DK157451C - Analogifremgangsmaade til fremstilling af 2,4-diamino-6-alkoxybenzyl-5-methylpyridooe2,3-daapyrimidiner eller farmaceutisk acceptable syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 2,4-diamino-6-alkoxybenzyl-5-methylpyridooe2,3-daapyrimidiner eller farmaceutisk acceptable syreadditionssalte deraf

Info

Publication number
DK157451C
DK157451C DK254780A DK254780A DK157451C DK 157451 C DK157451 C DK 157451C DK 254780 A DK254780 A DK 254780A DK 254780 A DK254780 A DK 254780A DK 157451 C DK157451 C DK 157451C
Authority
DK
Denmark
Prior art keywords
daapyrimidines
alkoxybenzyl
diamino
analogy
preparation
Prior art date
Application number
DK254780A
Other languages
English (en)
Other versions
DK157451B (da
DK254780A (da
Inventor
Eugene Michael Grivsky
David Stanley Duch
Carl William Sigel
Charles Adam Nichol
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK254780A publication Critical patent/DK254780A/da
Publication of DK157451B publication Critical patent/DK157451B/da
Application granted granted Critical
Publication of DK157451C publication Critical patent/DK157451C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK254780A 1979-06-14 1980-06-13 Analogifremgangsmaade til fremstilling af 2,4-diamino-6-alkoxybenzyl-5-methylpyridooe2,3-daapyrimidiner eller farmaceutisk acceptable syreadditionssalte deraf DK157451C (da)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
GB7920705 1979-06-14
GB7920704 1979-06-14
GB7920703 1979-06-14
GB7920706 1979-06-14
GB7920704 1979-06-14
GB7920703 1979-06-14
GB7920706 1979-06-14
GB7920705 1979-06-14

Publications (3)

Publication Number Publication Date
DK254780A DK254780A (da) 1980-12-15
DK157451B DK157451B (da) 1990-01-08
DK157451C true DK157451C (da) 1990-05-21

Family

ID=27449125

Family Applications (1)

Application Number Title Priority Date Filing Date
DK254780A DK157451C (da) 1979-06-14 1980-06-13 Analogifremgangsmaade til fremstilling af 2,4-diamino-6-alkoxybenzyl-5-methylpyridooe2,3-daapyrimidiner eller farmaceutisk acceptable syreadditionssalte deraf

Country Status (12)

Country Link
EP (1) EP0021292B1 (da)
AU (1) AU532842B2 (da)
CA (1) CA1132137A (da)
DE (1) DE3062268D1 (da)
DK (1) DK157451C (da)
FI (1) FI66866C (da)
HU (1) HU184787B (da)
IE (1) IE49992B1 (da)
IL (1) IL60307A (da)
IT (1) IT1146940B (da)
MY (1) MY8500059A (da)
NZ (1) NZ194045A (da)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8702758D0 (en) * 1987-02-06 1987-03-11 Wellcome Found Treatment of disease
AU598093B2 (en) * 1987-02-07 1990-06-14 Wellcome Foundation Limited, The Pyridopyrimidines, methods for their preparation and pharmaceutical formulations thereof
US4889859A (en) * 1988-02-05 1989-12-26 The Trustees Of Princeton University Pyrido[2,3-d]pyrimidine derivatives
US5547954A (en) * 1994-05-26 1996-08-20 Fmc Corporation 2,4-Diamino-5,6-disubstituted-and 5,6,7-trisubstituted-5-deazapteridines as insecticides
US6498163B1 (en) 1997-02-05 2002-12-24 Warner-Lambert Company Pyrido[2,3-D]pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation
JP2001509805A (ja) * 1997-02-05 2001-07-24 ワーナー−ランバート・コンパニー 細胞増殖阻害剤としてのピリド〔2,3−d〕ピリミジンおよび4−アミノピリミジン
EP1806348A3 (en) * 1997-02-05 2008-01-02 Warner-Lambert Company LLC Pyrido [2, 3 -d] pyrimidines and 4-amino-primidines as inhibitors of cellular proliferation
BR9911590A (pt) * 1998-05-26 2001-02-13 Warner Lambert Co Pirimidinas bicìclicas e 3,4-diidropirimidinas bicìclicas como inibidores da proliferação celular
EP1801112A1 (en) * 1998-05-26 2007-06-27 Warner-Lambert Company LLC Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
EP1180369A4 (en) 1999-05-24 2002-07-24 Sankyo Co ANTI-FAS ANTIBODY MEDICAL COMPOSITIONS
KR20060111716A (ko) 2002-01-22 2006-10-27 워너-램버트 캄파니 엘엘씨 2-(피리딘-2-일아미노)-피리도[2,3-d]피리미딘-7-온

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2937284A (en) * 1958-05-01 1960-05-17 Burroughs Wellcome Co 2, 4-diamino-5, 6-dialkylpyrido (2, 3-d) pyrimidines and method
GB970583A (en) * 1961-07-19 1964-09-23 Wellcome Found 2,4-diaminopyrido[2,3-d]pyrimidines
US3322765A (en) * 1963-10-30 1967-05-30 Burroughs Wellcome Co 2, 4-diamino-6-benzylpyrido-(2, 3-d) pyrimidines and method

Also Published As

Publication number Publication date
DK157451B (da) 1990-01-08
FI801912A (fi) 1980-12-15
IL60307A0 (en) 1980-09-16
EP0021292B1 (en) 1983-03-09
FI66866C (fi) 1984-12-10
MY8500059A (en) 1985-12-31
IT8048968A0 (it) 1980-06-13
HU184787B (en) 1984-10-29
NZ194045A (en) 1984-09-28
IE801220L (en) 1980-12-14
DK254780A (da) 1980-12-15
IE49992B1 (en) 1986-01-22
CA1132137A (en) 1982-09-21
EP0021292A1 (en) 1981-01-07
IT1146940B (it) 1986-11-19
IL60307A (en) 1984-02-29
DE3062268D1 (en) 1983-04-14
AU5927580A (en) 1980-12-18
AU532842B2 (en) 1983-10-13
FI66866B (fi) 1984-08-31

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