IT1146940B - Composti 2,4-diamminopirido (2,3-d) pirimidinici dotati di attivita' farmacologica e procedimento per la loro preparazione - Google Patents
Composti 2,4-diamminopirido (2,3-d) pirimidinici dotati di attivita' farmacologica e procedimento per la loro preparazioneInfo
- Publication number
- IT1146940B IT1146940B IT48968/80A IT4896880A IT1146940B IT 1146940 B IT1146940 B IT 1146940B IT 48968/80 A IT48968/80 A IT 48968/80A IT 4896880 A IT4896880 A IT 4896880A IT 1146940 B IT1146940 B IT 1146940B
- Authority
- IT
- Italy
- Prior art keywords
- diaminopyrid
- pyrimidinal
- procedure
- preparation
- pharmacological activity
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7920704 | 1979-06-14 | ||
GB7920703 | 1979-06-14 | ||
GB7920705 | 1979-06-14 | ||
GB7920706 | 1979-06-14 |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8048968A0 IT8048968A0 (it) | 1980-06-13 |
IT1146940B true IT1146940B (it) | 1986-11-19 |
Family
ID=27449125
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT48968/80A IT1146940B (it) | 1979-06-14 | 1980-06-13 | Composti 2,4-diamminopirido (2,3-d) pirimidinici dotati di attivita' farmacologica e procedimento per la loro preparazione |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0021292B1 (it) |
AU (1) | AU532842B2 (it) |
CA (1) | CA1132137A (it) |
DE (1) | DE3062268D1 (it) |
DK (1) | DK157451C (it) |
FI (1) | FI66866C (it) |
HU (1) | HU184787B (it) |
IE (1) | IE49992B1 (it) |
IL (1) | IL60307A (it) |
IT (1) | IT1146940B (it) |
MY (1) | MY8500059A (it) |
NZ (1) | NZ194045A (it) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8702758D0 (en) * | 1987-02-06 | 1987-03-11 | Wellcome Found | Treatment of disease |
EP0278686A1 (en) * | 1987-02-07 | 1988-08-17 | The Wellcome Foundation Limited | Pyridopyrimidines methods for their preparation and pharmaceutical formulations thereof |
US4889859A (en) * | 1988-02-05 | 1989-12-26 | The Trustees Of Princeton University | Pyrido[2,3-d]pyrimidine derivatives |
US5547954A (en) * | 1994-05-26 | 1996-08-20 | Fmc Corporation | 2,4-Diamino-5,6-disubstituted-and 5,6,7-trisubstituted-5-deazapteridines as insecticides |
EP1806348A3 (en) * | 1997-02-05 | 2008-01-02 | Warner-Lambert Company LLC | Pyrido [2, 3 -d] pyrimidines and 4-amino-primidines as inhibitors of cellular proliferation |
US6498163B1 (en) | 1997-02-05 | 2002-12-24 | Warner-Lambert Company | Pyrido[2,3-D]pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation |
ATE391719T1 (de) * | 1997-02-05 | 2008-04-15 | Warner Lambert Co | Pyrido (2,3-d) pyrimidine und 4-amino-primidine als inhibitoren der zellulären proliferation |
EP1801112A1 (en) * | 1998-05-26 | 2007-06-27 | Warner-Lambert Company LLC | Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation |
EA003640B1 (ru) | 1998-05-26 | 2003-08-28 | Варнер-Ламберт Компани | Бициклические пиримидины и бициклические 3,4-дигидропиримидины как ингибиторы клеточной пролиферации |
PL352159A1 (en) | 1999-05-24 | 2003-07-28 | Sankyo Co | Pharmaceutical compositions containing antibody against the fas |
CN101906104B (zh) | 2002-01-22 | 2013-06-05 | 沃尼尔·朗伯有限责任公司 | 2-(吡啶-2-基氨基)-吡啶并[2,3-d]嘧啶-7-酮 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2937284A (en) * | 1958-05-01 | 1960-05-17 | Burroughs Wellcome Co | 2, 4-diamino-5, 6-dialkylpyrido (2, 3-d) pyrimidines and method |
GB970583A (en) * | 1961-07-19 | 1964-09-23 | Wellcome Found | 2,4-diaminopyrido[2,3-d]pyrimidines |
US3322765A (en) * | 1963-10-30 | 1967-05-30 | Burroughs Wellcome Co | 2, 4-diamino-6-benzylpyrido-(2, 3-d) pyrimidines and method |
-
1980
- 1980-06-13 FI FI801912A patent/FI66866C/fi not_active IP Right Cessation
- 1980-06-13 EP EP80103325A patent/EP0021292B1/en not_active Expired
- 1980-06-13 DK DK254780A patent/DK157451C/da not_active IP Right Cessation
- 1980-06-13 HU HU801494A patent/HU184787B/hu not_active IP Right Cessation
- 1980-06-13 IE IE1220/80A patent/IE49992B1/en not_active IP Right Cessation
- 1980-06-13 DE DE8080103325T patent/DE3062268D1/de not_active Expired
- 1980-06-13 IL IL60307A patent/IL60307A/xx unknown
- 1980-06-13 AU AU59275/80A patent/AU532842B2/en not_active Expired
- 1980-06-13 IT IT48968/80A patent/IT1146940B/it active
- 1980-06-13 CA CA354,009A patent/CA1132137A/en not_active Expired
- 1980-06-13 NZ NZ194045A patent/NZ194045A/en unknown
-
1985
- 1985-12-30 MY MY59/85A patent/MY8500059A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
CA1132137A (en) | 1982-09-21 |
DK157451B (da) | 1990-01-08 |
MY8500059A (en) | 1985-12-31 |
IE49992B1 (en) | 1986-01-22 |
HU184787B (en) | 1984-10-29 |
DK157451C (da) | 1990-05-21 |
EP0021292B1 (en) | 1983-03-09 |
IT8048968A0 (it) | 1980-06-13 |
IL60307A0 (en) | 1980-09-16 |
AU5927580A (en) | 1980-12-18 |
FI66866B (fi) | 1984-08-31 |
FI66866C (fi) | 1984-12-10 |
DK254780A (da) | 1980-12-15 |
IL60307A (en) | 1984-02-29 |
NZ194045A (en) | 1984-09-28 |
AU532842B2 (en) | 1983-10-13 |
FI801912A (fi) | 1980-12-15 |
EP0021292A1 (en) | 1981-01-07 |
DE3062268D1 (en) | 1983-04-14 |
IE801220L (en) | 1980-12-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19970628 |