zh
Publication of ITMI912071A1 publication Critical patent/ITMI912071A1/it
Application granted granted Critical
Publication of IT1251114B publication Critical patent/IT1251114B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer

Abstract

Sono descritti preparati farmaceutici destinati alla somministrazione vaginale di farmaci antivirali, preferibilmente di acyclovir. Forme farmaceutiche adatte sono:a) compresse vaginali erodibili e compresse vaginali effervescenti b) compresse effervescenti destinate alla preparazione di bagni medicati e/o granulare effervescente o solubile o dispersibile in acqua per la preparazione di bagni medicati c) compresse ad un solo strato (in genere destinate ad un rilascio immediato della sostanza attiva o al rilascio prolungato o sostenuto)d) compresse a due o più strati (essendo ciascuno dei differenti strati progettato per determinare differenti velocità di rilascio).
ITMI912071A 1991-07-26 1991-07-26 Forme farmaceutiche antivirali per applicazione vaginale IT1251114B (it)

Priority Applications (10)

Application Number Priority Date Filing Date Title
ITMI912071A IT1251114B (it) 1991-07-26 1991-07-26 Forme farmaceutiche antivirali per applicazione vaginale
EP92915980A EP0596935B1 (en) 1991-07-26 1992-07-20 Antiviral pharmaceutical compositions for vaginal administration
DE69205579T DE69205579T2 (de) 1991-07-26 1992-07-20 Virushemmende pharmazeutische zubereitungen zur vaginalen verabreichung.
PCT/EP1992/001655 WO1993002662A1 (en) 1991-07-26 1992-07-20 Antiviral pharmaceutical compositions for vaginal administration
DK92915980.4T DK0596935T3 (da) 1991-07-26 1992-07-20 Antivirale farmaceutiske midler til vaginal administration
JP5503217A JPH06509348A (ja) 1991-07-26 1992-07-20 経膣投与用の抗ウイルス性薬剤組成物
AU23454/92A AU2345492A (en) 1991-07-26 1992-07-20 Antiviral pharmaceutical compositions for vaginal administration
AT92915980T ATE129149T1 (de) 1991-07-26 1992-07-20 Virushemmende pharmazeutische zubereitungen zur vaginalen verabreichung.
CA002114216A CA2114216A1 (en) 1991-07-26 1992-07-20 Antiviral pharmaceutical compositions for vaginal administration
CN92111077A CN1082894A (zh) 1991-07-26 1992-08-24 阴道给药的抗病毒药物组合物

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI912071A IT1251114B (it) 1991-07-26 1991-07-26 Forme farmaceutiche antivirali per applicazione vaginale
CN92111077A CN1082894A (zh) 1991-07-26 1992-08-24 阴道给药的抗病毒药物组合物

Publications (3)

Publication Number Publication Date
ITMI912071A0 ITMI912071A0 (it) 1991-07-26
ITMI912071A1 ITMI912071A1 (it) 1993-01-27
IT1251114B true IT1251114B (it) 1995-05-04

Family

ID=36790864

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI912071A IT1251114B (it) 1991-07-26 1991-07-26 Forme farmaceutiche antivirali per applicazione vaginale

Country Status (10)

Country Link
EP (1) EP0596935B1 (it)
JP (1) JPH06509348A (it)
CN (1) CN1082894A (it)
AT (1) ATE129149T1 (it)
AU (1) AU2345492A (it)
CA (1) CA2114216A1 (it)
DE (1) DE69205579T2 (it)
DK (1) DK0596935T3 (it)
IT (1) IT1251114B (it)
WO (1) WO1993002662A1 (it)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4139883A1 (de) * 1991-11-29 1993-06-03 Michael Prof Dr Dittgen Verfahren zur herstellung bioadhaesiver arzneimittel
FR2710265B1 (fr) * 1993-09-22 1995-10-20 Adir Composition pharmaceutique bioadhésive pour la libération contrôlée de principes actifs.
DE4404011A1 (de) * 1994-02-09 1995-08-10 Jenapharm Gmbh Neue, adhäsiv wirkende Zubereitungen für mit Flüssigkeit benetzte Oberflächen, Verfahren und Vorrichtung zur Erfassung der Adhäsionszeit diesbezüglicher Zubereitungen
US6818672B1 (en) 1999-10-05 2004-11-16 Columbia Laboratories, Inc. Treating endometriosis or infertility, or improving fertility
UA74168C2 (uk) * 1999-10-05 2005-11-15 Коламбіа Леборетеріс (Бермуда) Лімітед Лікування ендометріозу або безпліддя, або покращення плідності та застосування бета-адренергічного агоніста для виробництва лікарського засобу
BR0007360A (pt) * 1999-12-23 2001-08-14 Johnson & Johnson Composição de liberação controlada
JP2001240558A (ja) * 2000-02-29 2001-09-04 Nippon Suisan Kaisha Ltd 多価不飽和脂肪酸を経粘膜吸収促進剤として含有する固形製剤。
EP1318790A4 (en) * 2000-09-19 2006-02-01 Cima Labs Inc PHARMACEUTICAL COMPOSITIONS FOR RECTAL AND VAGINAL ADMINISTRATION
MY144021A (en) * 2003-09-19 2011-07-29 Drugtech Corp Pharmaceutical delivery system
CA2548915C (en) 2003-12-31 2012-10-16 Cima Labs Inc. Generally linear effervescent oral fentanyl dosage form and methods of administering
US7862833B2 (en) 2003-12-31 2011-01-04 Cima Labs, Inc. Effervescent oral opiate dosage forms and methods of administering opiates
EP2662086A1 (en) * 2012-05-08 2013-11-13 Progressare Medinvest B.V. Composition for the treatment or prevention of urinary tract infections and dosage form

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3388041A (en) * 1964-01-27 1968-06-11 Richardson Merrell Inc High dosage sustained release tablet
JPS52156913A (en) * 1976-06-21 1977-12-27 Toko Yakuhin Kogyo Kk Production of injectionable medicine
JPS5562012A (en) * 1978-11-06 1980-05-10 Teijin Ltd Slow-releasing preparation
JPS58152809A (ja) * 1982-03-05 1983-09-10 Eisai Co Ltd 安定な発泡性「膣」坐剤
US4389393A (en) * 1982-03-26 1983-06-21 Forest Laboratories, Inc. Sustained release therapeutic compositions based on high molecular weight hydroxypropylmethylcellulose
IT1187750B (it) * 1985-10-15 1987-12-23 Eurand Spa Procedimento per la preparazione di compresse,anche a rilascio prolungato,di iscsorbide-5-mononitrato stabilizzato e formulazioni cosi' ottenute
IT1213323B (it) * 1986-08-07 1989-12-20 Crinos Industria Farmaco Composizione per uso locale ad atti vita' spermicida virulicida ,disinfettante e/o battericida
NZ222698A (en) * 1987-01-08 1990-02-26 Squibb & Sons Inc Bioadhesive suppository formulations comprising a medicament, water, a hydrocolloid and low melting point base
US4983393A (en) * 1987-07-21 1991-01-08 Maximed Corporation Intra-vaginal device and method for sustained drug release

Also Published As

Publication number Publication date
EP0596935A1 (en) 1994-05-18
DE69205579D1 (de) 1995-11-23
DE69205579T2 (de) 1996-04-04
DK0596935T3 (da) 1996-01-22
ITMI912071A0 (it) 1991-07-26
EP0596935B1 (en) 1995-10-18
JPH06509348A (ja) 1994-10-20
AU2345492A (en) 1993-03-02
ITMI912071A1 (it) 1993-01-27
CA2114216A1 (en) 1993-02-18
WO1993002662A1 (en) 1993-02-18
CN1082894A (zh) 1994-03-02
ATE129149T1 (de) 1995-11-15

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19960725