IT1118098B - Analoghi delle tia diazotil cefalosporine particolarmente utili come antibatterici e procedimento per la loro preparazione - Google Patents

Analoghi delle tia diazotil cefalosporine particolarmente utili come antibatterici e procedimento per la loro preparazione

Info

Publication number
IT1118098B
IT1118098B IT68975/78A IT6897578A IT1118098B IT 1118098 B IT1118098 B IT 1118098B IT 68975/78 A IT68975/78 A IT 68975/78A IT 6897578 A IT6897578 A IT 6897578A IT 1118098 B IT1118098 B IT 1118098B
Authority
IT
Italy
Prior art keywords
diazotyl
antibacterials
cephalosporins
tia
analogues
Prior art date
Application number
IT68975/78A
Other languages
English (en)
Italian (it)
Other versions
IT7868975A0 (it
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of IT7868975A0 publication Critical patent/IT7868975A0/it
Application granted granted Critical
Publication of IT1118098B publication Critical patent/IT1118098B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D505/00Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IT68975/78A 1977-08-25 1978-08-24 Analoghi delle tia diazotil cefalosporine particolarmente utili come antibatterici e procedimento per la loro preparazione IT1118098B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP52102261A JPS609718B2 (ja) 1977-08-25 1977-08-25 チアジアゾリルチオセフアロスポリン類縁抗生物質

Publications (2)

Publication Number Publication Date
IT7868975A0 IT7868975A0 (it) 1978-08-24
IT1118098B true IT1118098B (it) 1986-02-24

Family

ID=14322642

Family Applications (1)

Application Number Title Priority Date Filing Date
IT68975/78A IT1118098B (it) 1977-08-25 1978-08-24 Analoghi delle tia diazotil cefalosporine particolarmente utili come antibatterici e procedimento per la loro preparazione

Country Status (34)

Country Link
US (1) US4201782A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS609718B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AR (1) AR220539A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) AT361121B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU517618B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE869955A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BG (1) BG34338A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1101417A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH637396A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CS (1) CS203927B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DD (1) DD137230A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE2837264A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK372878A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES472817A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI65432C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2401165A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1576796A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR70260B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HU177900B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE47630B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL55429A0 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1118098B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX5328E (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL190554C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO782866L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ188173A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PH (1) PH17508A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PL (1) PL110656B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT68434A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RO (1) RO75070A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE452010B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SU (1) SU812182A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
YU (1) YU43999B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA784753B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4259485A (en) * 1979-04-24 1981-03-31 Eli Lilly And Company Crystallization process
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
DE3373475D1 (en) * 1982-12-14 1987-10-15 Beecham Group Plc Process for the preparation of beta-lactam compounds
JPS60123490A (ja) * 1983-12-07 1985-07-02 Shionogi & Co Ltd マロニルオキサセフェムカルボン酸誘導体
US6013835A (en) * 1995-06-07 2000-01-11 Hfm International, Inc. Method and apparatus for preparing purified terephthalic acid
US6197794B1 (en) 1998-01-08 2001-03-06 Celltech Therapeutics Limited Phenylalanine derivatives
US6329372B1 (en) 1998-01-27 2001-12-11 Celltech Therapeutics Limited Phenylalanine derivatives
DE69919334T2 (de) 1998-02-26 2005-08-04 Celltech Therapeutics Ltd., Slough Phenylalaninderivate als inhibitoren von alpha4 integrinen
GB9805655D0 (en) 1998-03-16 1998-05-13 Celltech Therapeutics Ltd Chemical compounds
US6521626B1 (en) 1998-03-24 2003-02-18 Celltech R&D Limited Thiocarboxamide derivatives
GB9811159D0 (en) 1998-05-22 1998-07-22 Celltech Therapeutics Ltd Chemical compounds
GB9811969D0 (en) 1998-06-03 1998-07-29 Celltech Therapeutics Ltd Chemical compounds
GB9812088D0 (en) 1998-06-05 1998-08-05 Celltech Therapeutics Ltd Chemical compounds
GB9814414D0 (en) 1998-07-03 1998-09-02 Celltech Therapeutics Ltd Chemical compounds
GB9821061D0 (en) 1998-09-28 1998-11-18 Celltech Therapeutics Ltd Chemical compounds
GB9821222D0 (en) 1998-09-30 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9821406D0 (en) * 1998-10-01 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9825652D0 (en) 1998-11-23 1999-01-13 Celltech Therapeutics Ltd Chemical compounds
US6518283B1 (en) 1999-05-28 2003-02-11 Celltech R&D Limited Squaric acid derivatives
US6534513B1 (en) 1999-09-29 2003-03-18 Celltech R&D Limited Phenylalkanoic acid derivatives
US6455539B2 (en) 1999-12-23 2002-09-24 Celltech R&D Limited Squaric acid derivates
EP1332132B1 (en) 2000-04-17 2007-10-10 UCB Pharma, S.A. Enamine derivatives as cell adhesion molecules
US6403608B1 (en) 2000-05-30 2002-06-11 Celltech R&D, Ltd. 3-Substituted isoquinolin-1-yl derivatives
US6545013B2 (en) 2000-05-30 2003-04-08 Celltech R&D Limited 2,7-naphthyridine derivatives
US6740654B2 (en) 2000-07-07 2004-05-25 Celltech R & D Limited Squaric acid derivatives
US6649756B2 (en) * 2000-07-13 2003-11-18 Wyeth, Five Giralda Farms Process improvement in the preparation of (4r, 5s, 6s)-3-[[(2r,3r)-2-[[[(s)-2-amino-3-methyl-1-oxobutyl]amino]methyl]tetrahydro-3-furanyl]thio]-6-[(r)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
CA2417059A1 (en) 2000-08-02 2002-02-07 Celltech R&D Limited 3-substituted isoquinolin-1-yl derivatives
CN102827191B (zh) * 2012-09-24 2015-03-11 浙江东邦药业有限公司 一种氧头孢类化合物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL178005C (nl) * 1972-11-06 1986-01-02 Merck & Co Inc Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
US4031083A (en) * 1975-10-24 1977-06-21 Yeda Research And Development Co., Ltd. Cephalosporin antibiotics
US4045438A (en) * 1975-10-24 1977-08-30 Yeda Research And Development Co. Ltd. Cephalosporin antibiotics
FR2361114A1 (fr) * 1975-11-12 1978-03-10 Shionogi & Co Procede de preparation d'analogues de cephalosporine a propriete antibacterienne et nouveaux produits ainsi obtenus
CA1085392A (en) * 1976-03-25 1980-09-09 Masayuki Narisada Arylmalonamido-1-oxadethiacephalosporins

Also Published As

Publication number Publication date
DE2837264C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1991-06-13
CA1101417A (en) 1981-05-19
BE869955A (fr) 1978-12-18
DD137230A5 (de) 1979-08-22
JPS609718B2 (ja) 1985-03-12
DE2837264A1 (de) 1979-03-01
PT68434A (en) 1978-09-01
DK372878A (da) 1979-02-26
SU812182A3 (ru) 1981-03-07
HU177900B (en) 1982-01-28
FR2401165B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1982-06-25
AU3923878A (en) 1980-02-28
NO782866L (no) 1979-02-27
AT361121B (de) 1981-02-25
GB1576796A (en) 1980-10-15
CS203927B2 (en) 1981-03-31
AR220539A1 (es) 1980-11-14
RO75070A (ro) 1980-10-30
IE47630B1 (en) 1984-05-16
AU517618B2 (en) 1981-08-13
GR70260B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1982-09-02
CH637396A5 (de) 1983-07-29
YU43999B (en) 1990-02-28
SE7808950L (sv) 1979-02-26
NZ188173A (en) 1981-05-15
SE452010B (sv) 1987-11-09
FI782586A7 (fi) 1979-02-26
FR2401165A1 (fr) 1979-03-23
US4201782A (en) 1980-05-06
FI65432C (fi) 1984-05-10
ZA784753B (en) 1979-08-29
PH17508A (en) 1984-09-07
JPS5436288A (en) 1979-03-16
PL110656B1 (en) 1980-07-31
PL209215A1 (pl) 1979-06-04
ATA620378A (de) 1980-07-15
IT7868975A0 (it) 1978-08-24
IL55429A0 (en) 1978-10-31
YU202878A (en) 1982-10-31
BG34338A3 (bg) 1983-08-15
ES472817A1 (es) 1979-02-16
NL190554C (nl) 1994-04-18
FI65432B (fi) 1984-01-31
IE781703L (en) 1979-02-25
MX5328E (es) 1983-06-22
NL7808802A (nl) 1979-02-27
NL190554B (nl) 1993-11-16

Similar Documents

Publication Publication Date Title
IT1118098B (it) Analoghi delle tia diazotil cefalosporine particolarmente utili come antibatterici e procedimento per la loro preparazione
IT1108491B (it) Derivati di amminotiazoli particolarment utili come immunostimolanti e procedimento per la loro preparazione
IT1091037B (it) Particelle di percarbonato sodico e procedimento per la loro preparazione
IT1104127B (it) Feniletanolammine sostituite utili come componenti di farmaci e procedimento per la loro preparazione
IT1165618B (it) Particelle di percarbonato sodico e procedimento per la loro preparazione
IT1118095B (it) Derivati dell acido cicloalchiliden metilfenilacetico particolarmente utili come medicamenti e procedimento per la loro preparazione
IT1107226B (it) Procedimento per la preparazione di derivati alogeno metilici di acido gamma-amminobutirrico utili come agenti farmacologici e prodotto ottenuto
IT1129264B (it) Derivati di acido cicloesancarbossilico particolarmente utili come antiulcera e procedimento per la loro preparazione
IT7820957A0 (it) Derivati di acido 1-azaxantone-3-carbossilico eprocedimento per la loro preparazione.
IT1115153B (it) Analoghi di cefalosporina e procedimento per la loro preparazione
IT7969279A0 (it) 4 1 benzossazepine loro tia analoghi e procedimento per la loro preparazione
MX4950E (es) Procedimiento para la preparacion de tioesteres de acido clavulanico
MX5006E (es) Procedimiento para la preparacion de acido ciclohexancarboxilico
IT1192795B (it) Analoghi di cefalosporina e procedimento per la loro preparazione
IT7869726A0 (it) Derivati della tetraidroftalammide particolarmente utili come erbicidi e procedimento per la loro preparazione
IT1070073B (it) Composti di carbammato sulfenil carbammoil fluoruri particolarmente utili come insetticidi e procedimento per la loro preparazione
MX5207E (es) Procedimiento para la preparacion de 3-fenoxi-alfa-vinilbencilesteres de acido vinilciclopropancarboxilico
AR218294A1 (es) Procedimiento para la preparacion de derivados de acido oleanoico
IT1165187B (it) Analoghi di cefalosporina e procedimento per la loro preparazione
MX5206E (es) Procedimiento para la preparacion de fenoxi-alfa-vinil-bencil-esteres de acido ciclopropancarboxilico
IT7968397A0 (it) Derivati di cefalosporine partico larmente utili come microbicidi eprocedimento per la loro preparazione
IT1147712B (it) 3 4 di desossi canamicina a e suoi derivati particolarmente utili come antibatterici e procedimento per la loro preparazione
IT1119096B (it) Derivati della benzotiazocina e della benzotiazonina particolarmente utili come medicamenti e procedimento per la loro preparazione
IT7831061A0 (it) Composti analoghi della cefalosporina e procedimenti per la loro preparazione.
IT7967856A0 (it) Derivati delle ftalidil isochinoleine particolarmente utili come medicamenti e procedimento per la loro preparazione

Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19950831